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MX2019010098A - Antiandrogenos para el tratamiento del cancer de prostata resistente a la castracion no metastasico. - Google Patents

Antiandrogenos para el tratamiento del cancer de prostata resistente a la castracion no metastasico.

Info

Publication number
MX2019010098A
MX2019010098A MX2019010098A MX2019010098A MX2019010098A MX 2019010098 A MX2019010098 A MX 2019010098A MX 2019010098 A MX2019010098 A MX 2019010098A MX 2019010098 A MX2019010098 A MX 2019010098A MX 2019010098 A MX2019010098 A MX 2019010098A
Authority
MX
Mexico
Prior art keywords
antiandrogens
treatment
prostate cancer
castration
metastasic
Prior art date
Application number
MX2019010098A
Other languages
English (en)
Other versions
MX379847B (es
Inventor
Chen Isan
Original Assignee
Aragon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49293921&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2019010098(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aragon Pharmaceuticals Inc filed Critical Aragon Pharmaceuticals Inc
Publication of MX2019010098A publication Critical patent/MX2019010098A/es
Publication of MX379847B publication Critical patent/MX379847B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
    • A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/28—Antiandrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Reproductive Health (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicinal Preparation (AREA)

Abstract

En la presente invencion se describen antiandrogenos para usarse en el tratamiento de cancer de prostata resistente a la castracion no metastasico.
MX2019010098A 2012-09-26 2013-09-23 Antiandrogenos para el tratamiento del cancer de prostata resistente a la castracion no metastasico MX379847B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261705900P 2012-09-26 2012-09-26
PCT/US2013/061197 WO2014052237A1 (en) 2012-09-26 2013-09-23 Anti-androgens for the treatment of non-metastatic castrate-resistant prostate cancer

Publications (2)

Publication Number Publication Date
MX2019010098A true MX2019010098A (es) 2019-10-15
MX379847B MX379847B (es) 2025-03-11

Family

ID=49293921

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2019010098A MX379847B (es) 2012-09-26 2013-09-23 Antiandrogenos para el tratamiento del cancer de prostata resistente a la castracion no metastasico
MX2015003909A MX371020B (es) 2012-09-26 2013-09-23 Antiandrógenos para el tratamiento del cáncer de próstata resistente a la castración no metastásico.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2015003909A MX371020B (es) 2012-09-26 2013-09-23 Antiandrógenos para el tratamiento del cáncer de próstata resistente a la castración no metastásico.

Country Status (36)

Country Link
US (8) US9884054B2 (es)
EP (3) EP2900224A1 (es)
JP (4) JP6351597B2 (es)
KR (3) KR20210013342A (es)
CN (4) CN109908114A (es)
AU (4) AU2013323861C1 (es)
BR (1) BR112015006705A8 (es)
CA (1) CA2885415C (es)
CL (1) CL2015000715A1 (es)
CR (1) CR20150140A (es)
CY (1) CY1123716T1 (es)
DK (1) DK3305285T3 (es)
EA (3) EA037806B1 (es)
EC (1) ECSP15011764A (es)
ES (1) ES2836424T3 (es)
GT (1) GT201500071A (es)
HK (1) HK1212221A1 (es)
HR (1) HRP20201721T1 (es)
HU (1) HUE051211T2 (es)
IL (3) IL237692B2 (es)
IN (1) IN2015DN02387A (es)
LT (1) LT3305285T (es)
MX (2) MX379847B (es)
MY (1) MY180834A (es)
NI (1) NI201500042A (es)
NZ (3) NZ705815A (es)
PE (1) PE20150765A1 (es)
PH (3) PH12018502570B1 (es)
PT (1) PT3305285T (es)
RS (1) RS60976B1 (es)
SG (3) SG10201912719TA (es)
SI (1) SI3305285T1 (es)
SM (1) SMT202000573T1 (es)
UA (3) UA124967C2 (es)
WO (1) WO2014052237A1 (es)
ZA (1) ZA201808499B (es)

Families Citing this family (13)

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Publication number Priority date Publication date Assignee Title
LT3124481T (lt) 2010-02-16 2018-06-11 Aragon Pharmaceuticals, Inc. Androgeno receptorių moduliatoriai ir jų panaudojimas
AP2014007657A0 (en) 2011-12-16 2014-05-31 Olema Pharmaceuticals Inc Novel benzopyran compounds, compositions and uses thereof
AU2013323861C1 (en) 2012-09-26 2024-05-02 Aragon Pharmaceuticals, Inc. Anti-androgens for the treatment of non-metastatic castrate-resistant prostate cancer
JOP20200097A1 (ar) 2013-01-15 2017-06-16 Aragon Pharmaceuticals Inc معدل مستقبل أندروجين واستخداماته
TWI709403B (zh) 2014-12-05 2020-11-11 美商艾瑞岡醫藥公司 抗癌症組成物（二）
PL3226841T3 (pl) * 2014-12-05 2025-03-03 Aragon Pharmaceuticals, Inc. Kompozycje przeciwnowotworowe
KR102348325B1 (ko) * 2014-12-05 2022-01-06 아라곤 파마슈티컬스, 인코포레이티드 항암 조성물
KR101718226B1 (ko) 2015-08-05 2017-03-20 울산대학교 산학협력단 사쿠라소사포닌 화합물을 유효성분으로 포함하는 안드로겐 수용체 관련 질환의 예방 또는 치료용 조성물
TWI726969B (zh) 2016-01-11 2021-05-11 比利時商健生藥品公司 用作雄性激素受體拮抗劑之經取代之硫尿囊素衍生物
FI3490560T3 (fi) * 2016-07-29 2025-02-27 Janssen Pharmaceutica Nv Niraparibi käytettäväksi eturauhassyövän hoitomenetelmässä
CN111479560A (zh) * 2017-10-16 2020-07-31 阿拉贡药品公司 用于治疗非转移性去势难治性前列腺癌的抗雄激素
AU2020215176B2 (en) * 2019-01-30 2025-02-27 Aragon Pharmaceuticals, Inc. Anti-androgens for the treatment of metastatic castration-sensitive prostate cancer
CA3160121A1 (en) * 2019-11-04 2021-05-14 Aragon Pharmaceuticals, Inc. Androgen receptor inhibitors for the treatment of non-metastatic castration-resistant prostate cancer in subjects with severe hepatic impairment

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