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MX2016010871A - Regimen de dosificacion del compuesto de factor de crecimiento de fibroblastos 18. - Google Patents

Regimen de dosificacion del compuesto de factor de crecimiento de fibroblastos 18.

Info

Publication number
MX2016010871A
MX2016010871A MX2016010871A MX2016010871A MX2016010871A MX 2016010871 A MX2016010871 A MX 2016010871A MX 2016010871 A MX2016010871 A MX 2016010871A MX 2016010871 A MX2016010871 A MX 2016010871A MX 2016010871 A MX2016010871 A MX 2016010871A
Authority
MX
Mexico
Prior art keywords
dosing regimen
fgf
weeks
compound dosing
new dosing
Prior art date
Application number
MX2016010871A
Other languages
English (en)
Inventor
Christoph H Ladel
Guehring Hans
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of MX2016010871A publication Critical patent/MX2016010871A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/18Growth factors; Growth regulators
    • A61K38/1825Fibroblast growth factor [FGF]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/475Growth factors; Growth regulators
    • C07K14/50Fibroblast growth factor [FGF]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/18Growth factors; Growth regulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/19Cytokines; Lymphokines; Interferons
    • A61K38/20Interleukins [IL]
    • A61K38/2006IL-1
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/04Drugs for skeletal disorders for non-specific disorders of the connective tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Organic Chemistry (AREA)
  • Zoology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención proporciona un nuevo régimen de dosificación para la administración de FGF18 en el tratamiento de un trastorno del cartílago tal como, por ejemplo, la osteoartritis o la lesión del cartílago; se proporciona específicamente un plan de tratamiento preferido que comprende administraciones cada 3 semanas o cada 5 semanas de un compuesto de FGF-18 por ciclo de tratamiento; el nuevo régimen de dosificación puede incluir la co-administración de un fármaco anti-inflamatorio.
MX2016010871A 2014-02-20 2015-02-20 Regimen de dosificacion del compuesto de factor de crecimiento de fibroblastos 18. MX2016010871A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP14000600 2014-02-20
PCT/EP2015/053624 WO2015124727A1 (en) 2014-02-20 2015-02-20 Fgf-18 compound dosing regimen

Publications (1)

Publication Number Publication Date
MX2016010871A true MX2016010871A (es) 2016-11-17

Family

ID=50151088

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2016010872A MX2016010872A (es) 2014-02-20 2015-02-20 Regimen de dosificacion del compuesto de factor de crecimiento de fibroblastos 18.
MX2016010871A MX2016010871A (es) 2014-02-20 2015-02-20 Regimen de dosificacion del compuesto de factor de crecimiento de fibroblastos 18.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
MX2016010872A MX2016010872A (es) 2014-02-20 2015-02-20 Regimen de dosificacion del compuesto de factor de crecimiento de fibroblastos 18.

Country Status (25)

Country Link
US (2) US9724388B2 (es)
EP (2) EP3119417B1 (es)
JP (2) JP6431082B2 (es)
KR (2) KR102410988B1 (es)
CN (2) CN106232622A (es)
AR (2) AR099510A1 (es)
AU (2) AU2015220773B2 (es)
BR (2) BR112016018696A2 (es)
CA (2) CA2938793A1 (es)
DK (2) DK3119417T3 (es)
ES (2) ES2688551T3 (es)
HR (2) HRP20181570T1 (es)
HU (1) HUE040350T2 (es)
IL (2) IL247083B (es)
LT (2) LT3107559T (es)
MX (2) MX2016010872A (es)
NZ (1) NZ723148A (es)
PL (2) PL3119417T3 (es)
PT (2) PT3119417T (es)
RS (2) RS57853B1 (es)
RU (2) RU2691946C2 (es)
SG (2) SG11201606502YA (es)
SI (2) SI3119417T1 (es)
WO (2) WO2015124731A1 (es)
ZA (2) ZA201605548B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ723177A (en) 2014-02-20 2021-12-24 Merck Patent Gmbh Implant comprising fgf-18
BR112016018696A2 (pt) 2014-02-20 2017-10-17 Merck Patent Gmbh regime de dosagem com composto de fgf-18
JP6787904B2 (ja) 2015-01-29 2020-11-18 アレス トレーディング ソシエテ アノニム 高度に正に荷電したタンパク質のイムノアッセイ
RU2743075C2 (ru) 2016-02-22 2021-02-15 Новартис Аг Способы применения агонистов fxr
US11467169B2 (en) * 2017-09-29 2022-10-11 Merck Patent Gmbh Inflammatory biomarkers for predicting responsiveness to FGF-18 compound
US11513128B2 (en) 2017-09-29 2022-11-29 Merck Patent Gmbh Metabolic biomarkers for predicting responsiveness to FGF-18 compound
IL281333B2 (en) 2018-09-10 2025-11-01 Merck Patent Gmbh A method for reducing risk in a clinical trial
WO2020161341A1 (en) * 2019-02-08 2020-08-13 Merck Patent Gmbh Treatment of patients at risk of rapid progression of osteoarthritis
WO2025077768A1 (en) * 2023-10-11 2025-04-17 Sichuan Real & Best Biotech Co., Ltd. Compositions and methods for treating arthritis

