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MX2010009561A - Compuestos amida, composiciones y usos de los mismos. - Google Patents

Compuestos amida, composiciones y usos de los mismos.

Info

Publication number
MX2010009561A
MX2010009561A MX2010009561A MX2010009561A MX2010009561A MX 2010009561 A MX2010009561 A MX 2010009561A MX 2010009561 A MX2010009561 A MX 2010009561A MX 2010009561 A MX2010009561 A MX 2010009561A MX 2010009561 A MX2010009561 A MX 2010009561A
Authority
MX
Mexico
Prior art keywords
compositions
amide compounds
compounds
anxiety
inflammation
Prior art date
Application number
MX2010009561A
Other languages
English (en)
Inventor
John Kincaid
Zhi-Liang Wei
Yeyu Cao
Carl Kaub
Sumithra Gowlugari
Zhan Wang
Original Assignee
Renovis Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Renovis Inc filed Critical Renovis Inc
Publication of MX2010009561A publication Critical patent/MX2010009561A/es

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
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Abstract

Se proveen compuestos de conformidad con la fórmula 1: (ver fórmula 1) en donde A, B, W, X', L, R1, R3, R4b, y m' son como se definió en la presente invención; se proveen compuestos y composiciones farmacéuticas de los mismos útiles para la prevención y tratamiento de una variedad de condiciones en mamíferos incluyendo humanos, incluyendo a manera de ejemplo no limitante, dolor, inflamación, trastornos cognitivos, ansiedad, depresión, y otros.
MX2010009561A 2008-02-29 2009-02-27 Compuestos amida, composiciones y usos de los mismos. MX2010009561A (es)

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PCT/US2009/001249 WO2009110985A2 (en) 2008-02-29 2009-02-27 Amide compounds, compositions and uses thereof

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WO2009110985A2 (en) 2009-09-11
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