MA39838B1 - Composés bicycliques hétéroaryle ou aryle fusionnés et leur utilisation en tant qu'inhibiteurs irak4 - Google Patents
Composés bicycliques hétéroaryle ou aryle fusionnés et leur utilisation en tant qu'inhibiteurs irak4Info
- Publication number
- MA39838B1 MA39838B1 MA39838A MA39838A MA39838B1 MA 39838 B1 MA39838 B1 MA 39838B1 MA 39838 A MA39838 A MA 39838A MA 39838 A MA39838 A MA 39838A MA 39838 B1 MA39838 B1 MA 39838B1
- Authority
- MA
- Morocco
- Prior art keywords
- bicyclic heteroaryl
- fused aryl
- aryl compounds
- irak4 inhibitors
- irak4
- Prior art date
Links
- 229940127590 IRAK4 inhibitor Drugs 0.000 title 1
- 125000003118 aryl group Chemical group 0.000 title 1
Classifications
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/056—Ortho-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring
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- A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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- C07C235/66—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems and singly-bound oxygen atoms, bound to the same carbon skeleton
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US201461975473P | 2014-04-04 | 2014-04-04 | |
| EP15717250.3A EP3126330B1 (fr) | 2014-04-04 | 2015-03-26 | Composés bicycliques hétéroaryle ou aryle fusionnés et leur utilisation en tant qu'inhibiteurs irak4 |
| PCT/IB2015/052251 WO2015150995A1 (fr) | 2014-04-04 | 2015-03-26 | Composés à base d'hétéroaryle ou d'aryle fusionné-bicyclique et leur utilisation comme composés inhibiteurs de l'irak 4 |
Publications (2)
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| MA39838A MA39838A (fr) | 2017-02-08 |
| MA39838B1 true MA39838B1 (fr) | 2019-05-31 |
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| MA39838A MA39838B1 (fr) | 2014-04-04 | 2015-03-26 | Composés bicycliques hétéroaryle ou aryle fusionnés et leur utilisation en tant qu'inhibiteurs irak4 |
| MA52856A MA52856B1 (fr) | 2014-04-04 | 2015-03-26 | Composés bicycliques hétéroaryle ou aryle fusionnés et leur utilisation en tant qu'inhibiteurs irak4 |
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