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MX2016003979A - Metodo para profilaxis o tratamiento de lupus eritematoso sistemico y/o nefritis lupica. - Google Patents

Metodo para profilaxis o tratamiento de lupus eritematoso sistemico y/o nefritis lupica.

Info

Publication number
MX2016003979A
MX2016003979A MX2016003979A MX2016003979A MX2016003979A MX 2016003979 A MX2016003979 A MX 2016003979A MX 2016003979 A MX2016003979 A MX 2016003979A MX 2016003979 A MX2016003979 A MX 2016003979A MX 2016003979 A MX2016003979 A MX 2016003979A
Authority
MX
Mexico
Prior art keywords
prophylaxis
treatment
lupus erythematosus
systemic lupus
nephritis
Prior art date
Application number
MX2016003979A
Other languages
English (en)
Inventor
Toru Kawamura
Yasushi Fujitani
Masayuki Takizawa
Original Assignee
Millennium Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Millennium Pharm Inc filed Critical Millennium Pharm Inc
Publication of MX2016003979A publication Critical patent/MX2016003979A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente invención brinda un método para profilaxis o el tratamiento de lupus eritematoso sistémico y/o nefritis lúpica en un paciente que lo necesita, que comprende administrarle una cantidad eficaz de ácido [(1R)-1-({[(2,5-diclorobenzoil)amino]acet il}amino)-3-metilbutil]borónico o un éster de ácido cítrico de éste o una sal farmacéuticamente aceptable de estos a un paciente.
MX2016003979A 2013-10-03 2014-10-02 Metodo para profilaxis o tratamiento de lupus eritematoso sistemico y/o nefritis lupica. MX2016003979A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201361886403P 2013-10-03 2013-10-03
PCT/US2014/058738 WO2015051067A1 (en) 2013-10-03 2014-10-02 Method for the prophylaxis or treatment of systemic lupus erythematosus and/or lupus nephritis

Publications (1)

Publication Number Publication Date
MX2016003979A true MX2016003979A (es) 2016-06-15

Family

ID=51842818

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016003979A MX2016003979A (es) 2013-10-03 2014-10-02 Metodo para profilaxis o tratamiento de lupus eritematoso sistemico y/o nefritis lupica.

Country Status (10)

Country Link
US (2) US20160250238A1 (es)
EP (1) EP3052105A1 (es)
JP (1) JP2016531886A (es)
KR (1) KR20160058886A (es)
CN (1) CN105705149A (es)
BR (1) BR112016007237A2 (es)
CA (1) CA2925935A1 (es)
EA (1) EA201690686A1 (es)
MX (1) MX2016003979A (es)
WO (1) WO2015051067A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4046633A1 (en) * 2018-06-27 2022-08-24 Algernon Pharmaceuticals Inc. The use of repirinast in the prophylaxis or treatment of renal fibrosis or kidney disease
CN115515578A (zh) * 2020-05-07 2022-12-23 诺罗瑞韦有限公司 用于治疗抑郁症的环丝氨酸和己酮可可碱联合疗法
CN121041156A (zh) * 2025-08-27 2025-12-02 复皙药业(上海)有限公司 含有替普瑞酮的具有祛红功效的膏霜及其制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6083903A (en) 1994-10-28 2000-07-04 Leukosite, Inc. Boronic ester and acid compounds, synthesis and uses
EP1355910B1 (en) 2001-01-25 2011-03-09 The United States of America, represented by the Secretary, Department of Health and Human Services Formulation of boronic acid compounds
US7442830B1 (en) 2007-08-06 2008-10-28 Millenium Pharmaceuticals, Inc. Proteasome inhibitors
KR20150010802A (ko) * 2007-08-06 2015-01-28 밀레니엄 파머슈티컬스 인코퍼레이티드 프로테아좀 억제제
KR101691093B1 (ko) * 2008-06-17 2016-12-29 밀레니엄 파머슈티컬스 인코퍼레이티드 보로네이트 에스테르 화합물 및 이의 제약학적 조성물
AR075090A1 (es) 2008-09-29 2011-03-09 Millennium Pharm Inc Derivados de acido 1-amino-2-ciclobutiletilboronico inhibidores de proteosoma,utiles como agentes anticancerigenos, y composiciones farmaceuticas que los comprenden.
TW201103904A (en) 2009-06-11 2011-02-01 Hoffmann La Roche Janus kinase inhibitor compounds and methods
MX2012011298A (es) 2010-03-31 2012-11-06 Millennium Pharm Inc Derivados del acido 1-amino-2-ciclopropiletilboronico.
TW201309303A (zh) 2011-03-03 2013-03-01 Cephalon Inc 用於治療狼瘡的蛋白酶體抑制劑
WO2012177835A1 (en) * 2011-06-22 2012-12-27 Cephalon, Inc. Proteasome inhibitors and processes for their preparation, purification and use

Also Published As

Publication number Publication date
JP2016531886A (ja) 2016-10-13
US20180099000A1 (en) 2018-04-12
CA2925935A1 (en) 2015-04-09
BR112016007237A2 (pt) 2017-09-12
WO2015051067A1 (en) 2015-04-09
EA201690686A1 (ru) 2016-08-31
CN105705149A (zh) 2016-06-22
US20160250238A1 (en) 2016-09-01
KR20160058886A (ko) 2016-05-25
EP3052105A1 (en) 2016-08-10

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