MX2015013051A - 1-hidroxi-benzooxaboroles como agentes antiparasitarios. - Google Patents
1-hidroxi-benzooxaboroles como agentes antiparasitarios.Info
- Publication number
- MX2015013051A MX2015013051A MX2015013051A MX2015013051A MX2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A MX 2015013051 A MX2015013051 A MX 2015013051A
- Authority
- MX
- Mexico
- Prior art keywords
- benzooxaboroles
- hydroxy
- compounds
- controlling
- antiparasitic agents
- Prior art date
Links
- 239000003096 antiparasitic agent Substances 0.000 title 1
- 229940125687 antiparasitic agent Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 6
- 241001465754 Metazoa Species 0.000 abstract 3
- 244000079386 endoparasite Species 0.000 abstract 3
- 206010061217 Infestation Diseases 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 238000009472 formulation Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/025—Boronic and borinic acid compounds
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
- A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Environmental Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Dentistry (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Tropical Medicine & Parasitology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Epidemiology (AREA)
- Steroid Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
Abstract
Se proporcionan compuestos útiles para controlar endoparásitos tanto en animales como en agricultura. Además se proporcionan métodos para controlar infestaciones de endoparásitos de un animal al administrar una cantidad efectiva de un compuesto como se describe antes, o una sal farmacéuticamente aceptable del mismo, a un animal, así como formulaciones para controlar infestaciones de endoparásitos que usa los compuestos descritos antes o una sal aceptable de los mismos, y un portador aceptable. Los compuestos reclamados son descritos mediante la siguiente fórmula de Markush: Un ejemplo típico de un compuesto de acuerdo con la fórmula anterior es: Un ejemplo típico para un compuesto de acuerdo con la fórmula anterior es: (véase formula).
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361786839P | 2013-03-15 | 2013-03-15 | |
| PCT/US2014/020966 WO2014149793A1 (en) | 2013-03-15 | 2014-03-06 | 1 -hydroxy-benzooxaboroles as antiparasitic agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2015013051A true MX2015013051A (es) | 2016-05-05 |
Family
ID=50382679
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2015013051A MX2015013051A (es) | 2013-03-15 | 2014-03-06 | 1-hidroxi-benzooxaboroles como agentes antiparasitarios. |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US9617285B2 (es) |
| EP (1) | EP2970339B1 (es) |
| JP (1) | JP6121043B2 (es) |
| KR (1) | KR101727421B1 (es) |
| CN (1) | CN105051048B (es) |
| AR (1) | AR094961A1 (es) |
| AU (1) | AU2014237862B2 (es) |
| BR (1) | BR112015020823A8 (es) |
| CA (1) | CA2899972A1 (es) |
| CY (1) | CY1119473T1 (es) |
| DK (1) | DK2970339T3 (es) |
| EA (1) | EA027430B1 (es) |
| ES (1) | ES2645687T3 (es) |
| HR (1) | HRP20171517T1 (es) |
| HU (1) | HUE035545T2 (es) |
| LT (1) | LT2970339T (es) |
| MX (1) | MX2015013051A (es) |
| NO (1) | NO2904426T3 (es) |
| PL (1) | PL2970339T3 (es) |
| PT (1) | PT2970339T (es) |
| RS (1) | RS56532B1 (es) |
| SI (1) | SI2970339T1 (es) |
| TW (1) | TW201506031A (es) |
| WO (1) | WO2014149793A1 (es) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10070649B2 (en) | 2013-01-30 | 2018-09-11 | Agrofresh Inc. | Volatile applications against pathogens |
