MX2020006468A - Composiciones y metodos para el tratamiento o prevencion de sintomas vasomotores. - Google Patents
Composiciones y metodos para el tratamiento o prevencion de sintomas vasomotores.Info
- Publication number
- MX2020006468A MX2020006468A MX2020006468A MX2020006468A MX2020006468A MX 2020006468 A MX2020006468 A MX 2020006468A MX 2020006468 A MX2020006468 A MX 2020006468A MX 2020006468 A MX2020006468 A MX 2020006468A MX 2020006468 A MX2020006468 A MX 2020006468A
- Authority
- MX
- Mexico
- Prior art keywords
- compositions
- treating
- methods
- vasomotor symptoms
- preventing vasomotor
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente descripción está dirigida a composiciones que comprenden como un ingrediente activo, una dosis más baja de ácido 4-({(1-ciclopropilisoquinolin-3-il)[4- (trifluorometoxi)benc il]amino}sulfonil)benzoico o una sal farmacéuticamente aceptable del mismo para tratar o prevenir los síntomas vasomotores en un sujeto, y métodos que comprenden administrar dicho compuesto o la sal farmacéuticamente aceptable del mismo a una dosis más baja, respectivamente.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762607666P | 2017-12-19 | 2017-12-19 | |
| PCT/JP2018/046544 WO2019124366A1 (en) | 2017-12-19 | 2018-12-18 | Compositions and methods for treating or preventing vasomotor symptoms |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2020006468A true MX2020006468A (es) | 2021-01-08 |
Family
ID=65023968
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2020006468A MX2020006468A (es) | 2017-12-19 | 2018-12-18 | Composiciones y metodos para el tratamiento o prevencion de sintomas vasomotores. |
Country Status (16)
| Country | Link |
|---|---|
| US (3) | US11471452B2 (es) |
| EP (2) | EP3727383A1 (es) |
| JP (2) | JP7265551B2 (es) |
| KR (1) | KR20200100746A (es) |
| CN (1) | CN111465395A (es) |
| AR (1) | AR113963A1 (es) |
| AU (1) | AU2018391882A1 (es) |
| BR (1) | BR112020012111A2 (es) |
| CA (1) | CA3085292A1 (es) |
| CO (1) | CO2020007091A2 (es) |
| IL (1) | IL275258A (es) |
| MX (1) | MX2020006468A (es) |
| PH (1) | PH12020550932A1 (es) |
| SG (1) | SG11202005383RA (es) |
| TW (1) | TW201929855A (es) |
| WO (1) | WO2019124366A1 (es) |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR112013023330B8 (pt) | 2011-03-16 | 2022-09-27 | Mitsubishi Tanabe Pharma Corp | Compostos de sulfonamida tendo atividade antagonista trpm8 |
| BR112013033316A2 (pt) * | 2011-06-24 | 2017-01-31 | Amgen Inc | antagonista de trpm8 e seu uso em tratamentos |
| JP5985453B2 (ja) | 2012-09-14 | 2016-09-06 | 田辺三菱製薬株式会社 | 医薬組成物 |
| WO2014042238A1 (ja) | 2012-09-14 | 2014-03-20 | 田辺三菱製薬株式会社 | スルホンアミド化合物 |
| CA2959231C (en) | 2013-10-22 | 2022-06-21 | Edward Tak Wei | Di-isopropyl-phosphinoyl-alkane (dapa) compounds as topical agents for the treatment of sensory discomfort |
| ES2957232T3 (es) * | 2016-06-13 | 2024-01-15 | Mitsubishi Tanabe Pharma Corp | Composiciones para el tratamiento o la prevención de síntomas vasomotores |
-
2018
- 2018-12-18 WO PCT/JP2018/046544 patent/WO2019124366A1/en not_active Ceased
- 2018-12-18 AU AU2018391882A patent/AU2018391882A1/en not_active Abandoned
- 2018-12-18 KR KR1020207020762A patent/KR20200100746A/ko not_active Withdrawn
- 2018-12-18 AR ARP180103696A patent/AR113963A1/es not_active Application Discontinuation
- 2018-12-18 EP EP18834076.4A patent/EP3727383A1/en not_active Withdrawn
- 2018-12-18 EP EP22172496.6A patent/EP4059500A1/en not_active Withdrawn
- 2018-12-18 JP JP2020533860A patent/JP7265551B2/ja active Active
- 2018-12-18 CA CA3085292A patent/CA3085292A1/en active Pending
- 2018-12-18 US US15/733,253 patent/US11471452B2/en active Active
- 2018-12-18 CN CN201880081744.7A patent/CN111465395A/zh active Pending
- 2018-12-18 MX MX2020006468A patent/MX2020006468A/es unknown
- 2018-12-18 SG SG11202005383RA patent/SG11202005383RA/en unknown
- 2018-12-18 BR BR112020012111-8A patent/BR112020012111A2/pt unknown
- 2018-12-18 TW TW107145704A patent/TW201929855A/zh unknown
-
2020
- 2020-06-10 CO CONC2020/0007091A patent/CO2020007091A2/es unknown
- 2020-06-10 IL IL275258A patent/IL275258A/en unknown
- 2020-06-18 PH PH12020550932A patent/PH12020550932A1/en unknown
-
2022
- 2022-07-20 US US17/813,619 patent/US20220401434A1/en not_active Abandoned
-
2023
- 2023-04-14 JP JP2023066312A patent/JP2023089175A/ja not_active Withdrawn
-
2024
- 2024-09-04 US US18/824,168 patent/US20250057831A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| PH12020550932A1 (en) | 2021-05-10 |
| US20220401434A1 (en) | 2022-12-22 |
| IL275258A (en) | 2020-07-30 |
| JP7265551B2 (ja) | 2023-04-26 |
| KR20200100746A (ko) | 2020-08-26 |
| CO2020007091A2 (es) | 2020-06-19 |
| US11471452B2 (en) | 2022-10-18 |
| US20200383968A1 (en) | 2020-12-10 |
| AU2018391882A2 (en) | 2022-06-23 |
| WO2019124366A1 (en) | 2019-06-27 |
| EP3727383A1 (en) | 2020-10-28 |
| JP2021506881A (ja) | 2021-02-22 |
| TW201929855A (zh) | 2019-08-01 |
| US20250057831A1 (en) | 2025-02-20 |
| CA3085292A1 (en) | 2019-06-27 |
| JP2023089175A (ja) | 2023-06-27 |
| SG11202005383RA (en) | 2020-07-29 |
| AR113963A1 (es) | 2020-07-01 |
| BR112020012111A2 (pt) | 2020-11-24 |
| EP4059500A1 (en) | 2022-09-21 |
| CN111465395A (zh) | 2020-07-28 |
| AU2018391882A1 (en) | 2020-07-02 |
| RU2020123723A (ru) | 2022-01-20 |
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