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MX2013002430A - Formas de dosis de disolucion de rápida de agonistas de 5-ht2c. - Google Patents

Formas de dosis de disolucion de rápida de agonistas de 5-ht2c.

Info

Publication number
MX2013002430A
MX2013002430A MX2013002430A MX2013002430A MX2013002430A MX 2013002430 A MX2013002430 A MX 2013002430A MX 2013002430 A MX2013002430 A MX 2013002430A MX 2013002430 A MX2013002430 A MX 2013002430A MX 2013002430 A MX2013002430 A MX 2013002430A
Authority
MX
Mexico
Prior art keywords
dosage forms
fast
ht2c agonists
dissolve dosage
ht2c
Prior art date
Application number
MX2013002430A
Other languages
English (en)
Inventor
Yun Shan
Scott Stirn
Anthony C Blackburn
Anna Shifrina
Original Assignee
Arena Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc
Publication of MX2013002430A publication Critical patent/MX2013002430A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
    • C07D223/14—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D223/16—Benzazepines; Hydrogenated benzazepines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Child & Adolescent Psychology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se describen sales del agonista del receptor 5-HT2c (R)-8-cloro-1-metil-2, 3, 4, 5-tetrahidro-1H-3-benzazepina, y formas de dosis que las comprenden que son útiles para, entre otras cosas, el manejo del peso.
MX2013002430A 2010-09-01 2011-08-31 Formas de dosis de disolucion de rápida de agonistas de 5-ht2c. MX2013002430A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40258910P 2010-09-01 2010-09-01
PCT/US2011/049953 WO2012030951A1 (en) 2010-09-01 2011-08-31 Fast-dissolve dosage forms of 5-ht2c agonists

Publications (1)

Publication Number Publication Date
MX2013002430A true MX2013002430A (es) 2013-07-22

Family

ID=44645827

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013002430A MX2013002430A (es) 2010-09-01 2011-08-31 Formas de dosis de disolucion de rápida de agonistas de 5-ht2c.

Country Status (11)

Country Link
US (1) US20140148442A1 (es)
EP (1) EP2611781A1 (es)
JP (1) JP2013536858A (es)
KR (1) KR20130138768A (es)
CN (1) CN103189358A (es)
AU (1) AU2011296027A1 (es)
CA (1) CA2808900A1 (es)
IN (1) IN2013DN02552A (es)
MX (1) MX2013002430A (es)
SG (2) SG10201506873WA (es)
WO (1) WO2012030951A1 (es)

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EP3485878A1 (en) 2010-09-01 2019-05-22 Arena Pharmaceuticals, Inc. Modified-release dosage forms of 5-ht2c agonists useful for weight management
EP2939677A1 (en) 2010-09-01 2015-11-04 Arena Pharmaceuticals, Inc. Administration of lorcaserin to indviduals with renal impairment
MX2013002421A (es) 2010-09-01 2013-05-17 Arena Pharm Inc Sales no hidroscopicas de agonistas de 5-ht2c.
WO2012030938A1 (en) 2010-09-01 2012-03-08 Arena Pharmaceuticals, Inc. Salts of lorcaserin with optically active acids
WO2014058441A1 (en) 2012-10-09 2014-04-17 Arena Pharmaceuticals, Inc. Method of weight management
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EP2868656A1 (en) * 2013-11-05 2015-05-06 LEK Pharmaceuticals d.d. Stabilized amorphous lorcaserin hydrochloride
CN104936947B (zh) * 2013-12-27 2017-03-08 杭州普晒医药科技有限公司 氯卡色林盐及其晶体、其制备方法和用途
US9981912B2 (en) 2014-04-21 2018-05-29 Hangzhou Pushai Pharmaceutical Technology Co., Ltd. Cocrystal of lorcaserin, preparation methods, pharmaceutical compositions and uses thereof
CN103901151A (zh) * 2014-04-23 2014-07-02 湖北朗昕生化药业有限公司 一种hplc法检测氯卡色林盐酸盐含量的方法
TW201618787A (zh) 2014-10-30 2016-06-01 艾尼納製藥公司 組合物及方法
CN109475586A (zh) 2016-06-29 2019-03-15 康纳塞斯创新公司 脱羧的大麻树脂、其用途和制备其的方法

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Also Published As

Publication number Publication date
SG188363A1 (en) 2013-04-30
KR20130138768A (ko) 2013-12-19
SG10201506873WA (en) 2015-10-29
AU2011296027A1 (en) 2013-04-04
JP2013536858A (ja) 2013-09-26
CN103189358A (zh) 2013-07-03
EP2611781A1 (en) 2013-07-10
CA2808900A1 (en) 2012-03-08
IN2013DN02552A (es) 2015-08-07
WO2012030951A1 (en) 2012-03-08
US20140148442A1 (en) 2014-05-29

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