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20040136970A1 (en) * 2002-10-07 2004-07-15 Ellsworth Jeff L. Methods for administering FGF18
ES2706848T3 (es) * 2004-07-06 2019-04-01 Zymogenetics Inc Composición farmacéutica que comprende FGF18 y antagonista de IL-1 y método de uso
AU2006326870A1 (en) * 2005-12-22 2007-06-28 Apollo Life Sciences Transdermal delivery of pharmaceutical agents
CA2658511C (en) * 2006-08-25 2019-02-19 Ares Trading S.A. Use of fgf-18 compound to treat cartilage disorders
BRPI0715728A8 (pt) * 2006-08-25 2018-04-03 Ares Trading Sa tratamento de distúrbios cartilaginosos
DE102006043260A1 (de) * 2006-09-11 2008-03-27 Krones Ag Etikettieranlage
WO2012127506A1 (en) * 2011-03-22 2012-09-27 Advinus Therapeutics Limited Substituted fused tricyclic compounds, compositions and medicinal applications thereof
NZ723177A (en) 2014-02-20 2021-12-24 Merck Patent Gmbh Implant comprising fgf-18
WO2015124735A1 (en) 2014-02-20 2015-08-27 Merck Patent Gmbh Fgf-18 in graft transplantation and tissue engineering procedures
BR112016018696A2 (pt) 2014-02-20 2017-10-17 Merck Patent Gmbh regime de dosagem com composto de fgf-18

Also Published As

Publication number Publication date
PL3119417T3 (pl) 2019-01-31
RU2016137292A (ru) 2018-03-21
IL247083B (en) 2019-09-26
SG11201606502YA (en) 2016-09-29
AU2015220777B2 (en) 2020-10-22
RU2016137289A (ru) 2018-03-21
IL247084B (en) 2019-09-26
EP3107559A1 (en) 2016-12-28
US9889179B2 (en) 2018-02-13
AU2015220773B2 (en) 2020-10-08
RU2691946C2 (ru) 2019-06-19
US9724388B2 (en) 2017-08-08
HRP20181570T1 (hr) 2018-11-30
SI3119417T1 (sl) 2018-11-30
PT3107559T (pt) 2018-10-31
HUE040350T2 (hu) 2019-03-28
DK3107559T3 (en) 2018-10-15
US20170072017A1 (en) 2017-03-16
DK3119417T3 (en) 2018-10-22
NZ723148A (en) 2022-08-26
MX2016010872A (es) 2016-11-17
NZ723139A (en) 2022-12-23
HRP20181572T1 (hr) 2018-11-30
CN106456713A (zh) 2017-02-22
ZA201605548B (en) 2018-12-19
AR099510A1 (es) 2016-07-27
US20170056474A1 (en) 2017-03-02
AU2015220773A1 (en) 2016-09-01
RU2016137289A3 (es) 2018-10-19
ZA201605547B (en) 2019-09-25
AU2015220777A1 (en) 2016-09-01
CA2938791A1 (en) 2015-08-27
KR20160116000A (ko) 2016-10-06
CN106232622A (zh) 2016-12-14
ES2689071T3 (es) 2018-11-08
JP6431083B2 (ja) 2018-11-28
KR20160116001A (ko) 2016-10-06
AR099558A1 (es) 2016-08-03
EP3107559B1 (en) 2018-07-11
JP2017507142A (ja) 2017-03-16
SG11201606505UA (en) 2016-09-29
JP6431082B2 (ja) 2018-11-28
KR102410986B1 (ko) 2022-06-17
JP2017512194A (ja) 2017-05-18
PT3119417T (pt) 2018-10-31
LT3107559T (lt) 2018-10-25
EP3119417B1 (en) 2018-07-11
BR112016018696A2 (pt) 2017-10-17
IL247084A0 (en) 2016-09-29
SI3107559T1 (sl) 2018-11-30
ES2688551T3 (es) 2018-11-05
WO2015124727A1 (en) 2015-08-27
WO2015124731A1 (en) 2015-08-27
RS57853B1 (sr) 2018-12-31
RS57709B1 (sr) 2018-12-31
EP3119417A1 (en) 2017-01-25
LT3119417T (lt) 2018-10-25
RU2016137292A3 (es) 2018-09-17
RU2700582C2 (ru) 2019-09-18
IL247083A0 (en) 2016-09-29
PL3107559T3 (pl) 2019-01-31
CA2938793A1 (en) 2015-08-27
BR112016018685A2 (pt) 2017-10-17
KR102410988B1 (ko) 2022-06-17

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