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MX2018003962A - Proceso para producir fosfinatos. - Google Patents

Proceso para producir fosfinatos.

Info

Publication number
MX2018003962A
MX2018003962A MX2018003962A MX2018003962A MX2018003962A MX 2018003962 A MX2018003962 A MX 2018003962A MX 2018003962 A MX2018003962 A MX 2018003962A MX 2018003962 A MX2018003962 A MX 2018003962A MX 2018003962 A MX2018003962 A MX 2018003962A
Authority
MX
Mexico
Prior art keywords
phosphinates
producing
produce
pharmaceutical
amino acids
Prior art date
Application number
MX2018003962A
Other languages
English (en)
Other versions
MX377470B (es
Inventor
Joachim RESSEL Hans-
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of MX2018003962A publication Critical patent/MX2018003962A/es
Publication of MX377470B publication Critical patent/MX377470B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/48—Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof
    • C07F9/4866—Phosphonous acids [RP(OH)2] including [RHP(=O)(OH)]; Thiophosphonous acids including [RP(SH)2], [RHP(=S)(SH)]; Derivatives thereof the ester moiety containing a substituent or structure which is considered as characteristic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
    • C07F9/32—Esters thereof
    • C07F9/3205—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/3211—Esters of acyclic saturated acids which can have further substituents on alkyl
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N57/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds
    • A01N57/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic phosphorus compounds having alternatively specified atoms bound to the phosphorus atom and not covered by a single one of groups A01N57/10, A01N57/18, A01N57/26, A01N57/34
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J27/00—Catalysts comprising the elements or compounds of halogens, sulfur, selenium, tellurium, phosphorus or nitrogen; Catalysts comprising carbon compounds
    • B01J27/14—Phosphorus; Compounds thereof
    • B01J27/16—Phosphorus; Compounds thereof containing oxygen, i.e. acids, anhydrides and their derivates with N, S, B or halogens without carriers or on carriers based on C, Si, Al or Zr; also salts of Si, Al and Zr
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
    • C07F9/301—Acyclic saturated acids which can have further substituents on alkyl
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
    • C07F9/32—Esters thereof
    • C07F9/3205—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/3223—Esters of cycloaliphatic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4071—Esters thereof the ester moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4075—Esters with hydroxyalkyl compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Medicinal Chemistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Materials Engineering (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)

Abstract

La presente invención se refiere, principalmente, a un proceso para producir fosfinatos particulares (monoésteres del ácido fosfonoso) y a la utilización de los mismos para producir sustancias biológicamente activas las cuales se pueden utilizar en el sector farmacéutico o agroquímico, preferentemente para producir aminoácidos que contienen fósforo.
MX2018003962A 2015-09-29 2016-09-26 Proceso para producir fosfinatos. MX377470B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP15187469 2015-09-29
PCT/EP2016/072786 WO2017055193A1 (de) 2015-09-29 2016-09-26 Verfahren zur Herstellung von Phosphinaten

Publications (2)

Publication Number Publication Date
MX2018003962A true MX2018003962A (es) 2018-06-08
MX377470B MX377470B (es) 2025-03-10

Family

ID=54252056

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2018003962A MX377470B (es) 2015-09-29 2016-09-26 Proceso para producir fosfinatos.

Country Status (11)

Country Link
US (2) US10501485B2 (es)
EP (1) EP3356376B1 (es)
JP (1) JP6826110B2 (es)
KR (1) KR20180059466A (es)
CN (1) CN108137629B (es)
BR (1) BR112018006414B1 (es)
ES (1) ES2754603T3 (es)
IL (1) IL258301A (es)
MX (1) MX377470B (es)
TW (1) TWI721019B (es)
WO (1) WO2017055193A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201840578A (zh) * 2017-02-22 2018-11-16 以色列商亞當阿甘公司 製備甲基膦酸丁基酯的方法
CN110386950A (zh) * 2019-07-18 2019-10-29 石家庄瑞凯化工有限公司 一种草铵膦铵盐的合成方法
CN111909199B (zh) * 2020-08-06 2021-09-14 浙江新安化工集团股份有限公司 一种甲基亚膦酸二乙酯精馏高沸物资源化利用的方法
CN115109086B (zh) * 2021-03-23 2024-08-16 利尔化学股份有限公司 制备烷基膦酸酯的方法
CN116621873A (zh) * 2023-05-25 2023-08-22 福华通达化学股份公司 一种制备甲基乙基次膦酸乙酯以及甲基乙基次膦酸铝盐的方法

