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MX2007009061A - Preparacion farmaceutica para la anticoncepcion oral. - Google Patents

Preparacion farmaceutica para la anticoncepcion oral.

Info

Publication number
MX2007009061A
MX2007009061A MX2007009061A MX2007009061A MX2007009061A MX 2007009061 A MX2007009061 A MX 2007009061A MX 2007009061 A MX2007009061 A MX 2007009061A MX 2007009061 A MX2007009061 A MX 2007009061A MX 2007009061 A MX2007009061 A MX 2007009061A
Authority
MX
Mexico
Prior art keywords
daily dose
ethinyl estradiol
dienogest
pharmaceutical preparation
composition
Prior art date
Application number
MX2007009061A
Other languages
English (en)
Inventor
Thomas Graser
Claus Claussen
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of MX2007009061A publication Critical patent/MX2007009061A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/567Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Una preparacion farmaceutica para la anticoncepcion oral, que contiene como primer componente de principio activo 17(-cianometil-17-(-hidroxiestra-4,9-dien-3-ona (dienogest) en una dosis diaria de 1,5 mg de dienogest y como segundo componente de principio activo 17(-etinilestradiol (etinilestradiol) en una dosis diaria de 0,015 o 0,020 mg de etinilestradiol o 2,0 mg de dienogest y 0,015 mg de etinilestradiol, se administra junto con uno o varios portadores farmaceuticamente aceptables en al menos 21 dias de un ciclo menstrual de 28 dias. Ademas, la preparacion farmaceutica contiene 7 o menos unidades de dosis diarias sin principio activo.
MX2007009061A 2005-02-15 2006-02-15 Preparacion farmaceutica para la anticoncepcion oral. MX2007009061A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05003179A EP1690543A1 (de) 2005-02-15 2005-02-15 Pharmazeutisches Präparat zur Kontrazeption
PCT/EP2006/001354 WO2006087173A1 (de) 2005-02-15 2006-02-15 Pharmazeutisches präparat zur kontrazeption

Publications (1)

Publication Number Publication Date
MX2007009061A true MX2007009061A (es) 2007-09-11

Family

ID=34933759

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2007009061A MX2007009061A (es) 2005-02-15 2006-02-15 Preparacion farmaceutica para la anticoncepcion oral.

Country Status (20)

Country Link
EP (2) EP1690543A1 (es)
JP (1) JP2008527018A (es)
KR (1) KR20070086380A (es)
CN (1) CN101119732A (es)
AR (1) AR053545A1 (es)
AU (1) AU2006215818A1 (es)
BR (1) BRPI0606724A2 (es)
CA (1) CA2590004A1 (es)
CR (1) CR9324A (es)
DO (1) DOP2006000035A (es)
EA (1) EA200701091A1 (es)
IL (1) IL183635A0 (es)
MX (1) MX2007009061A (es)
NO (1) NO20072687L (es)
PA (1) PA8663401A1 (es)
PE (1) PE20061291A1 (es)
TW (1) TW200640468A (es)
UA (1) UA85003C2 (es)
WO (1) WO2006087173A1 (es)
ZA (1) ZA200707910B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1774970A1 (de) * 2005-10-13 2007-04-18 Bayer Schering Pharma AG Verfahren zur Herstellung eines einphasigen pharmazeutischen Präparates zur Therapie der dysfunktionellen uterinen Blutung, enthaltend Ethinylestradiol und Dienogest
WO2009049813A2 (de) * 2007-10-11 2009-04-23 Bayer Schering Pharma Aktiengesellschaft Verfahren zur herstellung eines einphasischen pharmazeutischen präparates zur begrenzung/minderung des risikos einer tiefen-venen-thrombose in einheit mit einer oralen kontrazeption
EP2055306A1 (de) * 2007-11-05 2009-05-06 Bayer Schering Pharma AG Verwendung eines Gestagens in Kombination mit einem Estrogen und einem oder mehreren pharmazeutisch annehmbaren hilfsstoffen/Trägern zur laktosefreien oralen Kontrazeption

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR9710566A (pt) * 1996-07-26 1999-08-17 American Home Prod M-todo anticoncepcional monof sico e um kit compreendendo uma combina-Æo de uma progestina e estrog-nio

Also Published As

Publication number Publication date
PA8663401A1 (es) 2006-12-07
BRPI0606724A2 (pt) 2009-07-14
DOP2006000035A (es) 2006-09-15
UA85003C2 (ru) 2008-12-10
KR20070086380A (ko) 2007-08-27
ZA200707910B (en) 2009-08-26
NO20072687L (no) 2007-11-13
JP2008527018A (ja) 2008-07-24
CN101119732A (zh) 2008-02-06
EA200701091A1 (ru) 2008-02-28
TW200640468A (en) 2006-12-01
CR9324A (es) 2007-10-11
WO2006087173A1 (de) 2006-08-24
PE20061291A1 (es) 2006-12-07
AU2006215818A1 (en) 2006-08-24
EP1690543A1 (de) 2006-08-16
AR053545A1 (es) 2007-05-09
EP1853273A1 (de) 2007-11-14
CA2590004A1 (en) 2006-08-24
IL183635A0 (en) 2007-10-31

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal