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MA28634B1 - Dérivés de phénol et thiophénol 3-ou 4-monosubstitués utiles comme ligands de H3 - Google Patents

Dérivés de phénol et thiophénol 3-ou 4-monosubstitués utiles comme ligands de H3

Info

Publication number
MA28634B1
MA28634B1 MA29438A MA29438A MA28634B1 MA 28634 B1 MA28634 B1 MA 28634B1 MA 29438 A MA29438 A MA 29438A MA 29438 A MA29438 A MA 29438A MA 28634 B1 MA28634 B1 MA 28634B1
Authority
MA
Morocco
Prior art keywords
ligands
derivatives useful
thiophenol derivatives
monosubstituted phenol
monosubstituted
Prior art date
Application number
MA29438A
Other languages
English (en)
Inventor
Patrick Bernardelli
Andrew Michael Cronin
Alexis Denis
Stephen Martin Denton
Henry Jacobelli
Mark Ian Kemp
Edwige Lorthiois
Fiona Rousseau
Delphine Serradeil-Civit
Fabrice Vergne
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP04291187A external-priority patent/EP1593679A1/fr
Priority claimed from GB0504564A external-priority patent/GB0504564D0/en
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of MA28634B1 publication Critical patent/MA28634B1/fr

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    • C07D309/04—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D309/06—Radicals substituted by oxygen atoms
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MA29438A 2004-05-07 2006-11-07 Dérivés de phénol et thiophénol 3-ou 4-monosubstitués utiles comme ligands de H3 MA28634B1 (fr)

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EP04291187A EP1593679A1 (fr) 2004-05-07 2004-05-07 Dérivés de phénol 3- ou 4-monosubstitués utiles comme ligands de H3
GB0504564A GB0504564D0 (en) 2005-03-04 2005-03-04 New compounds

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JP5813101B2 (ja) 2010-06-04 2015-11-17 アルバニー モレキュラー リサーチ， インコーポレイテッド グリシントランスポーター−１阻害剤、その作製方法および使用方法
WO2012037258A1 (fr) 2010-09-16 2012-03-22 Abbott Laboratories Procédés de préparation de dérivés cyclopropyliques substitués en 1,2
KR101586966B1 (ko) * 2011-10-26 2016-01-19 화이자 리미티드 나트륨 채널 조절제로서 유용한 (4-페닐이미다졸-2-일) 에틸아민 유도체
WO2014095534A1 (fr) * 2012-12-19 2014-06-26 Basf Se Nouveaux triazoles et imidazoles substitués et leur utilisation en tant que fongicides
JP6253668B2 (ja) * 2013-01-09 2017-12-27 アリーナ ファーマシューティカルズ， インコーポレイテッド 認識障害の処置のためのヒスタミンｈ３受容体調節因子としてのビフェニル−エチル−ピロリジン誘導体
TWI731317B (zh) * 2013-12-10 2021-06-21 美商健臻公司 原肌球蛋白相關之激酶（ｔｒｋ）抑制劑
JP6606183B2 (ja) 2014-12-18 2019-11-13 ジェンザイム・コーポレーション トロポミオシン関連キナーゼ（ｔｒｋ）阻害剤の医薬製剤
CN113336715B (zh) * 2021-08-04 2021-11-23 山东海利尔化工有限公司 一种含二氧戊环的三唑类化合物及其中间体的制备方法

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