| US11039617B2 (en) | 2013-01-30 | 2021-06-22 | Agrofresh Inc. | Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness |
| WO2016001834A1 (en) | 2014-07-01 | 2016-01-07 | Daiichi Sankyo Company, Limited | Tricyclic benzoxaboroles as antibacterial agents |
| TW201735792A (zh) | 2016-03-07 | 2017-10-16 | 農業保鮮股份有限公司 | 使用苯并氧雜硼雜環戊烯化合物和防腐氣體作為作物的抗微生物劑之協同方法 |
| CA3026316A1 (en) | 2016-06-03 | 2017-12-07 | Basf Se | Benzoxaborole compounds |
| WO2018156554A1 (en) * | 2017-02-21 | 2018-08-30 | Dow Agrosciences Llc | 1-HYDROXY-1,3-DIHYDROBENZO[c][1,2]OXABOROLES AND THEIR USE AS HERBICIDES |
| CN108864160A (zh) * | 2017-05-16 | 2018-11-23 | 苏州旺山旺水生物医药有限公司 | 含硼小分子的制备方法 |
| WO2019025250A1 (en) | 2017-08-04 | 2019-02-07 | Basf Se | SUBSTITUTED TRIFLUOROMETHYLOXADIAZOLES FOR COMBATING PHYTOPATHOGENIC FUNGI |
| EP3716766A4 (en) | 2017-11-30 | 2021-12-22 | Boragen, Inc. | BENZOXABOROLE COMPOUNDS AND THEIR FORMULATIONS |
| CA3148168A1 (en) | 2018-08-18 | 2020-02-27 | Chun Yu Liu | Solid forms of substituted benzoxaborole and compositions thereof |
| US20230340530A1 (en) | 2020-08-31 | 2023-10-26 | Pfizer Inc. | Methods of Protecting RNA |
| CN112321510A (zh) * | 2020-10-27 | 2021-02-05 | 无锡双启科技有限公司 | 一种4-溴-5-甲基-1h-吲唑的制备方法 |
| CN112745270B (zh) * | 2020-12-30 | 2023-02-24 | 河北医科大学 | 新化合物及其制备苯唑草酮中间体的方法 |
| EP4137485A1 (en) * | 2021-08-20 | 2023-02-22 | Henkel AG & Co. KGaA | Vinyl ethers |
Family Cites Families (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6239077B1 (en) | 1998-05-01 | 2001-05-29 | Nihon Nohyaku Co., Ltd. | Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof |
| CN1531426A (zh) | 2000-12-20 | 2004-09-22 | ��˹��ŵ�� | 有机化合物 |
| AR035531A1 (es) | 2001-01-22 | 2004-06-02 | Novartis Ag | Composicion para el control de plagas endoparasiticas en ganados y animales domesticos, un metodo para su control y el uso de dicha composicion para la preparacion de medicamentos |
| TWI236341B (en) | 2001-06-15 | 2005-07-21 | Novartis Ag | Aminoacetonitrile compounds for use in the control of endoparasites |
| AR038156A1 (es) | 2002-01-21 | 2004-12-29 | Novartis Ag | Compuestos de amidoacetonitrilo, proceso para su preparacion, composicion para controlar los parasitos, y uso de estos compuestos para preparar una composicion farmaceutica |
| TW200305556A (en) | 2002-03-21 | 2003-11-01 | Novartis Ag | Organic compounds |
| TW200400931A (en) | 2002-05-22 | 2004-01-16 | Novartis Ag | Organic compounds |
| TW200400004A (en) | 2002-05-22 | 2004-01-01 | Novartis Ag | Organic compounds |
| AR039961A1 (es) | 2002-06-06 | 2005-03-09 | Novartis Ag | Derivados de amidoacetonitrilo y su uso como pesticida |
| TW200400932A (en) | 2002-06-19 | 2004-01-16 | Novartis Ag | Organic compounds |
| GB0402677D0 (en) | 2003-11-06 | 2004-03-10 | Novartis Ag | Organic compounds |
| AR046757A1 (es) | 2003-12-10 | 2005-12-21 | Novartis Ag | Amidoacetonitrilos utiles como pesticidas |
| TW200613251A (en) | 2004-06-10 | 2006-05-01 | Novartis Ag | Organic compounds |
| KR101337045B1 (ko) * | 2005-02-16 | 2013-12-05 | 아나코르 파마슈티칼스 인코포레이티드 | 보론함유 소분자 |
| EP1910278A1 (en) | 2005-07-25 | 2008-04-16 | Novartis AG | Amidonitrile compounds |
| AU2006333527B2 (en) | 2005-12-30 | 2013-08-01 | Anacor Pharmaceuticals, Llc | Boron-containing small molecules |
| EP2125766B1 (en) | 2007-02-21 | 2011-07-06 | Pfizer Limited | Benzofuran antiparasitic agents |
| US20100026457A1 (en) * | 2008-08-04 | 2010-02-04 | Cooper Technologies Company | Location of Tagged Boxes |
| KR101782311B1 (ko) | 2008-10-21 | 2017-09-27 | 메리얼 인코포레이티드 | 티오아미드 화합물, 이의 제조 방법 및 사용 방법 |
