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MX2019000047A - Inhibidores peptídicos de la acumulación de alfa-sinucleína basados en estructuras. - Google Patents

Inhibidores peptídicos de la acumulación de alfa-sinucleína basados en estructuras.

Info

Publication number
MX2019000047A
MX2019000047A MX2019000047A MX2019000047A MX2019000047A MX 2019000047 A MX2019000047 A MX 2019000047A MX 2019000047 A MX2019000047 A MX 2019000047A MX 2019000047 A MX2019000047 A MX 2019000047A MX 2019000047 A MX2019000047 A MX 2019000047A
Authority
MX
Mexico
Prior art keywords
synuclein
alpha
peptide inhibitors
based peptide
synuclein aggregation
Prior art date
Application number
MX2019000047A
Other languages
English (en)
Inventor
S Eisenberg David
Smriti Sangwan
Jiang Lin
Original Assignee
Univ California
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ California filed Critical Univ California
Publication of MX2019000047A publication Critical patent/MX2019000047A/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/08Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/10Peptides having 12 to 20 amino acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02Linear peptides containing at least one abnormal peptide link
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • C07K14/4701Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
    • C07K14/4711Alzheimer's disease; Amyloid plaque core protein
    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N33/00Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
    • G01N33/48Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
    • G01N33/68Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving proteins, peptides or amino acids
    • G01N33/6893Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving proteins, peptides or amino acids related to diseases not provided for elsewhere
    • G01N33/6896Neurological disorders, e.g. Alzheimer's disease
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2319/00Fusion polypeptide
    • C07K2319/01Fusion polypeptide containing a localisation/targetting motif
    • C07K2319/10Fusion polypeptide containing a localisation/targetting motif containing a tag for extracellular membrane crossing, e.g. TAT or VP22
    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N2800/00Detection or diagnosis of diseases
    • G01N2800/28Neurological disorders
    • G01N2800/2835Movement disorders, e.g. Parkinson, Huntington, Tourette

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Neurology (AREA)
  • Biochemistry (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Microbiology (AREA)
  • Pathology (AREA)
  • General Physics & Mathematics (AREA)
  • Analytical Chemistry (AREA)
  • Physics & Mathematics (AREA)
  • Food Science & Technology (AREA)
  • Cell Biology (AREA)
  • Biotechnology (AREA)
  • Psychology (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)

Abstract

La presente invención se relaciona con péptidos inhibidores que se unen a moléculas de a-sinucleína y que inhiben la acumulación amiloidogénica de a-sinucleína, la citotoxicidad de a-sinucleína y la propagación de la a-sinucleína. Se describen métodos para fabricar y usar los péptidos inhibidores (por ejemplo, para tratar sujetos con afecciones o enfermedades que se encuentran mediadas por a-sinucleína, tal como enfermedad de Parkinson, demencia con cuerpos de Lewy o AMS).
MX2019000047A 2016-06-29 2017-06-29 Inhibidores peptídicos de la acumulación de alfa-sinucleína basados en estructuras. MX2019000047A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662356410P 2016-06-29 2016-06-29
PCT/US2017/040106 WO2018005867A2 (en) 2016-06-29 2017-06-29 Structure-based peptide inhibitors of alpha-synuclein aggregation

Publications (1)

Publication Number Publication Date
MX2019000047A true MX2019000047A (es) 2019-07-04

Family

ID=60786477

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2019000047A MX2019000047A (es) 2016-06-29 2017-06-29 Inhibidores peptídicos de la acumulación de alfa-sinucleína basados en estructuras.
MX2023009652A MX2023009652A (es) 2016-06-29 2019-01-07 Inhibidores peptidicos de la acumulacion de alfa-sinucleina basados en estructuras.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2023009652A MX2023009652A (es) 2016-06-29 2019-01-07 Inhibidores peptidicos de la acumulacion de alfa-sinucleina basados en estructuras.

Country Status (10)

Country Link
US (3) US10815271B2 (es)
EP (1) EP3478311A4 (es)
JP (3) JP6968839B2 (es)
KR (2) KR20230109776A (es)
CN (2) CN109641028A (es)
CA (1) CA3029676A1 (es)
IL (1) IL263913B2 (es)
MX (2) MX2019000047A (es)
RU (1) RU2766711C2 (es)
WO (1) WO2018005867A2 (es)

