[go: up one dir, main page]

MX2011007779A - Formulaciones galenicas de compuestos organicos. - Google Patents

Formulaciones galenicas de compuestos organicos.

Info

Publication number
MX2011007779A
MX2011007779A MX2011007779A MX2011007779A MX2011007779A MX 2011007779 A MX2011007779 A MX 2011007779A MX 2011007779 A MX2011007779 A MX 2011007779A MX 2011007779 A MX2011007779 A MX 2011007779A MX 2011007779 A MX2011007779 A MX 2011007779A
Authority
MX
Mexico
Prior art keywords
core
tablet
organic compounds
outer coating
dosage form
Prior art date
Application number
MX2011007779A
Other languages
English (en)
Inventor
Stefan Hirsch
Sabine Desset-Brethes
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40770648&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2011007779(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MX2011007779A publication Critical patent/MX2011007779A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0087Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Vascular Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente solicitud se refiere a una forma de dosificación unitaria sólida para su administración oral en la forma de una tableta que tiene un núcleo y un recubrimiento externo, en donde: - el núcleo de la tableta comprende una cantidad terapéuticamente efectiva de Alisquireno, o de una sal farmacéuticamente aceptable del mismo, y - el recubrimiento externo está en la forma de un recubrimiento de película, el cual tiene propiedades enmascaradoras de sabor y/o una funcionalidad de liberación controlada. De preferencia, la tableta de núcleo es parte de un sistema de múltiples partículas, en particular una minitableta. La forma de dosificación oral sólida es en particular adecuada para uso pediátrico.
MX2011007779A 2009-01-28 2010-01-27 Formulaciones galenicas de compuestos organicos. MX2011007779A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP09151496 2009-01-28
PCT/EP2010/050886 WO2010086312A1 (en) 2009-01-28 2010-01-27 Galenic formulations of organic compounds

Publications (1)

Publication Number Publication Date
MX2011007779A true MX2011007779A (es) 2011-08-12

Family

ID=40770648

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2011007779A MX2011007779A (es) 2009-01-28 2010-01-27 Formulaciones galenicas de compuestos organicos.

Country Status (27)

Country Link
US (1) US20110287100A1 (es)
EP (1) EP2391345B1 (es)
JP (1) JP2012516299A (es)
KR (1) KR20110117199A (es)
CN (1) CN102300558A (es)
AR (1) AR075179A1 (es)
AU (1) AU2010209787B2 (es)
BR (1) BRPI1007452A2 (es)
CA (1) CA2749531A1 (es)
CL (1) CL2011001817A1 (es)
CO (1) CO6400184A2 (es)
EC (1) ECSP11011289A (es)
ES (1) ES2525648T3 (es)
IL (1) IL213918A0 (es)
MA (1) MA33060B1 (es)
MX (1) MX2011007779A (es)
MY (1) MY153852A (es)
NZ (1) NZ593622A (es)
PE (1) PE20110943A1 (es)
PL (1) PL2391345T3 (es)
PT (1) PT2391345E (es)
RU (1) RU2535090C2 (es)
SG (1) SG172226A1 (es)
TN (1) TN2011000307A1 (es)
TW (1) TWI468191B (es)
WO (1) WO2010086312A1 (es)
ZA (1) ZA201104489B (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5822758B2 (ja) * 2011-03-02 2015-11-24 第一三共ヘルスケア株式会社 速溶性防湿フィルムコーティング製剤及びその製造方法
EP2596802A1 (en) * 2011-11-23 2013-05-29 PLS-Design GmbH Pharmaceutical composition for treatment of allergic reactions
PT3411021T (pt) * 2016-02-03 2025-08-06 Novartis Ag Nova utilização de uma combinação de sacubitril e valsartan
US12171878B2 (en) 2018-08-10 2024-12-24 Kissei Pharmaceutical Co., Ltd. Sucroferric oxyhydroxide-containing granules and pharmaceutical composition
JP7681511B2 (ja) 2019-02-22 2025-05-22 キャタレント・ユーケー・スウィンドン・ザイディス・リミテッド インライン混合中の懸濁液の通気の最小化
BR112021016485A2 (pt) 2019-02-22 2021-10-13 Catalent U.K. Swindon Zydis Limited Minimização de aglomeração de material de revestimento de partícula de fármaco durante armazenamento para estabilizar tempos de desintegração de produtos farmacêuticos
GB2597578B (en) 2019-02-22 2023-04-26 Catalent Uk Swindon Zydis Ltd Preserving functionally-coated API particles produced by solventless mixing processes in aqueous suspension
BR112021016421A2 (pt) 2019-02-22 2021-10-13 Catalent U.K. Swindon Zydis Limited Minimização de aglomeração, aeração e preservação do revestimento de composições farmacêuticas que compreendem ibuprofeno
WO2021011538A1 (en) * 2019-07-15 2021-01-21 R.P. Scherer Technologies, Llc Capsule dosage forms, methods of preparation and methods of use thereof
AR123109A1 (es) 2020-07-31 2022-10-26 Catalent Uk Swindon Zydis Ltd Composiciones farmacéuticas que comprenden ifa
EP4255495A4 (en) 2020-12-03 2025-10-08 Battelle Memorial Institute COMPOSITIONS OF POLYMERIC NANOPARTICLES AND DNA NANOSTRUCTURES AND METHODS FOR NON-VIRAL DELIVERY
WO2022216977A1 (en) 2021-04-07 2022-10-13 Batelle Memorial Institute Rapid design, build, test, and learn technologies for identifying and using non-viral carriers
WO2025072751A1 (en) 2023-09-29 2025-04-03 Battelle Memorial Institute Polymer nanoparticle compositions for in vivo expression of polypeptides
WO2025105451A1 (ja) * 2023-11-17 2025-05-22 第一三共ヘルスケア株式会社 固形製剤
US12441996B2 (en) 2023-12-08 2025-10-14 Battelle Memorial Institute Use of DNA origami nanostructures for molecular information based data storage systems