| AU2010281439A1 (en) | 2009-07-28 | 2012-03-15 | Anacor Pharmaceuticals, Inc. | Trisubstituted boron-containing molecules |
| WO2011019612A1 (en) | 2009-08-14 | 2011-02-17 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| EP2314292A1 (en) | 2009-10-20 | 2011-04-27 | Novartis AG | Endoparasiticidal compositions |
| WO2011049971A1 (en) * | 2009-10-20 | 2011-04-28 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| UY32992A (es) | 2009-11-23 | 2011-04-29 | Novartis Ag | Compuestos orgánicos |
| SI3030519T1 (sl) * | 2013-08-09 | 2022-04-29 | Glaxosmithkline Intellectual Property (No.2) Limited | Triciklične benzoksaborolne spojine in njihove uporabe |
-
2014
- 2014-02-28 AR ARP140100676A patent/AR094961A1/es unknown
- 2014-03-06 EP EP14712939.9A patent/EP2970339B1/en active Active
- 2014-03-06 TW TW103107747A patent/TW201506031A/zh unknown
- 2014-03-06 SI SI201430345T patent/SI2970339T1/sl unknown
- 2014-03-06 US US14/760,208 patent/US9617285B2/en not_active Expired - Fee Related
- 2014-03-06 LT LTEP14712939.9T patent/LT2970339T/lt unknown
- 2014-03-06 HU HUE14712939A patent/HUE035545T2/en unknown
- 2014-03-06 CA CA2899972A patent/CA2899972A1/en not_active Abandoned
- 2014-03-06 RS RS20171064A patent/RS56532B1/sr unknown
- 2014-03-06 MX MX2015013051A patent/MX2015013051A/es unknown
- 2014-03-06 WO PCT/US2014/020966 patent/WO2014149793A1/en not_active Ceased
- 2014-03-06 PT PT147129399T patent/PT2970339T/pt unknown
- 2014-03-06 PL PL14712939T patent/PL2970339T3/pl unknown
- 2014-03-06 AU AU2014237862A patent/AU2014237862B2/en not_active Ceased
- 2014-03-06 EA EA201591512A patent/EA027430B1/ru not_active IP Right Cessation
- 2014-03-06 ES ES14712939.9T patent/ES2645687T3/es active Active
- 2014-03-06 JP JP2016500695A patent/JP6121043B2/ja active Active
- 2014-03-06 KR KR1020157024782A patent/KR101727421B1/ko not_active Expired - Fee Related
- 2014-03-06 BR BR112015020823A patent/BR112015020823A8/pt active Search and Examination
- 2014-03-06 HR HRP20171517TT patent/HRP20171517T1/hr unknown
- 2014-03-06 DK DK14712939.9T patent/DK2970339T3/en active
- 2014-03-06 CN CN201480014758.9A patent/CN105051048B/zh not_active Expired - Fee Related
- 2014-11-18 NO NO14799476A patent/NO2904426T3/no unknown
-
2017
- 2017-10-20 CY CY20171101096T patent/CY1119473T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DK2970339T3 (en) | 2017-10-02 |
| EA201591512A1 (ru) | 2016-01-29 |
| EP2970339A1 (en) | 2016-01-20 |
| EP2970339B1 (en) | 2017-08-16 |
| WO2014149793A1 (en) | 2014-09-25 |
| PL2970339T3 (pl) | 2018-01-31 |
| HUE035545T2 (en) | 2018-05-28 |
| CY1119473T1 (el) | 2018-03-07 |
| EA201591512A9 (ru) | 2016-04-29 |
| ES2645687T3 (es) | 2017-12-07 |
| CA2899972A1 (en) | 2014-09-25 |
| TW201506031A (zh) | 2015-02-16 |
| BR112015020823A8 (pt) | 2019-09-17 |
| KR101727421B1 (ko) | 2017-04-14 |
| JP6121043B2 (ja) | 2017-04-26 |
| NO2904426T3 (es) | 2018-02-10 |
| KR20150119154A (ko) | 2015-10-23 |
| AU2014237862A1 (en) | 2015-08-13 |
| AR094961A1 (es) | 2015-09-09 |
| PT2970339T (pt) | 2017-11-14 |
| SI2970339T1 (sl) | 2017-10-30 |
| CN105051048B (zh) | 2017-03-15 |
| AU2014237862B2 (en) | 2017-01-12 |
| HRP20171517T1 (hr) | 2017-11-17 |
| RS56532B1 (sr) | 2018-02-28 |
| EA027430B1 (ru) | 2017-07-31 |
| JP2016516032A (ja) | 2016-06-02 |
| LT2970339T (lt) | 2017-11-10 |
| CN105051048A (zh) | 2015-11-11 |
| US20150353581A1 (en) | 2015-12-10 |
| US9617285B2 (en) | 2017-04-11 |
| BR112015020823A2 (pt) | 2017-07-18 |
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