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MA41107A - Compositions anti-cancéreuses - Google Patents

Compositions anti-cancéreuses

Info

Publication number
MA41107A
MA41107A MA041107A MA41107A MA41107A MA 41107 A MA41107 A MA 41107A MA 041107 A MA041107 A MA 041107A MA 41107 A MA41107 A MA 41107A MA 41107 A MA41107 A MA 41107A
Authority
MA
Morocco
Prior art keywords
cancer compositions
cancer
compositions
Prior art date
Application number
MA041107A
Other languages
English (en)
Other versions
MA41107B1 (fr
Inventor
Dennis Martin Hester
Jason Michael Vaughn
Original Assignee
Aragon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52006906&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA41107(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aragon Pharmaceuticals Inc filed Critical Aragon Pharmaceuticals Inc
Publication of MA41107A publication Critical patent/MA41107A/fr
Publication of MA41107B1 publication Critical patent/MA41107B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1652Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682Processes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
MA41107A 2014-12-05 2015-12-03 Compositions anti-cancéreuses MA41107B1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14196594 2014-12-05
PCT/US2015/063661 WO2016090098A1 (fr) 2014-12-05 2015-12-03 Compositions anti-cancéreuses
EP15817641.2A EP3226841B1 (fr) 2014-12-05 2015-12-03 Compositions anticancéreuses

Publications (2)

Publication Number Publication Date
MA41107A true MA41107A (fr) 2017-10-10
MA41107B1 MA41107B1 (fr) 2025-01-31

Family

ID=52006906

Family Applications (1)

Application Number Title Priority Date Filing Date
MA41107A MA41107B1 (fr) 2014-12-05 2015-12-03 Compositions anti-cancéreuses

Country Status (29)

Country Link
US (3) US20170360754A1 (fr)
EP (2) EP4494636A3 (fr)
JP (2) JP6937692B2 (fr)
KR (2) KR102348320B1 (fr)
CN (2) CN114886852A (fr)
AR (1) AR102926A1 (fr)
AU (3) AU2015358490B2 (fr)
BR (1) BR112017011788A2 (fr)
CA (1) CA2969656A1 (fr)
CL (1) CL2017001371A1 (fr)
CO (1) CO2017005572A2 (fr)
CR (1) CR20170216A (fr)
EA (1) EA201791222A1 (fr)
ES (1) ES2996833T3 (fr)
HR (1) HRP20241719T1 (fr)
HU (1) HUE069689T2 (fr)
IL (2) IL252323B (fr)
MA (1) MA41107B1 (fr)
MD (1) MD3226841T2 (fr)
MX (2) MX387933B (fr)
NZ (1) NZ770528A (fr)
PH (1) PH12017500964A1 (fr)
PL (1) PL3226841T3 (fr)
RS (1) RS66323B1 (fr)
SG (1) SG11201704267VA (fr)
SM (1) SMT202400518T1 (fr)
TW (2) TWI754258B (fr)
UA (1) UA120950C2 (fr)
WO (1) WO2016090098A1 (fr)

