[go: up one dir, main page]

MX2010002868A - N6-(ferrocenmetil)quinazolin-2,4,6-triamina (h2), sus derivados y profarmacos, como agentes antimicrobianos antiparasitarios, antiprotozoarios y antileishmanias. - Google Patents

N6-(ferrocenmetil)quinazolin-2,4,6-triamina (h2), sus derivados y profarmacos, como agentes antimicrobianos antiparasitarios, antiprotozoarios y antileishmanias.

Info

Publication number
MX2010002868A
MX2010002868A MX2010002868A MX2010002868A MX2010002868A MX 2010002868 A MX2010002868 A MX 2010002868A MX 2010002868 A MX2010002868 A MX 2010002868A MX 2010002868 A MX2010002868 A MX 2010002868A MX 2010002868 A MX2010002868 A MX 2010002868A
Authority
MX
Mexico
Prior art keywords
antileishmania
antiprotozoal
antiparasitic
quinazolin
triamine
Prior art date
Application number
MX2010002868A
Other languages
English (en)
Inventor
Norma Del Carmen Galindo Sevilla
Francisco Hernandez Luis
Original Assignee
Norma Del Carmen Galindo Sevilla
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Norma Del Carmen Galindo Sevilla filed Critical Norma Del Carmen Galindo Sevilla
Priority to MX2010002868A priority Critical patent/MX2010002868A/es
Priority to ES11775335.0T priority patent/ES2618367T3/es
Priority to PCT/MX2011/000025 priority patent/WO2011136631A1/es
Priority to US13/643,949 priority patent/US8664384B2/en
Priority to EP11775335.0A priority patent/EP2599783B1/en
Priority to CN201180021289.XA priority patent/CN102918051B/zh
Publication of MX2010002868A publication Critical patent/MX2010002868A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F17/00—Metallocenes
    • C07F17/02—Metallocenes of metals of Groups 8, 9 or 10 of the Periodic Table
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/555—Heterocyclic compounds containing heavy metals, e.g. hemin, hematin, melarsoprol
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

El uso del compuesto N6(ferrocenmetil)quinazolin-2,4,6-triamina (H2), sus derivados y profármacos que presentan actividad como antimicrobiano (antibiótico, microbicida), antiparasitario (parasiticida), antiprotozoario (protozocida), antileishmania (leishmanicida) y su empleo como fármaco en vertebrados, humanos y animales.
MX2010002868A 2010-03-16 2010-03-16 N6-(ferrocenmetil)quinazolin-2,4,6-triamina (h2), sus derivados y profarmacos, como agentes antimicrobianos antiparasitarios, antiprotozoarios y antileishmanias. MX2010002868A (es)

Priority Applications (6)

Application Number Priority Date Filing Date Title
MX2010002868A MX2010002868A (es) 2010-03-16 2010-03-16 N6-(ferrocenmetil)quinazolin-2,4,6-triamina (h2), sus derivados y profarmacos, como agentes antimicrobianos antiparasitarios, antiprotozoarios y antileishmanias.
ES11775335.0T ES2618367T3 (es) 2010-03-16 2011-02-21 N6-(ferrocenmetil)quinazolin-2,4,6-triamina (H2), sus derivados y profármacos, como agentes antileishmanias, antiprotozoarios, antiparasitarios y antimicrobianos
PCT/MX2011/000025 WO2011136631A1 (es) 2010-03-16 2011-02-21 N6 -(ferrocenmetil)quinazolin-2,4,6-triamina (h2), sus derivados y profarmacos, como agentes antimicrobianos antiparasitarios, antiprotozoarios y antileishmanias
US13/643,949 US8664384B2 (en) 2010-03-16 2011-02-21 N6-(ferrocenmethyl)quinazolin-2,4,6-triamina (H2) and the derivatives and prodrugs thereof as antileishmanial, antiprotozoal, antiparasitic and antimicrobial agents
EP11775335.0A EP2599783B1 (en) 2010-03-16 2011-02-21 N6-(ferrocenmethyl)quinazolin-2,4,6-triamin (h2) and the derivatives and prodrugs thereof as antileishmanial, antiprotozoal, antiparasitic and antimicrobial agents
CN201180021289.XA CN102918051B (zh) 2010-03-16 2011-02-21 N6-(甲基二茂铁)喹唑啉-2,4,6-三胺(h2)和其衍生物,以及用作抗菌剂、抗寄生虫剂、抗原虫和抗利什曼虫剂的药物前体

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
MX2010002868A MX2010002868A (es) 2010-03-16 2010-03-16 N6-(ferrocenmetil)quinazolin-2,4,6-triamina (h2), sus derivados y profarmacos, como agentes antimicrobianos antiparasitarios, antiprotozoarios y antileishmanias.

Publications (1)

Publication Number Publication Date
MX2010002868A true MX2010002868A (es) 2011-09-21

Family

ID=44861732

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2010002868A MX2010002868A (es) 2010-03-16 2010-03-16 N6-(ferrocenmetil)quinazolin-2,4,6-triamina (h2), sus derivados y profarmacos, como agentes antimicrobianos antiparasitarios, antiprotozoarios y antileishmanias.