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY119161A (en) 1994-04-18 2005-04-30 Novartis Ag Delta-amino-gamma-hydroxy-omega-aryl-alkanoic acid amides with enzyme especially renin inhibiting activities
DE19842753A1 (de) * 1998-09-18 2000-03-23 Bayer Ag Agitationsunabhängige pharmazeutische Retardzubereitungen und Verfahren zu ihrer Herstellung
US6248363B1 (en) * 1999-11-23 2001-06-19 Lipocine, Inc. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
AR034813A1 (es) * 2001-07-20 2004-03-17 Novartis Ag Composiciones farmaceuticas y uso de las mismas
US20040266743A1 (en) * 2003-05-09 2004-12-30 Pharmacia Corporation Combination of an aldosterone receptor antagonist and a renin inhibitor
MY144477A (en) 2004-03-17 2011-09-30 Novartis Ag Galenic formulations of organic compounds
US20070224260A1 (en) * 2004-04-15 2007-09-27 Dr. Reddy's Laboratories Limited Dosage Form Having Polymorphic Stability
ES2384637T3 (es) * 2004-10-08 2012-07-10 Novartis Ag Uso de inhibidores de la renina para la prevención o el tratamiento de disfunción diastólica o insuficiencia cardiaca diastólica
ES2364538T3 (es) * 2007-09-28 2011-09-06 Novartis Ag Combinación farmacéutica de alisquireno y valsartán.

Also Published As

Publication number Publication date
TWI468191B (zh) 2015-01-11
PT2391345E (pt) 2014-12-03
PE20110943A1 (es) 2012-01-22
TN2011000307A1 (en) 2012-12-17
RU2011135417A (ru) 2013-03-10
EP2391345B1 (en) 2014-09-03
HK1161125A1 (en) 2012-08-24
CA2749531A1 (en) 2010-08-05
CN102300558A (zh) 2011-12-28
AU2010209787A1 (en) 2011-07-14
WO2010086312A1 (en) 2010-08-05
SG172226A1 (en) 2011-07-28
CO6400184A2 (es) 2012-03-15
AU2010209787B2 (en) 2013-06-06
KR20110117199A (ko) 2011-10-26
MY153852A (en) 2015-03-31
TW201038300A (en) 2010-11-01
AR075179A1 (es) 2011-03-16
ECSP11011289A (es) 2011-09-30
EP2391345A1 (en) 2011-12-07
PL2391345T3 (pl) 2015-03-31
NZ593622A (en) 2013-12-20
JP2012516299A (ja) 2012-07-19
CL2011001817A1 (es) 2012-01-13
MA33060B1 (fr) 2012-02-01
ES2525648T3 (es) 2014-12-26
IL213918A0 (en) 2011-07-31
BRPI1007452A2 (pt) 2016-02-16
ZA201104489B (en) 2012-02-29
RU2535090C2 (ru) 2014-12-10
US20110287100A1 (en) 2011-11-24

Similar Documents

Publication Publication Date Title
MX2011007779A (es) Formulaciones galenicas de compuestos organicos.
MY152279A (en) Immediate release pharmaceutical compositions comprising oxycodone and naloxone
WO2008040534A3 (en) Non-mucoadhesive film dosage forms
EP4538227A3 (en) Sodium thiosulfate-containing pharmaceutical compositions
HK1221646A1 (zh) 高剂量普利多匹定用於治疗亨廷顿舞蹈症的用途
NZ589437A (en) Immediate release tablet comprising 5-azacytidine and a non-enteric coating applied with an ethanol solvent
WO2012007159A3 (en) Novel gastro-retentive dosage forms
TN2010000135A1 (en) Galenical formulations of organic compounds
NZ605469A (en) Nalbuphine-based formulations and uses thereof
HK1206246A1 (en) Use of high dose laquinimod for treating multiple sclerosis
PL2205279T3 (pl) Farmaceutyczna kombinacja aliskirenu i walsartanu
MY152951A (en) Solid pharmaceutical fixed dose compositions comprising irbesartan and amlodipine, their preparation and their therapeutic application
WO2011037976A3 (en) Pramipexole pharmaceutical formulations
SG141358A1 (en) Treatment of psychiatric patients with reduced heptaic function with paliperidone
WO2010012459A3 (en) A process for the preparation of solifenacin salts and their inclusion into pharmaceutical dosage forms
WO2007145863A3 (en) Sustained release formulation of naltrexone
GB2455875B (en) A process for the preparation of an orally administered unit dose tablet
WO2010044097A3 (en) Novel dosage form of paliperidone and process for preparing the same
GB0703674D0 (en) A Process For The Preparation of an Orally Administered Unit Dose Tablet
WO2013098268A3 (en) Tablets and dry-coated agents
JO3239B1 (ar) تركيبات جالينية من مركبات عضوية
GB0920721D0 (en) An orally administered anthelmintic unit dose tablet and process for the preparation thereof
ATE546133T1 (de) Orale dosierform mit trisubstituierten glycerin- verbindungen
WO2010035245A3 (en) Extended release dosage form of ropinirole
MX2011009846A (es) Formulaciones galenicas de una combinacion de dosis fija de valsartan y alisquireno.

Legal Events

Date Code Title Description
FA Abandonment or withdrawal