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MX371020B (es) 2012-09-26 2020-01-13 Aragon Pharmaceuticals Inc Antiandrógenos para el tratamiento del cáncer de próstata resistente a la castración no metastásico.
US20170360754A1 (en) 2014-12-05 2017-12-21 Aragon Pharmaceuticals, Inc. Anticancer compositions
KR102387089B1 (ko) 2014-12-05 2022-04-14 아라곤 파마슈티컬스, 인코포레이티드 항암 조성물
SG11202003402QA (en) 2017-10-16 2020-05-28 Aragon Pharmaceuticals Inc Anti-androgens for the treatment of non-metastatic castration-resistant prostate cancer
WO2020144649A1 (fr) 2019-01-10 2020-07-16 Aragon Pharmaceuticals, Inc. Composition pharmaceutique comprenant de l'enzalutamide dispersé dans une compote de pomme
EP3918607A1 (fr) 2019-01-30 2021-12-08 Janssen Pharmaceutica NV Méthodes de traitement du cancer de la prostate sur la base de sous-types moléculaires
SG11202107712SA (en) 2019-01-30 2021-08-30 Aragon Pharmaceuticals Inc Anti-androgens for the treatment of metastatic castration-sensitive prostate cancer
WO2020239478A1 (fr) 2019-05-28 2020-12-03 Pharma Mar, S.A. Trabectédine pour le traitement de sarcomes basé sur des marqueurs génomiques
EP3811932A1 (fr) 2019-10-22 2021-04-28 Zentiva K.S. Forme posologique d'apalutamide
EP4054572A1 (fr) 2019-11-04 2022-09-14 Aragon Pharmaceuticals, Inc. Inhibiteurs du récepteur des androgènes pour le traitement du cancer de la prostate non métastatique résistant à la castration chez des sujets présentant une déficience hépatique grave
WO2021245285A1 (fr) 2020-06-05 2021-12-09 Janssen Pharmaceutica Nv Méthodes de traitement du cancer de la prostate sur la base de sous-types moléculaires
WO2022049523A1 (fr) 2020-09-04 2022-03-10 Aragon Pharmaceuticals, Inc. Méthodes de traitement du cancer de la prostate
WO2022195407A1 (fr) 2021-03-19 2022-09-22 Aragon Pharmaceuticals, Inc. Méthodes de traitement du cancer de la prostate
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WO2023152611A1 (fr) 2022-02-11 2023-08-17 Aragon Pharmaceuticals, Inc. Apalutamide et relugolix pour le traitement du cancer de la prostate
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KR20250157532A (ko) 2023-03-16 2025-11-04 바이엘 컨수머 케어 악티엔게젤샤프트 호르몬 감수성 전립선암의 생화학적 재발이 있는 환자의 치료를 위한 안드로겐 수용체 길항제
WO2025153768A1 (fr) * 2024-01-18 2025-07-24 Nanoform Finland Oyj Composition contenant de l'apalutamide nanométrique cristallin
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Also Published As

Publication number Publication date
EA201791222A1 (ru) 2017-09-29
MX387933B (es) 2025-03-19
TWI702966B (zh) 2020-09-01
AU2021201979A1 (en) 2021-04-29
TW201630592A (zh) 2016-09-01
CL2017001371A1 (es) 2018-01-05
CN114886852A (zh) 2022-08-12
IL252323B (en) 2021-04-29
SMT202400518T1 (it) 2025-01-14
TWI754258B (zh) 2022-02-01
EP4494636A3 (fr) 2025-04-30
CR20170216A (es) 2017-08-30
MX2017007203A (es) 2017-08-28
PH12017500964A1 (en) 2017-10-18
CN106999431B (zh) 2022-03-04
ES2996833T3 (en) 2025-02-13
CA2969656A1 (fr) 2016-06-09
AU2015358490A1 (en) 2017-06-08
BR112017011788A2 (pt) 2017-12-26
UA120950C2 (uk) 2020-03-10
MA41107B1 (fr) 2025-01-31
AR102926A1 (es) 2017-04-05
MX2021013965A (es) 2022-01-04
US20240293374A1 (en) 2024-09-05
CN106999431A (zh) 2017-08-01
US20170360754A1 (en) 2017-12-21
HUE069689T2 (hu) 2025-04-28
KR20200141533A (ko) 2020-12-18
EP4494636A2 (fr) 2025-01-22
KR20170086656A (ko) 2017-07-26
JP7174006B2 (ja) 2022-11-17
JP2017536398A (ja) 2017-12-07
EP3226841A1 (fr) 2017-10-11
NZ731963A (en) 2024-03-22
IL252323A0 (en) 2017-07-31
CO2017005572A2 (es) 2017-09-20
EP3226841B1 (fr) 2024-10-09
SG11201704267VA (en) 2017-06-29
US20230233529A1 (en) 2023-07-27
NZ770528A (en) 2024-03-22
WO2016090098A1 (fr) 2016-06-09
IL279833B (en) 2022-03-01
US12303493B2 (en) 2025-05-20
RS66323B1 (sr) 2025-01-31
PL3226841T3 (pl) 2025-03-03
TW202031248A (zh) 2020-09-01
JP6937692B2 (ja) 2021-09-22
HRP20241719T1 (hr) 2025-02-14
AU2023202710A1 (en) 2023-05-18
EP3226841C0 (fr) 2024-10-09
JP2020143069A (ja) 2020-09-10
MD3226841T2 (ro) 2025-06-30
AU2021201979B2 (en) 2023-02-02
IL279833A (en) 2021-01-31
KR102348320B1 (ko) 2022-01-10
AU2015358490B2 (en) 2021-04-08

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