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MX2013005669A - Composiciones terapeuticas que comprenden hcl de rilpivirina y fumarato de disoproxilo de tenofovir. - Google Patents

Composiciones terapeuticas que comprenden hcl de rilpivirina y fumarato de disoproxilo de tenofovir.

Info

Publication number
MX2013005669A
MX2013005669A MX2013005669A MX2013005669A MX2013005669A MX 2013005669 A MX2013005669 A MX 2013005669A MX 2013005669 A MX2013005669 A MX 2013005669A MX 2013005669 A MX2013005669 A MX 2013005669A MX 2013005669 A MX2013005669 A MX 2013005669A
Authority
MX
Mexico
Prior art keywords
disoproxil fumarate
therapeutic compositions
tenofovir disoproxil
rilpivirine hcl
rilpivirine
Prior art date
Application number
MX2013005669A
Other languages
English (en)
Other versions
MX347512B (es
Inventor
Reza Oliyai
Lauren Wiser
Mark Menning
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45094284&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2013005669(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of MX2013005669A publication Critical patent/MX2013005669A/es
Publication of MX347512B publication Critical patent/MX347512B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invención proporciona tabletas de capas múltiples que contienen clorhidrato de rilpivirina, emtricitabina, y fumarato de disoproxilo de tenofivir. Las tabletas son útiles para el tratamiento de VIH.
MX2013005669A 2010-11-19 2011-11-18 Composiciones terapeuticas que comprenden hcl de rilpivirina y fumarato de disoproxilo de tenofovir. MX347512B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US41560010P 2010-11-19 2010-11-19
PCT/US2011/061515 WO2012068535A1 (en) 2010-11-19 2011-11-18 Therapeutic compositions comprising rilpivirine hcl and tenofovir disoproxil fumarate

Publications (2)

Publication Number Publication Date
MX2013005669A true MX2013005669A (es) 2013-11-04
MX347512B MX347512B (es) 2017-04-28

Family

ID=45094284

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013005669A MX347512B (es) 2010-11-19 2011-11-18 Composiciones terapeuticas que comprenden hcl de rilpivirina y fumarato de disoproxilo de tenofovir.

Country Status (36)

Country Link
US (1) US10857102B2 (es)
EP (2) EP2640362B2 (es)
JP (2) JP2014500261A (es)
KR (1) KR101923103B1 (es)
CN (2) CN103491948B (es)
AP (1) AP3816A (es)
AR (2) AR084500A1 (es)
AU (3) AU2011329642B2 (es)
BR (1) BR112013012245B1 (es)
CA (1) CA2818097C (es)
CL (1) CL2013001402A1 (es)
CO (1) CO6761300A2 (es)
CR (1) CR20130293A (es)
DK (1) DK2640362T4 (es)
EA (2) EA025852B1 (es)
EC (2) ECSP13012700A (es)
ES (1) ES2524408T5 (es)
HK (1) HK1206592A1 (es)
HR (1) HRP20140946T1 (es)
IL (1) IL226300B (es)
MA (1) MA34735B1 (es)
ME (1) ME01980B (es)
MX (1) MX347512B (es)
MY (1) MY185604A (es)
NZ (1) NZ610729A (es)
PE (3) PE20170521A1 (es)
PH (1) PH12013501002A1 (es)
PL (1) PL2640362T5 (es)
PT (1) PT2640362E (es)
RS (1) RS53691B1 (es)
SG (3) SG10201509521WA (es)
SM (1) SMT201400150B (es)
TW (1) TWI556840B (es)
UA (1) UA114075C2 (es)
WO (1) WO2012068535A1 (es)
ZA (1) ZA201304481B (es)

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WO2019113462A1 (en) 2017-12-07 2019-06-13 Emory University N4-hydroxycytidine and derivatives and anti-viral uses related thereto
KR20220028049A (ko) * 2019-07-03 2022-03-08 얀센 사이언시즈 아일랜드 언리미티드 컴퍼니 릴피비린으로 소아 환자에서의 hiv를 치료하는 방법
CN112137981A (zh) * 2020-11-02 2020-12-29 成都晶富医药科技有限公司 富马酸丙酚替诺福韦片及其制备工艺
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Also Published As

Publication number Publication date
WO2012068535A1 (en) 2012-05-24
ZA201304481B (en) 2022-03-30
UA114075C2 (xx) 2017-04-25
CA2818097A1 (en) 2012-05-24
DK2640362T3 (en) 2014-12-01
MX347512B (es) 2017-04-28
SG10201509521WA (en) 2015-12-30
AU2016208417B2 (en) 2018-04-05
EA201390651A1 (ru) 2013-11-29
EP2826466A1 (en) 2015-01-21
AP2013006931A0 (en) 2013-06-30
AR084500A1 (es) 2013-05-22
ECSP13012700A (es) 2013-08-30
TW201238612A (en) 2012-10-01
IL226300B (en) 2019-05-30
ES2524408T3 (es) 2014-12-09
PL2640362T5 (pl) 2022-05-02
EP2640362A1 (en) 2013-09-25
AU2011329642A1 (en) 2013-05-02
HK1190064A1 (en) 2014-06-27
US20130243857A1 (en) 2013-09-19
PE20170521A1 (es) 2017-05-27
PE20140163A1 (es) 2014-02-08
CL2013001402A1 (es) 2013-12-27
AR123409A2 (es) 2022-11-30
CR20130293A (es) 2013-10-03
AU2018202635A1 (en) 2018-05-10
EP2640362B2 (en) 2021-12-01
JP6138851B2 (ja) 2017-05-31
ME01980B (me) 2015-05-20
MY185604A (en) 2021-05-25
US10857102B2 (en) 2020-12-08
DK2640362T4 (da) 2022-03-07
ECSP19078196A (es) 2019-11-30
SG10201912527XA (en) 2020-02-27
ES2524408T5 (es) 2022-04-25
JP2015131853A (ja) 2015-07-23
HRP20140946T1 (hr) 2015-02-13
TWI556840B (zh) 2016-11-11
JP2014500261A (ja) 2014-01-09
AP3816A (en) 2016-09-30
PT2640362E (pt) 2014-11-28
SG190333A1 (en) 2013-06-28
PH12013501002A1 (en) 2013-09-09
AU2016208417A1 (en) 2016-08-18
BR112013012245B1 (pt) 2022-09-27
PE20211657A1 (es) 2021-08-24
EP2640362B1 (en) 2014-09-10
PL2640362T3 (pl) 2015-03-31
EA025852B1 (ru) 2017-02-28
KR20140037799A (ko) 2014-03-27
CN103491948B (zh) 2016-11-02
AU2011329642B2 (en) 2016-08-11
CN106511357A (zh) 2017-03-22
RS53691B1 (sr) 2015-04-30
CA2818097C (en) 2019-07-30
BR112013012245A2 (pt) 2016-08-09
EA201691695A1 (ru) 2017-11-30
SMT201400150B (it) 2015-01-15
KR101923103B1 (ko) 2018-11-28
MA34735B1 (fr) 2013-12-03
CN103491948A (zh) 2014-01-01
NZ610729A (en) 2015-10-30
CO6761300A2 (es) 2013-09-30
HK1206592A1 (en) 2016-01-15

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