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MX2016016399A - Proceso para la preparacion de 3,5-bis(haloalquil)pirazoles por medio de la acilacion de cetiminas. - Google Patents

Proceso para la preparacion de 3,5-bis(haloalquil)pirazoles por medio de la acilacion de cetiminas.

Info

Publication number
MX2016016399A
MX2016016399A MX2016016399A MX2016016399A MX2016016399A MX 2016016399 A MX2016016399 A MX 2016016399A MX 2016016399 A MX2016016399 A MX 2016016399A MX 2016016399 A MX2016016399 A MX 2016016399A MX 2016016399 A MX2016016399 A MX 2016016399A
Authority
MX
Mexico
Prior art keywords
ketimines
haloalkyl
bis
preparing
via acylation
Prior art date
Application number
MX2016016399A
Other languages
English (en)
Other versions
MX383114B (es
Inventor
Lui Norbert
Pazenok Sergii
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of MX2016016399A publication Critical patent/MX2016016399A/es
Publication of MX383114B publication Critical patent/MX383114B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención se refiere a un novedoso proceso para la preparación de derivados de 3,4-bis(haloalquil)pirazoles a través de la acilación de cetiminas.
MX2016016399A 2014-06-11 2015-06-08 Proceso para la preparación de 3,5-bis(haloalquil)pirazoles por medio de la acilación de cetiminas. MX383114B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP14172036 2014-06-11
PCT/EP2015/062685 WO2015189138A1 (en) 2014-06-11 2015-06-08 Process for preparing 3,5-bis(haloalkyl)pyrazoles via acylation of ketimines

Publications (2)

Publication Number Publication Date
MX2016016399A true MX2016016399A (es) 2017-04-06
MX383114B MX383114B (es) 2025-03-13

Family

ID=50896204

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016016399A MX383114B (es) 2014-06-11 2015-06-08 Proceso para la preparación de 3,5-bis(haloalquil)pirazoles por medio de la acilación de cetiminas.

Country Status (12)

Country Link
US (1) US9914704B2 (es)
EP (1) EP3154947B1 (es)
JP (1) JP6514722B2 (es)
KR (1) KR102430607B1 (es)
CN (1) CN106458918B (es)
BR (1) BR112016028700B1 (es)
DK (1) DK3154947T3 (es)
ES (1) ES2672581T3 (es)
IL (1) IL249282B (es)
MX (1) MX383114B (es)
TW (1) TWI669292B (es)
WO (1) WO2015189138A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20180021798A (ko) * 2015-06-26 2018-03-05 바이엘 크롭사이언스 악티엔게젤샤프트 α,α-디할로알킬아민 및 케트이민으로부터 할로알콕시- 및 할로알킬티오 그룹을 가지는 치환된 피라졸의 제조방법
KR102477317B1 (ko) * 2016-09-21 2022-12-13 바이엘 크롭사이언스 악티엔게젤샤프트 3-플루오로알킬-5-피라졸카복실레이트 및 3-플루오로알킬-5-피라졸카복실산의 제조방법

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4950790A (en) * 1988-11-14 1990-08-21 Air Products And Chemicals, Inc. Volatile fluorinated β-ketoimines and associated metal complexes
BR0014078A (pt) * 1999-09-17 2002-12-31 Millennium Pharm Inc Inibidores de fator xa
DE10161978A1 (de) * 2001-12-17 2003-06-26 Bayer Ag Verfahren zur Herstellung von 2-Halogenacyl-3-amino-acrylsäure-derivate
DE10215292A1 (de) * 2002-02-19 2003-08-28 Bayer Cropscience Ag Disubstitutierte Pyrazolylcarbocanilide
DE10349500A1 (de) 2003-10-23 2005-06-02 Bayer Cropscience Ag Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern
WO2008013622A2 (en) * 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
DE102006039909A1 (de) 2006-08-25 2008-03-13 Bayer Cropscience Ag Verfahren zum Herstellen von 3-Dihalomethyl-pyrazol-4-carbonsäurederivaten
NZ579248A (en) * 2007-03-28 2011-08-26 Neurosearch As Purinyl derivatives and their use as potassium channel modulators
EP2133341A1 (de) 2008-02-25 2009-12-16 Bayer CropScience AG Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4-carbonsäure-Derivaten
EP2100883A1 (de) 2008-03-10 2009-09-16 Bayer CropScience AG Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4carbonsäure-Derivaten
PE20091653A1 (es) * 2008-03-26 2009-11-14 Takeda Pharmaceutical Derivados sustituidos de pirazol y su uso
US8759527B2 (en) 2010-08-25 2014-06-24 Bayer Cropscience Ag Heteroarylpiperidine and -piperazine derivatives as fungicides
BR112014001880A2 (pt) * 2011-07-26 2017-02-21 Gruenenthal Gmbh derivados de carboxamida e ureia contendo pirazol heteroaromáticos substituídos como ligantes de receptor vaniloide
EP2623496A1 (de) * 2012-02-01 2013-08-07 Bayer CropScience AG Verfahren zur Herstellung von 3,5-bis (fluoralkyl)-pyrazol-4-carbonsäure-Derivaten und 3,5-bis(fluoralkyl)-pyrazolen
WO2014023667A1 (en) * 2012-08-07 2014-02-13 Bayer Cropscience Ag Method for the preparation of perfluoroalkyl containing pyrazoles carboxylates
ES2588386T3 (es) * 2012-08-30 2016-11-02 Bayer Cropscience Ag Procedimiento de descarboxilación de derivados de ácido 3,5-bis(haloalquil)-pirazol-4-carboxílico

Also Published As

Publication number Publication date
KR102430607B1 (ko) 2022-08-08
US9914704B2 (en) 2018-03-13
IL249282B (en) 2019-03-31
WO2015189138A1 (en) 2015-12-17
DK3154947T3 (en) 2018-06-18
KR20170018885A (ko) 2017-02-20
JP2017517530A (ja) 2017-06-29
US20170114020A1 (en) 2017-04-27
TWI669292B (zh) 2019-08-21
MX383114B (es) 2025-03-13
EP3154947B1 (en) 2018-03-28
IL249282A0 (en) 2017-02-28
BR112016028700B1 (pt) 2021-03-23
TW201613869A (en) 2016-04-16
CN106458918B (zh) 2019-07-09
BR112016028700A2 (pt) 2017-08-22
EP3154947A1 (en) 2017-04-19
ES2672581T3 (es) 2018-06-15
CN106458918A (zh) 2017-02-22
JP6514722B2 (ja) 2019-05-15

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