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MX2012005859A - Peptidos lineales especificos del receptor de melanocortina-1. - Google Patents

Peptidos lineales especificos del receptor de melanocortina-1.

Info

Publication number
MX2012005859A
MX2012005859A MX2012005859A MX2012005859A MX2012005859A MX 2012005859 A MX2012005859 A MX 2012005859A MX 2012005859 A MX2012005859 A MX 2012005859A MX 2012005859 A MX2012005859 A MX 2012005859A MX 2012005859 A MX2012005859 A MX 2012005859A
Authority
MX
Mexico
Prior art keywords
receptor
melanocortin
specific linear
linear peptides
peptides
Prior art date
Application number
MX2012005859A
Other languages
English (en)
Inventor
Wei Yang
Yi-Qun Shi
Original Assignee
Palatin Technologies Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Palatin Technologies Inc filed Critical Palatin Technologies Inc
Publication of MX2012005859A publication Critical patent/MX2012005859A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/665Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
    • C07K14/68Melanocyte-stimulating hormone [MSH]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Toxicology (AREA)
  • Endocrinology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)

Abstract

Péptidos lineales específicos del receptor de la melanocortina de formula (I), donde R1, R2, R3, R4, R5, R6, R7, R8, R9, y R10 son como se define en la memoria descriptiva, las composiciones y formulaciones que incluyen péptidos de la fórmula anterior o las sales de estos, y los métodos para prevenir, mejorar o tratar enfermedades, indicaciones afecciones y síndromes sensibles o mediados por el receptor de la melanocortinas-1.
MX2012005859A 2009-11-23 2010-11-23 Peptidos lineales especificos del receptor de melanocortina-1. MX2012005859A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26348609P 2009-11-23 2009-11-23
PCT/US2010/057700 WO2011063367A1 (en) 2009-11-23 2010-11-23 Melanocortin-1 receptor-specific linear peptides

Publications (1)

Publication Number Publication Date
MX2012005859A true MX2012005859A (es) 2012-12-17

Family

ID=44060072

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2012005859A MX2012005859A (es) 2009-11-23 2010-11-23 Peptidos lineales especificos del receptor de melanocortina-1.

Country Status (13)

Country Link
US (3) US8933194B2 (es)
EP (1) EP2504351A4 (es)
JP (1) JP2013511554A (es)
KR (1) KR20120102716A (es)
CN (1) CN102712674A (es)
AU (1) AU2010321739A1 (es)
BR (1) BR112012011780A2 (es)
CA (1) CA2781405A1 (es)
EA (1) EA201290295A1 (es)
IL (1) IL219946A0 (es)
MX (1) MX2012005859A (es)
WO (1) WO2011063367A1 (es)
ZA (1) ZA201203331B (es)

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EP2504352B1 (en) 2009-11-23 2018-11-14 Palatin Technologies, Inc. Melanocortin-1 receptor-specific cyclic peptides

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JP2013511554A (ja) 2013-04-04
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