MX2007004245A - Nuevos derivados de arilo azabiciclicos y su uso medico. - Google Patents
Nuevos derivados de arilo azabiciclicos y su uso medico.Info
- Publication number
- MX2007004245A MX2007004245A MX2007004245A MX2007004245A MX2007004245A MX 2007004245 A MX2007004245 A MX 2007004245A MX 2007004245 A MX2007004245 A MX 2007004245A MX 2007004245 A MX2007004245 A MX 2007004245A MX 2007004245 A MX2007004245 A MX 2007004245A
- Authority
- MX
- Mexico
- Prior art keywords
- diseases
- disorders
- aryl derivatives
- medical use
- azabicyclic aryl
- Prior art date
Links
- 125000003118 aryl group Chemical group 0.000 title abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 8
- 201000010099 disease Diseases 0.000 abstract 4
- 208000035475 disorder Diseases 0.000 abstract 4
- 210000003169 central nervous system Anatomy 0.000 abstract 2
- 230000001713 cholinergic effect Effects 0.000 abstract 2
- 210000001428 peripheral nervous system Anatomy 0.000 abstract 2
- 108010078791 Carrier Proteins Proteins 0.000 abstract 1
- 208000017701 Endocrine disease Diseases 0.000 abstract 1
- 206010061218 Inflammation Diseases 0.000 abstract 1
- 102000019315 Nicotinic acetylcholine receptors Human genes 0.000 abstract 1
- 108050006807 Nicotinic acetylcholine receptors Proteins 0.000 abstract 1
- 208000002193 Pain Diseases 0.000 abstract 1
- 208000007271 Substance Withdrawal Syndrome Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000030172 endocrine system disease Diseases 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 239000003446 ligand Substances 0.000 abstract 1
- 230000004770 neurodegeneration Effects 0.000 abstract 1
- 230000000144 pharmacologic effect Effects 0.000 abstract 1
- 102000005962 receptors Human genes 0.000 abstract 1
- 108020003175 receptors Proteins 0.000 abstract 1
- 230000016160 smooth muscle contraction Effects 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Esta invencion se relaciona con nuevos derivados de arilo azabiciclicos de la formula (1), que se encuentra que son ligandos colinergicos en los receptores de acetilcolina nicotinicos y moduladores de los receptores y transportadores de monoamina. Debido a su perfil farmacologico, los compuestos de la invencion pueden ser ??tiles para el tratamiento de las enfermedades o trastornos tan diversos como los relacionados con el sistema colinergico del sistema nervioso central (SNC), el sistema nervioso periferico (SNP), enfermedades o trastornos relacionados con contraccion del musculo liso, enfermedades o trastornos endocrinos, enfermedades O trastornos' relacionados con la neurodegeneracion, enfermedades o trastornos relacionados con inflamacion, dolor y sintomas de abstinencia causados por la terminacion del abuso de sustancias quimicas.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US61859804P | 2004-10-15 | 2004-10-15 | |
| DKPA200401582 | 2004-10-15 | ||
| PCT/EP2005/055263 WO2006040352A1 (en) | 2004-10-15 | 2005-10-14 | Novel azabicyclic aryl derivatives and their medical use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2007004245A true MX2007004245A (es) | 2007-06-12 |
Family
ID=39509634
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2007004245A MX2007004245A (es) | 2004-10-15 | 2005-10-14 | Nuevos derivados de arilo azabiciclicos y su uso medico. |
Country Status (3)
| Country | Link |
|---|---|
| JP (1) | JP2008516930A (es) |
| MX (1) | MX2007004245A (es) |
| NZ (1) | NZ553277A (es) |
-
2005
- 2005-10-14 MX MX2007004245A patent/MX2007004245A/es active IP Right Grant
- 2005-10-14 NZ NZ553277A patent/NZ553277A/en not_active IP Right Cessation
- 2005-10-14 JP JP2007536186A patent/JP2008516930A/ja not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| NZ553277A (en) | 2010-04-30 |
| JP2008516930A (ja) | 2008-05-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant or registration |