MX2019001007A - Uso novedoso de nectinib y una sal farmaceuticamente aceptable del mismo en el tratamiento contra enfermedades. - Google Patents
Uso novedoso de nectinib y una sal farmaceuticamente aceptable del mismo en el tratamiento contra enfermedades.Info
- Publication number
- MX2019001007A MX2019001007A MX2019001007A MX2019001007A MX2019001007A MX 2019001007 A MX2019001007 A MX 2019001007A MX 2019001007 A MX2019001007 A MX 2019001007A MX 2019001007 A MX2019001007 A MX 2019001007A MX 2019001007 A MX2019001007 A MX 2019001007A
- Authority
- MX
- Mexico
- Prior art keywords
- pharmaceutically acceptable
- gzd824
- acceptable salts
- treating diseases
- novel application
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención describe el uso de (3-((1H-pirazol[3,4-b]pir idin-5-sustituida)etinil)-4-metil-N-(4-((4-metilpiperazin-1-susti tuida)metil)-3-(trifluorometil)fenil)benzamida) y una sal farmacéuticamente aceptable de la misma en la elaboración de un medicamento para el tratamiento contra la leucemia linfoblástica aguda, en particular, la leucemia linfoblástica de linfocitos B precursores.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201610592371 | 2016-07-25 | ||
| CN201611040298.4A CN106580993B (zh) | 2016-07-25 | 2016-11-11 | 耐克替尼及其药学上可接受的盐在治疗疾病中的新的应用 |
| PCT/CN2017/081173 WO2018018950A1 (zh) | 2016-07-25 | 2017-04-20 | 耐克替尼及其药学上可接受的盐在治疗疾病中的新的应用 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2019001007A true MX2019001007A (es) | 2019-06-10 |
Family
ID=58592880
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2019001007A MX2019001007A (es) | 2016-07-25 | 2017-04-20 | Uso novedoso de nectinib y una sal farmaceuticamente aceptable del mismo en el tratamiento contra enfermedades. |
Country Status (10)
| Country | Link |
|---|---|
| US (3) | US20200330456A1 (es) |
| EP (1) | EP3488850B1 (es) |
| JP (1) | JP6724240B2 (es) |
| KR (1) | KR20190032425A (es) |
| CN (1) | CN106580993B (es) |
| AU (1) | AU2017303624A1 (es) |
| CA (1) | CA3031852A1 (es) |
| IL (1) | IL264407A (es) |
| MX (1) | MX2019001007A (es) |
| WO (1) | WO2018018950A1 (es) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN111035641B (zh) * | 2018-10-11 | 2022-04-12 | 暨南大学 | Gzd824及其药学上可接受的盐在治疗疾病中的新应用 |
| DK3713576T3 (da) * | 2018-12-03 | 2025-08-18 | Ascentage Pharma Suzhou Co Ltd | Forbindelse med formel (i) og ponatinib til brug ved behandling af kronisk myeloid leukæmi med bcr-abl-mutationer |
| CN110917157B (zh) * | 2020-01-21 | 2020-06-16 | 上海亚盛医药科技有限公司 | 含炔基化合物的药物组合物、其制备方法及应用 |
| US20230078120A1 (en) * | 2020-05-04 | 2023-03-16 | Ascentage Pharma (Suzhou) Co.,Ltd. | Methods for Treating Coronavirus Infections |
| WO2022105836A1 (en) * | 2020-11-19 | 2022-05-27 | Guangzhou Healthquest Pharma Co., Ltd. | Combination therapies for treating cancer |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101885722B (zh) * | 2010-07-01 | 2013-07-24 | 中国科学院广州生物医药与健康研究院 | 杂环炔苯类化合物及其药用组合物和应用 |
| US8846671B2 (en) * | 2010-07-01 | 2014-09-30 | Guangzhou Institute Of Biomedicine And Health, Chinese Academy Of Sciences | Heterocyclic alkynyl benzene compounds and medical compositions and uses thereof |
| CN103539784B (zh) * | 2012-07-09 | 2016-08-17 | 中国科学院广州生物医药与健康研究院 | 杂环苯甲酰胺类化合物、药用组合物及其应用 |
-
2016
- 2016-11-11 CN CN201611040298.4A patent/CN106580993B/zh active Active
-
2017
- 2017-04-20 KR KR1020197004252A patent/KR20190032425A/ko not_active Withdrawn
- 2017-04-20 AU AU2017303624A patent/AU2017303624A1/en not_active Abandoned
- 2017-04-20 JP JP2019503742A patent/JP6724240B2/ja active Active
- 2017-04-20 US US16/318,729 patent/US20200330456A1/en not_active Abandoned
- 2017-04-20 MX MX2019001007A patent/MX2019001007A/es unknown
- 2017-04-20 EP EP17833256.5A patent/EP3488850B1/en active Active
- 2017-04-20 WO PCT/CN2017/081173 patent/WO2018018950A1/zh not_active Ceased
- 2017-04-20 CA CA3031852A patent/CA3031852A1/en not_active Abandoned
-
2019
- 2019-01-22 IL IL264407A patent/IL264407A/en unknown
-
2021
- 2021-04-12 US US17/227,841 patent/US20210228573A1/en not_active Abandoned
-
2024
- 2024-12-12 US US18/978,741 patent/US20250170125A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| CA3031852A1 (en) | 2018-02-01 |
| WO2018018950A1 (zh) | 2018-02-01 |
| US20250170125A1 (en) | 2025-05-29 |
| AU2017303624A1 (en) | 2019-02-14 |
| CN106580993A (zh) | 2017-04-26 |
| EP3488850A1 (en) | 2019-05-29 |
| US20200330456A1 (en) | 2020-10-22 |
| JP6724240B2 (ja) | 2020-07-15 |
| JP2019522019A (ja) | 2019-08-08 |
| EP3488850A4 (en) | 2020-08-26 |
| EP3488850B1 (en) | 2024-06-19 |
| CN106580993B (zh) | 2018-11-30 |
| KR20190032425A (ko) | 2019-03-27 |
| US20210228573A1 (en) | 2021-07-29 |
| IL264407A (en) | 2019-02-28 |
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