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US10563681B2 (en) 2011-12-21 2020-02-18 Deka Products Limited Partnership System, method, and apparatus for clamping
CN109641028A (zh) * 2016-06-29 2019-04-16 加利福尼亚大学董事会 α-突触核蛋白聚集的基于结构的肽抑制剂
EP3596102B1 (en) 2017-03-15 2025-09-10 The Regents of the University of California Structure-based peptide inhibitors that target the tau vqiink fibrillization segment
EP4149505A1 (en) 2020-05-15 2023-03-22 Vib Vzw Means and methods for the treatment of pathological aggregation
EP3943947A1 (en) * 2020-07-22 2022-01-26 Universitat Autònoma de Barcelona Inhibitors of alpha-synuclein aggregation and uses thereof
CN116457466A (zh) * 2020-09-23 2023-07-18 西洛斯治疗有限公司 用于抑制α-突触核蛋白聚集的组合物和方法
CA3207656A1 (en) * 2021-02-08 2022-08-11 University Of British Columbia Anti-synucleinopathy peptide and methods to treat neurodegenerative diseases
EP4071165A1 (en) 2021-04-05 2022-10-12 Consejo Superior de Investigaciones Científicas (CSIC) A new non-aggregative splicing isoform of human tau is decreased in alzheimer s disease
US20240238366A1 (en) * 2021-05-11 2024-07-18 O-Force Co., Ltd. alpha-SYNUCLEIN AGGREGATION INHIBITOR, PHARMACEUTICAL COMPOSITION FOR alpha-SYNUCLEIN DISEASE, AND USE THEREOF
CN114645052B (zh) * 2021-07-01 2023-05-26 中国医学科学院医学生物学研究所 一种全脑过表达核易位人源α-突触核蛋白转基因鼠的高效构建方法
KR102793149B1 (ko) * 2021-11-24 2025-04-09 주식회사 윙스타바이오 아밀로이드 전구체 단백질에 대한 저해 활성을 갖는 펩타이드 및 이의 용도
EP4186918A1 (en) 2021-11-30 2023-05-31 Université de Rennes Inhibitory peptides for the diagnostic and/or treatment of tauopathies
WO2023108290A1 (en) * 2021-12-15 2023-06-22 The Governing Council Of The University Of Toronto Peptide inhibitors and methods for inhibiting protein aggregation in neurons and neurodegenerative diseases
KR20230131017A (ko) * 2022-03-04 2023-09-12 삼성전자주식회사 가속기에 대해 온-디멘드 체크포인트를 수행하는 전자 장치 및 그 동작 방법
DE102022105391A1 (de) 2022-03-08 2023-09-14 Forschungszentrum Jülich GmbH Entwicklung eines α-Synuclein Amyloidtracers
WO2023181070A1 (en) * 2022-03-23 2023-09-28 Council Of Scientific & Industrial Research PEPTIDE TO TREAT α-SYNUCLEIN AMYLOID BASED DISORDERS
US11932594B1 (en) 2023-10-31 2024-03-19 King Faisal University 8-((2-hydroxy-5-methylphenyl)diazenyl)naphthalene-1,3-disulfonic acid as an antioxidant compound
KR20250085855A (ko) 2023-12-04 2025-06-13 성균관대학교산학협력단 퇴행성 신경 질환 가속 전파 모델 및 이의 제조방법

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AU7186501A (en) * 2000-07-07 2002-01-21 Panacea Pharmaceuticals Inc Methods for preventing neural tissue damage and for the treatment of alpha-synuclein diseases
GB0216972D0 (en) * 2002-07-22 2002-08-28 Univ Lancaster Peptides and peptide derivaties for the treatment of &-synuclein-related diseases
US20070213253A1 (en) * 2003-06-22 2007-09-13 Koji Sode Synuclein Mutant Having Aggregation-Inhibitory Activity
JP2009542611A (ja) * 2006-07-03 2009-12-03 ザパロイド・リミテッド アルファ−シヌクレイン凝集の阻害
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Also Published As

Publication number Publication date
US20210002329A1 (en) 2021-01-07
CN116650617A (zh) 2023-08-29
US20190241613A1 (en) 2019-08-08
IL263913A (en) 2019-01-31
JP2023162287A (ja) 2023-11-08
EP3478311A4 (en) 2021-01-06
IL263913B1 (en) 2024-09-01
KR20190034214A (ko) 2019-04-01
KR102554448B1 (ko) 2023-07-11
RU2766711C2 (ru) 2022-03-15
WO2018005867A3 (en) 2018-02-01
US10815271B2 (en) 2020-10-27
KR20230109776A (ko) 2023-07-20
JP6968839B2 (ja) 2021-11-17
WO2018005867A2 (en) 2018-01-04
CA3029676A1 (en) 2018-01-04
JP2022025103A (ja) 2022-02-09
RU2019102202A3 (es) 2020-10-30
RU2019102202A (ru) 2020-07-29
US20230069905A1 (en) 2023-03-09
IL263913B2 (en) 2025-01-01
MX2023009652A (es) 2023-08-24
EP3478311A2 (en) 2019-05-08
CN109641028A (zh) 2019-04-16
JP7337132B2 (ja) 2023-09-01
US11390646B2 (en) 2022-07-19
JP2019524685A (ja) 2019-09-05

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