MX2012014970A - Composiciones farmaceuticas que comprenden ezetimiba y rosuvastatina de calcio amorfo novedoso. - Google Patents
Composiciones farmaceuticas que comprenden ezetimiba y rosuvastatina de calcio amorfo novedoso.Info
- Publication number
- MX2012014970A MX2012014970A MX2012014970A MX2012014970A MX2012014970A MX 2012014970 A MX2012014970 A MX 2012014970A MX 2012014970 A MX2012014970 A MX 2012014970A MX 2012014970 A MX2012014970 A MX 2012014970A MX 2012014970 A MX2012014970 A MX 2012014970A
- Authority
- MX
- Mexico
- Prior art keywords
- ezetimibe
- pharmaceutical compositions
- rosuvastatin calcium
- amorphous rosuvastatin
- novel amorphous
- Prior art date
Links
- OLNTVTPDXPETLC-XPWALMASSA-N ezetimibe Chemical compound N1([C@@H]([C@H](C1=O)CC[C@H](O)C=1C=CC(F)=CC=1)C=1C=CC(O)=CC=1)C1=CC=C(F)C=C1 OLNTVTPDXPETLC-XPWALMASSA-N 0.000 title abstract 2
- 229960000815 ezetimibe Drugs 0.000 title abstract 2
- 229960004796 rosuvastatin calcium Drugs 0.000 title abstract 2
- LALFOYNTGMUKGG-BGRFNVSISA-L rosuvastatin calcium Chemical compound [Ca+2].CC(C)C1=NC(N(C)S(C)(=O)=O)=NC(C=2C=CC(F)=CC=2)=C1\C=C\[C@@H](O)C[C@@H](O)CC([O-])=O.CC(C)C1=NC(N(C)S(C)(=O)=O)=NC(C=2C=CC(F)=CC=2)=C1\C=C\[C@@H](O)C[C@@H](O)CC([O-])=O LALFOYNTGMUKGG-BGRFNVSISA-L 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000002245 particle Substances 0.000 abstract 1
Landscapes
- Medicinal Preparation (AREA)
Abstract
La presente invención se refiere a un proceso para preparar una combinación farmacéutica de dosis fija que comprende (a) ezetimibe con un tamaño de partícula d90 menor a 10 µm, (b) rosuvastatina de calcio amorfo.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MX2012014970A MX2012014970A (es) | 2012-12-18 | 2012-12-18 | Composiciones farmaceuticas que comprenden ezetimiba y rosuvastatina de calcio amorfo novedoso. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MX2012014970A MX2012014970A (es) | 2012-12-18 | 2012-12-18 | Composiciones farmaceuticas que comprenden ezetimiba y rosuvastatina de calcio amorfo novedoso. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2012014970A true MX2012014970A (es) | 2013-08-27 |
Family
ID=49552931
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2012014970A MX2012014970A (es) | 2012-12-18 | 2012-12-18 | Composiciones farmaceuticas que comprenden ezetimiba y rosuvastatina de calcio amorfo novedoso. |
Country Status (1)
| Country | Link |
|---|---|
| MX (1) | MX2012014970A (es) |
Cited By (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2015044698A3 (en) * | 2013-09-30 | 2015-05-14 | Egis Gyógyszergyár Zrt. | Medical composition containing a cholesterol absorption inhibitor and cholesterol biosynthesis inhibitor |
| CN105873571A (zh) * | 2013-12-30 | 2016-08-17 | 韩美药品株式会社 | 包含依泽替米贝和瑞舒伐他汀的口服复合制剂 |
| WO2018041282A1 (en) * | 2016-09-05 | 2018-03-08 | Zentiva, K.S. | A pharmaceutical composition comprising rosuvastatin and ezetimibe and a preparation method thereof |
| WO2018041281A1 (en) * | 2016-09-05 | 2018-03-08 | Zentiva, K.S. | A pharmaceutical composition comprising rosuvastatin and ezetimibe and a preparation method thereof |
| WO2021019499A1 (en) | 2019-07-31 | 2021-02-04 | TECNIMEDE - Sociedade Técnico-medicinal, SA | Solid oral multiple-unit immediate release compositions, methods and uses thereof |
-
2012
- 2012-12-18 MX MX2012014970A patent/MX2012014970A/es unknown
Cited By (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2015044698A3 (en) * | 2013-09-30 | 2015-05-14 | Egis Gyógyszergyár Zrt. | Medical composition containing a cholesterol absorption inhibitor and cholesterol biosynthesis inhibitor |
| CN105722505A (zh) * | 2013-09-30 | 2016-06-29 | 埃吉斯药物私人有限公司 | 含有胆固醇吸收抑制剂和胆固醇生物合成抑制剂的药物组合物 |
| CN114796148A (zh) * | 2013-09-30 | 2022-07-29 | 埃吉斯药物私人有限公司 | 含有胆固醇吸收抑制剂和胆固醇生物合成抑制剂的药物组合物 |
| EA034711B1 (ru) * | 2013-09-30 | 2020-03-12 | Эгиш Дьёдьсердьяр Зрт. | Лекарственная композиция, содержащая ингибитор всасывания холестерина и ингибитор биосинтеза холестерина |
| AU2014374552B2 (en) * | 2013-12-30 | 2019-09-19 | Hanmi Pharm. Co., Ltd. | Composite formulation for oral administration comprising ezetimibe and rosuvastatin |
| US10434067B2 (en) | 2013-12-30 | 2019-10-08 | Hanmi Pharm. Co., Ltd. | Composite formulation for oral administration comprising ezetimibe and rosuvastatin |
| CN105873571B (zh) * | 2013-12-30 | 2019-10-22 | 韩美药品株式会社 | 包含依泽替米贝和瑞舒伐他汀的口服复合制剂 |
| EP3089739A4 (en) * | 2013-12-30 | 2017-08-02 | Hanmi Pharm. Co., Ltd. | Composite formulation for oral administration comprising ezetimibe and rosuvastatin |
| CN105873571A (zh) * | 2013-12-30 | 2016-08-17 | 韩美药品株式会社 | 包含依泽替米贝和瑞舒伐他汀的口服复合制剂 |
| WO2018041281A1 (en) * | 2016-09-05 | 2018-03-08 | Zentiva, K.S. | A pharmaceutical composition comprising rosuvastatin and ezetimibe and a preparation method thereof |
| WO2018041282A1 (en) * | 2016-09-05 | 2018-03-08 | Zentiva, K.S. | A pharmaceutical composition comprising rosuvastatin and ezetimibe and a preparation method thereof |
| CN110418637A (zh) * | 2016-09-05 | 2019-11-05 | 赛诺菲 | 包含瑞舒伐他汀和依泽替米贝的药物组合物及其制备方法 |
| US11786526B2 (en) | 2016-09-05 | 2023-10-17 | Sanofi | Pharmaceutical composition comprising rosuvastatin and ezetimibe and a preparation method thereof |
| WO2021019499A1 (en) | 2019-07-31 | 2021-02-04 | TECNIMEDE - Sociedade Técnico-medicinal, SA | Solid oral multiple-unit immediate release compositions, methods and uses thereof |
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