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MX2015008171A - Formulacion que comprende agomelatina amorfa. - Google Patents

Formulacion que comprende agomelatina amorfa.

Info

Publication number
MX2015008171A
MX2015008171A MX2015008171A MX2015008171A MX2015008171A MX 2015008171 A MX2015008171 A MX 2015008171A MX 2015008171 A MX2015008171 A MX 2015008171A MX 2015008171 A MX2015008171 A MX 2015008171A MX 2015008171 A MX2015008171 A MX 2015008171A
Authority
MX
Mexico
Prior art keywords
formulation
agomelatine
composition
amorphous
amorphous agomelatine
Prior art date
Application number
MX2015008171A
Other languages
English (en)
Inventor
Lisardo Álvarez Fernández
Rolf Keltjens
Jacobus Theodorus Henricus Eupen Van
Deepak Murpani
Sonia Garcia Jimenez
Original Assignee
Synthon Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthon Bv filed Critical Synthon Bv
Publication of MX2015008171A publication Critical patent/MX2015008171A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención se refiere a una composición de agomelatina y un copolímero de ácido metacrílico y divinilbenceno, a una formulación farmacéutica que comprende la composición y al uso de ya sea la composición o la formulación como un medicamento particularmente para el tratamiento del trastorno depresivo mayor.
MX2015008171A 2012-12-20 2013-12-17 Formulacion que comprende agomelatina amorfa. MX2015008171A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP2012076366 2012-12-20
PCT/EP2013/076842 WO2014095818A1 (en) 2012-12-20 2013-12-17 Formulation comprising amorphous agomelatine

Publications (1)

Publication Number Publication Date
MX2015008171A true MX2015008171A (es) 2015-09-16

Family

ID=49766107

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2015008171A MX2015008171A (es) 2012-12-20 2013-12-17 Formulacion que comprende agomelatina amorfa.

Country Status (2)

Country Link
MX (1) MX2015008171A (es)
WO (1) WO2014095818A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2705023A4 (en) * 2011-01-04 2014-11-19 Symed Labs Ltd PROCESSES FOR THE PREPARATION OF N- [2- (7-METHOXY-1-NAPHTHYLLELYHYL) ACETAMIDE
WO2017059877A1 (en) * 2015-10-07 2017-04-13 Rontis Hellas S.A. Pharmaceutical composition containing agomelatine and process for the preparation thereof
EP3466413A1 (en) 2017-10-09 2019-04-10 KRKA, d.d., Novo mesto Pharmaceutical composition containing agomelatine and process for the preparation thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2378573T3 (es) * 2006-03-16 2012-04-16 Tris Pharma, Inc. Formulaciones de liberación modificada que contienen complejos de fármaco-resina de intercambio iónico
CN101836966A (zh) * 2010-05-27 2010-09-22 北京万全阳光医药科技有限公司 一种含有阿戈美拉汀的口腔崩解片

Also Published As

Publication number Publication date
WO2014095818A1 (en) 2014-06-26

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