Country Status (6)

Country Link
US (1) US8664384B2 (es)
EP (1) EP2599783B1 (es)
CN (1) CN102918051B (es)
ES (1) ES2618367T3 (es)
MX (1) MX2010002868A (es)
WO (1) WO2011136631A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2821412A1 (en) * 2013-07-01 2015-01-07 Universität Zürich Organometallic 2-cyano-2-aminobenzoate-propyl derivates and their use as anthelmintics
JP2016533336A (ja) * 2013-09-26 2016-10-27 ウニヴェルズィテート チューリッヒ 駆虫薬として使用するためのビス−有機金属２−アミノ−３−ヒドロキシ−２−メチルプロパンニトリル誘導体
AU2014326685A1 (en) * 2013-09-26 2016-03-24 The University Of Melbourne Organometallic compounds for use as anthelmintics
CN104788503B (zh) * 2015-04-13 2017-08-08 桂林医学院 二茂铁‑喹诺酮酰胺类化合物及其制备方法和应用
CN115043886A (zh) * 2022-06-22 2022-09-13 广西民族大学 二茂铁酰胺衍生物及其合成方法和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB806772A (en) * 1956-03-29 1958-12-31 Wellcome Found Diaminoquinazolines and method of preparing
CN86100512A (zh) * 1986-02-21 1987-09-02 国家医药管理局上海医药工业研究院 有抗肿瘤作用的2，4-二氨基-6-(n-甲基或甲酰基-取代苄氨基)喹啉类衍生物合成
CN1049498A (zh) * 1989-08-16 1991-02-27 国家医药管理局上海医药工业研究院 2，4-二氨基-5-取代-6-(n-取代苄氨基)喹唑啉衍生物合成

Also Published As

Publication number Publication date
US20130109663A1 (en) 2013-05-02
ES2618367T3 (es) 2017-06-21
EP2599783A1 (en) 2013-06-05
WO2011136631A1 (es) 2011-11-03
EP2599783A4 (en) 2014-01-08
US8664384B2 (en) 2014-03-04
CN102918051B (zh) 2015-09-09
EP2599783B1 (en) 2016-12-14
CN102918051A (zh) 2013-02-06

Similar Documents

Publication Publication Date Title
MX2012011549A (es) Derivados de 3,5-difenil-isoxazolina sustituida como insecticidas y acaricidas.
MX2013002597A (es) Arilpirrolidinas pesticidas.
TW201611725A (en) Pest control agent
MY146638A (en) Insecticidal aryl isoxazoline derivatives
NZ613430A (en) Aminoindanes amides having a high fungicidal activity and their phytosanitary compositions
DK201470535A (en) Parasiticidal oral veterinary compositions comprising systemically-acting active agents, methods and uses thereof
DK2597963T3 (da) Dyrefodersammensætninger med antimikrobiel aktivitet
MX2012001787A (es) Carboxamidas como plaguicidas.
CR20130023A (es) Pirazolo[1,5-a]pirimidinas para tratamiento antiviral
MY161635A (en) Parasiticidal compositions comprising multiple active agents, methods and uses thereof
PL2836072T3 (pl) Kompozycja chwastobójcza zawierająca związek uracylowy jako składnik czynny
MD4127B1 (en) Use of di(m-S)-bis{chloro-[1-(pyridine-2-yl)ethanone-4-methylthiosemicarbazonato(1-)]copper} as substance with antimicrobial activity against Staphylococcus aureus
EP2594134A4 (en) AGROCHEMICALS WITH A 2,5-DIKETOPIPERAZINE DERIVATIVE ACTIVE SUBSTANCE
BR112012023500A2 (pt) "composições fungicidas que compreendem um micro-organismo de solubilização de fosfato e um composto ativo como fungicida"
MX349802B (es) Uso de aril- y hetarilcarboxamidas como endoparasiticidas.
UY33907A (es) Derivados de pirazol microbicidas
MX2012000955A (es) Carboxamidas pesticidas.
MX2010002868A (es) N6-(ferrocenmetil)quinazolin-2,4,6-triamina (h2), sus derivados y profarmacos, como agentes antimicrobianos antiparasitarios, antiprotozoarios y antileishmanias.
TW201204257A (en) Triazole-substituted anthranilamides as pesticides
IN2014MN02484A (es)
MX336431B (es) Derivados de azetidina como agentes antiparasitarios.
MX2013004311A (es) Compuestos antimicrobianos de polieter y poliol.
MX336430B (es) Derivados de dihidrofurano-azetadina como agentes antiparasitarios.
RU2009138209A (ru) N-замещенные амиды 2-гидрокси-4-оксо-4-(41-хлорфенил) 2-бутеновой кислоты, проявляющие противомикробную активность
EP2599493A4 (en) Antimicrobial activity enhancing agent

Legal Events

Date Code Title Description
FG Grant or registration