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3914345A (en) 1971-01-08 1975-10-21 Hoechst Ag Process for the manufacture of dialkyl-phosphinic acid esters
DE2415757C2 (de) 1974-04-01 1982-10-14 Hoechst Ag, 6000 Frankfurt Verfahren zur Herstellung phosphorhaltiger Ester
DE2519192C2 (de) 1975-04-30 1983-08-04 Hoechst Ag, 6230 Frankfurt Verfahren zur Herstellung phosphorhaltiger Ester
DE2717440C2 (de) * 1976-05-17 1984-04-05 Hoechst Ag, 6230 Frankfurt Unkrautbekämpfung mit [(3-Amino-3-carboxy)-propyl-1]-methylphosphinsäure-Derivaten
DE2849003A1 (de) * 1978-11-11 1980-08-21 Hoechst Ag Phosphorhaltige cyanhydrinderivate und verfahren zu ihrer herstellung
JPS56161310A (en) * 1980-05-16 1981-12-11 Sumitomo Chem Co Ltd Soil disinfectant
ATE22692T1 (de) * 1981-08-03 1986-10-15 Squibb & Sons Inc Phosphonamidate verbindungen.
DE3146196A1 (de) 1981-11-21 1983-05-26 Hoechst Ag, 6230 Frankfurt Verfahren zur herstellung phosphoniger saeuren
DE3146197A1 (de) 1981-11-21 1983-05-26 Hoechst Ag, 6230 Frankfurt Verfahren zur herstellung von phosphonigsaeuremonoalkylestern
JPS58188889A (ja) * 1982-04-26 1983-11-04 Sumitomo Chem Co Ltd α−ヒドロキシエチルホスフイン酸エステル、その製造法およびそれを有効成分とする植物病害防除剤
DE3319850C2 (de) * 1983-06-01 1985-05-09 Hoechst Ag, 6230 Frankfurt Verfahren zur Herstellung von phosphorhaltigen Cyanhydrinderivaten
US5166385A (en) 1989-03-23 1992-11-24 Hoechst Aktiengesellschaft Process for the preparation of phosphino compounds
DE3911230A1 (de) 1989-04-07 1990-10-11 Hoechst Ag Verfahren zur herstellung von alkylphosphonigsaeurediestern und/oder dialkylphosphinigsaeureestern
DE19736125A1 (de) 1997-08-20 1999-02-25 Hoechst Schering Agrevo Gmbh Verfahren zur Herstellung von Glufosinate und phosphorhaltige alpha-Aminonitrile als Zwischenprodukte
US20080146524A1 (en) * 2006-12-14 2008-06-19 Solvay Pharmaceuticals B.V. Selective inhibitors of neurotensin degrading enzymes
CN104892670A (zh) * 2015-05-13 2015-09-09 安徽国星生物化学有限公司 一种草铵膦及其类似物的制备方法

Also Published As

Publication number Publication date
CN108137629B (zh) 2020-09-01
US20200079804A1 (en) 2020-03-12
BR112018006414A2 (pt) 2018-10-09
JP2018534260A (ja) 2018-11-22
EP3356376B1 (de) 2019-08-07
MX377470B (es) 2025-03-10
TWI721019B (zh) 2021-03-11
CN108137629A (zh) 2018-06-08
KR20180059466A (ko) 2018-06-04
US20180265529A1 (en) 2018-09-20
US10501485B2 (en) 2019-12-10
ES2754603T3 (es) 2020-04-20
EP3356376A1 (de) 2018-08-08
BR112018006414B1 (pt) 2020-11-24
WO2017055193A1 (de) 2017-04-06
US10968241B2 (en) 2021-04-06
IL258301A (en) 2018-05-31
TW201726694A (zh) 2017-08-01
JP6826110B2 (ja) 2021-02-03

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