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MA35878B1 - Utilisation thérapeutique de dérivés d'imidazopyridine - Google Patents

Utilisation thérapeutique de dérivés d'imidazopyridine

Info

Publication number
MA35878B1
MA35878B1 MA37231A MA37231A MA35878B1 MA 35878 B1 MA35878 B1 MA 35878B1 MA 37231 A MA37231 A MA 37231A MA 37231 A MA37231 A MA 37231A MA 35878 B1 MA35878 B1 MA 35878B1
Authority
MA
Morocco
Prior art keywords
therapeutic use
imidazopyridine derivatives
phenyl ring
medicament
formulas
Prior art date
Application number
MA37231A
Other languages
English (en)
Inventor
Chantal Alcouffe
Corentin Herbert
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47630451&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA35878(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of MA35878B1 publication Critical patent/MA35878B1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

L'invention concerne l'utilisation de composés représentés par la formule (i) dans laquelle r2 et r3 forment ensemble avec les atomes de carbone du noyau phényle auquel ils sont liés un hétérocycle azoté à 6 chaînons correspondant à l'une des formules (a), (b) et (c) dans laquelle les lignes ondulées représentent le noyau phényle auquel r2 et r3 sont liés, ou d'un sel de ceux-ci pharmaceutiquement acceptable, pour préparer un médicament afin de traiter le cancer de la vessie.
MA37231A 2012-01-04 2014-07-23 Utilisation thérapeutique de dérivés d'imidazopyridine MA35878B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR1250075A FR2985185B1 (fr) 2012-01-04 2012-01-04 Utilisation en therapeutique de derives d'imidazopyridine
PCT/IB2013/050048 WO2013102860A1 (fr) 2012-01-04 2013-01-03 Utilisation thérapeutique de dérivés d'imidazopyridine

Publications (1)

Publication Number Publication Date
MA35878B1 true MA35878B1 (fr) 2014-12-01

Family

ID=47630451

Family Applications (1)

Application Number Title Priority Date Filing Date
MA37231A MA35878B1 (fr) 2012-01-04 2014-07-23 Utilisation thérapeutique de dérivés d'imidazopyridine

Country Status (24)

Country Link
US (1) US9732078B2 (fr)
EP (1) EP2800566B1 (fr)
JP (1) JP6067032B2 (fr)
KR (1) KR102046196B1 (fr)
CN (1) CN104144687B (fr)
AU (1) AU2013207082B2 (fr)
BR (1) BR112014016632A8 (fr)
CA (1) CA2860413C (fr)
CL (1) CL2014001784A1 (fr)
CO (1) CO7020916A2 (fr)
EA (1) EA027058B1 (fr)
ES (1) ES2560619T3 (fr)
FR (1) FR2985185B1 (fr)
HK (1) HK1198690A1 (fr)
IL (1) IL233493A (fr)
MA (1) MA35878B1 (fr)
MX (1) MX336340B (fr)
PH (1) PH12014501537A1 (fr)
PL (1) PL2800566T3 (fr)
SG (1) SG11201403793UA (fr)
TW (1) TWI557122B (fr)
UY (1) UY34564A (fr)
WO (1) WO2013102860A1 (fr)
ZA (1) ZA201404928B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2994141A4 (fr) * 2013-05-10 2016-11-23 Nimbus Apollo Inc Inhibiteurs de l'acc et utilisations associées
KR102627756B1 (ko) * 2017-03-22 2024-01-23 쑤저우 바이지부공 파마수티컬 테크널러지 컴퍼니 리미티드 브루톤 타이로신 키나제 억제제
CN115490687B (zh) * 2022-09-19 2023-10-27 国家烟草质量监督检验中心 3-苯并呋喃基硫咪唑并吡啶衍生物及其制备方法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2859997B1 (fr) 2003-09-18 2006-02-03 Sanofi Synthelabo Nouveaux derives d'indolizine 1,2,3,6,7,8 substituee, inhibiteurs des fgfs, leur procede de preparation et les compositions pharmaceutiques les contenant.
FR2883286B1 (fr) * 2005-03-16 2008-10-03 Sanofi Aventis Sa NOUVEAUX DERIVES D'IMIDAZO[1,5-a]PYRIDINES, INHIBITEURS DE FGFs, LEUR PROCEDE DE PREPARATION ET LES COMPOSITIONS PHARMACEUTIQUES LES CONTENANT
FR2896247B1 (fr) * 2006-01-13 2008-02-29 Sanofi Aventis Sa Composes dimeres agonistes des recepteurs des fgfs (fgfrs), leur procede de preparation et leur application en therapeutique
EP1891955A1 (fr) 2006-07-24 2008-02-27 Sanofi-Aventis Utilisation de dérivés de indolizines, inhibiteurs de FGF, pour la préparation d'un médicament pour le traitement d'affections dégénératives des articulations
CN1887878A (zh) 2006-07-26 2007-01-03 浙江大学 三嗪氮氧化物及合成方法和用途
FR2962437B1 (fr) * 2010-07-06 2012-08-17 Sanofi Aventis Derives d'imidazopyridine, leur procede de preparation et leur application en therapeutique

Also Published As

Publication number Publication date
CN104144687B (zh) 2017-09-05
CA2860413A1 (fr) 2013-07-11
CL2014001784A1 (es) 2014-10-17
UY34564A (es) 2013-09-02
EP2800566B1 (fr) 2015-10-28
PL2800566T3 (pl) 2016-04-29
US9732078B2 (en) 2017-08-15
EA027058B1 (ru) 2017-06-30
IL233493A (en) 2017-02-28
CO7020916A2 (es) 2014-08-11
HK1198690A1 (en) 2015-05-29
EA201491307A1 (ru) 2014-11-28
JP6067032B2 (ja) 2017-01-25
AU2013207082B2 (en) 2017-06-15
BR112014016632A8 (pt) 2017-07-04
AU2013207082A1 (en) 2014-07-31
TW201333008A (zh) 2013-08-16
MX2014008244A (es) 2014-11-25
ZA201404928B (en) 2015-10-28
MX336340B (es) 2016-01-15
SG11201403793UA (en) 2014-08-28
ES2560619T3 (es) 2016-02-22
IL233493A0 (en) 2014-08-31
PH12014501537A1 (en) 2014-10-08
FR2985185B1 (fr) 2013-12-27
CN104144687A (zh) 2014-11-12
FR2985185A1 (fr) 2013-07-05
BR112014016632A2 (pt) 2017-06-13
KR20140107667A (ko) 2014-09-04
KR102046196B1 (ko) 2019-11-18
TWI557122B (zh) 2016-11-11
US20140343054A1 (en) 2014-11-20
CA2860413C (fr) 2020-02-25
WO2013102860A1 (fr) 2013-07-11
EP2800566A1 (fr) 2014-11-12
JP2015505311A (ja) 2015-02-19

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