MX2012014796A - Proceso para preparar 4-hidroxipiridinas. - Google Patents
Proceso para preparar 4-hidroxipiridinas.Info
- Publication number
- MX2012014796A MX2012014796A MX2012014796A MX2012014796A MX2012014796A MX 2012014796 A MX2012014796 A MX 2012014796A MX 2012014796 A MX2012014796 A MX 2012014796A MX 2012014796 A MX2012014796 A MX 2012014796A MX 2012014796 A MX2012014796 A MX 2012014796A
- Authority
- MX
- Mexico
- Prior art keywords
- hydroxypyridines
- preparing
- formula
- description
- meaning defined
- Prior art date
Links
- GCNTZFIIOFTKIY-UHFFFAOYSA-N 4-hydroxypyridine Chemical class OC1=CC=NC=C1 GCNTZFIIOFTKIY-UHFFFAOYSA-N 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/63—One oxygen atom
- C07D213/68—One oxygen atom attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/06—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
- C07D213/08—Preparation by ring-closure
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
La presente invención se refiere a un proceso para preparar 4-hidroxípiridinas de la fórmula I (ver Fórmula) en donde R1, R2, R3 y R4 tienen los significados definidos en la descripción.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35712810P | 2010-06-22 | 2010-06-22 | |
| EP10166877 | 2010-06-22 | ||
| PCT/IB2011/052681 WO2011161612A1 (en) | 2010-06-22 | 2011-06-20 | Process for preparing 4-hydroxypyridines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2012014796A true MX2012014796A (es) | 2013-04-03 |
Family
ID=45370915
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2012014796A MX2012014796A (es) | 2010-06-22 | 2011-06-20 | Proceso para preparar 4-hidroxipiridinas. |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US8716487B2 (es) |
| EP (1) | EP2585436B1 (es) |
| JP (1) | JP5984801B2 (es) |
| CN (1) | CN102947270B (es) |
| BR (1) | BR112012032671A2 (es) |
| ES (1) | ES2539379T3 (es) |
| MX (1) | MX2012014796A (es) |
| WO (1) | WO2011161612A1 (es) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103664761A (zh) * | 2013-12-06 | 2014-03-26 | 常熟市联创化学有限公司 | 一种4-吡啶酚的制备方法 |
| EP3548466B1 (en) | 2016-12-01 | 2022-01-12 | Syngenta Participations AG | Process for preparation of intermediate of pesticidally active heterocyclic derivatives with sulfur containing substituents |
| TWI795381B (zh) | 2016-12-21 | 2023-03-11 | 比利時商健生藥品公司 | 作為malt1抑制劑之吡唑衍生物 |
| CA3093445A1 (en) | 2018-03-08 | 2019-11-28 | Incyte Corporation | Aminopyrazine diol compounds as pi3k-.gamma. inhibitors |
| US11046658B2 (en) | 2018-07-02 | 2021-06-29 | Incyte Corporation | Aminopyrazine derivatives as PI3K-γ inhibitors |
| CA3129623A1 (en) | 2019-02-22 | 2020-08-27 | Janssen Pharmaceutica Nv | Crystalline form of 1-(1-oxo-1,2-dihydroisoquinolin-5-yl)-5-(trifluoromethyl)-n-(2-(trifluoromethyl)pyridin-4-yl)-1h-pyrazole-4-carboxamide monohydrate |
| EP3953345B1 (en) | 2019-04-11 | 2023-04-05 | Janssen Pharmaceutica NV | Pyridine rings containing derivatives as malt1 inhibitors |
| TW202517614A (zh) | 2023-07-12 | 2025-05-01 | 瑞士商先正達農作物保護股份公司 | 2-(三氟甲基)吡啶-4-胺的合成 |
| CN116925023B (zh) * | 2023-07-18 | 2025-11-21 | 江苏桐孚高新材料有限公司 | 2-全氟烷基-4h-吡喃-4-酮衍生物的改进合成方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6059236B2 (ja) * | 1977-07-06 | 1985-12-24 | 日清製粉株式会社 | γ−ピロン誘導体、その製造方法およびそれらの化合物からなる農業用薬剤 |
| JPS58170758A (ja) * | 1983-03-14 | 1983-10-07 | Nisshin Flour Milling Co Ltd | γ−ピリドン誘導体 |
| FR2650825B1 (fr) * | 1989-08-11 | 1991-12-06 | Isochem Sa | Nouvelle pyranone, procede pour sa preparation, son application a la preparation d'une nouvelle pyridinone et son procede de preparation |
| US5625069A (en) * | 1996-07-22 | 1997-04-29 | Development Center For Biotechnology | Process for preparing 2-cyano-3,5-dimethyl-4-methoxypyridine |
| CN100383123C (zh) * | 2004-03-12 | 2008-04-23 | 南通市东昌化工有限公司 | 4-羟基吡啶的生产方法 |
| DE102006059710A1 (de) | 2006-12-18 | 2008-06-19 | Freie Universität Berlin | Substituierte 4-Hydroxypyridine |
| EP2303828B1 (de) | 2008-06-25 | 2014-07-30 | Basf Se | Verfahren zur herstellung von substituierten biphenylen |
-
2011
- 2011-06-20 ES ES11797708.2T patent/ES2539379T3/es active Active
- 2011-06-20 US US13/805,567 patent/US8716487B2/en not_active Expired - Fee Related
- 2011-06-20 MX MX2012014796A patent/MX2012014796A/es active IP Right Grant
- 2011-06-20 EP EP11797708.2A patent/EP2585436B1/en active Active
- 2011-06-20 BR BR112012032671A patent/BR112012032671A2/pt not_active IP Right Cessation
- 2011-06-20 CN CN201180031044.5A patent/CN102947270B/zh not_active Expired - Fee Related
- 2011-06-20 WO PCT/IB2011/052681 patent/WO2011161612A1/en not_active Ceased
- 2011-06-20 JP JP2013516014A patent/JP5984801B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP2013530984A (ja) | 2013-08-01 |
| US8716487B2 (en) | 2014-05-06 |
| EP2585436B1 (en) | 2015-03-18 |
| BR112012032671A2 (pt) | 2015-09-15 |
| JP5984801B2 (ja) | 2016-09-06 |
| US20130096312A1 (en) | 2013-04-18 |
| CN102947270A (zh) | 2013-02-27 |
| ES2539379T3 (es) | 2015-06-30 |
| EP2585436A4 (en) | 2014-04-23 |
| EP2585436A1 (en) | 2013-05-01 |
| CN102947270B (zh) | 2015-04-08 |
| WO2011161612A1 (en) | 2011-12-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration |