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MA28554B1 - Dérivés de morpholine - Google Patents

Dérivés de morpholine

Info

Publication number
MA28554B1
MA28554B1 MA29417A MA29417A MA28554B1 MA 28554 B1 MA28554 B1 MA 28554B1 MA 29417 A MA29417 A MA 29417A MA 29417 A MA29417 A MA 29417A MA 28554 B1 MA28554 B1 MA 28554B1
Authority
MA
Morocco
Prior art keywords
morpholine derivatives
morpholine
derivatives
Prior art date
Application number
MA29417A
Other languages
English (en)
Inventor
Paul Vincent Fish
Malcolm Christian Mackenny
Alan Stobie
Florian Wakenhut
Gavin Alistair Whitlock
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32482498&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA28554(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of MA28554B1 publication Critical patent/MA28554B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Obesity (AREA)
  • Pulmonology (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Immunology (AREA)
  • Pregnancy & Childbirth (AREA)
MA29417A 2004-04-30 2006-10-30 Dérivés de morpholine MA28554B1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0409744.0A GB0409744D0 (en) 2004-04-30 2004-04-30 Novel compounds

Publications (1)

Publication Number Publication Date
MA28554B1 true MA28554B1 (fr) 2007-04-03

Family

ID=32482498

Family Applications (1)

Application Number Title Priority Date Filing Date
MA29417A MA28554B1 (fr) 2004-04-30 2006-10-30 Dérivés de morpholine

Country Status (33)

Country Link
US (3) US20050250775A1 (fr)
EP (1) EP1744754A1 (fr)
JP (2) JP4181622B2 (fr)
KR (4) KR20090006888A (fr)
CN (1) CN1950089A (fr)
AP (1) AP2006003767A0 (fr)
AR (1) AR048934A1 (fr)
AU (1) AU2005237301A1 (fr)
BR (1) BRPI0510515A (fr)
CA (1) CA2564990C (fr)
CR (1) CR8717A (fr)
DO (1) DOP2005000064A (fr)
EA (1) EA200601802A1 (fr)
EC (1) ECSP066958A (fr)
GB (1) GB0409744D0 (fr)
GE (1) GEP20084549B (fr)
GT (1) GT200500098A (fr)
IL (1) IL178313A0 (fr)
MA (1) MA28554B1 (fr)
MX (1) MXPA06012640A (fr)
NI (1) NI200600257A (fr)
NL (1) NL1028927C2 (fr)
NO (1) NO20064282L (fr)
NZ (1) NZ550054A (fr)
PA (1) PA8631601A1 (fr)
PE (1) PE20060305A1 (fr)
SV (1) SV2005002099A (fr)
TN (1) TNSN06347A1 (fr)
TW (2) TW200914431A (fr)
UA (1) UA86970C2 (fr)
UY (1) UY28873A1 (fr)
WO (1) WO2005105100A1 (fr)
ZA (1) ZA200608661B (fr)

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AP2006003771A0 (en) * 2004-04-30 2006-10-31 Warner Lambert Co Substituted morpholine compounds for the treatmentof central nervous system disorders
GB0409744D0 (en) * 2004-04-30 2004-06-09 Pfizer Ltd Novel compounds
WO2007062336A2 (fr) * 2005-11-18 2007-05-31 Astrazeneca Ab Formes de sels
EP1951257A4 (fr) * 2005-11-18 2008-11-05 Astrazeneca Ab Formes cristallines
WO2007062339A2 (fr) * 2005-11-18 2007-05-31 Astrazeneca Ab Formulations liquides
US8389510B2 (en) * 2005-11-18 2013-03-05 Astrazeneca Ab Crystalline forms
EP1951693A4 (fr) * 2005-11-18 2012-05-30 Astrazeneca Ab Formulations solides
AU2007209903B2 (en) * 2006-02-01 2012-09-13 Merck Sharp & Dohme Corp. Potassium channel inhibitors
EP1892530A1 (fr) * 2006-08-25 2008-02-27 Boehringer Ingelheim Pharma GmbH & Co. KG Procédé de détermination de l'activité de transport d'une protéine de transport
KR101103118B1 (ko) * 2007-11-02 2012-01-04 동아제약주식회사 신규한 1,3-디히드로-5-이소벤조퓨란카르보니트릴 유도체 화합물 및 이를 함유하는 조루증 치료용 약학조성물
EP2318362B1 (fr) * 2008-07-24 2013-09-25 Theravance, Inc. Composés de 3-(phénoxyphénylméthyl)pyrrolidine
WO2010085589A2 (fr) 2009-01-22 2010-07-29 G&H Brands Llc Produit médicamenteux désensibilisateur
WO2010120910A1 (fr) * 2009-04-15 2010-10-21 Theravance, Inc. Composés 3-(phénoxypyrrolidin-3-yl-méthyle) hétéroaryle, 3-(phénylpyrrolidin-3-ylméthoxy) hétéroaryle, et 3-(hétéroarylpyrrolidin-3-ylméthoxy) hétéroaryle
US7994209B2 (en) 2009-07-13 2011-08-09 Theravance, Inc. 3-phenoxymethylpyrrolidine compounds
WO2011011231A1 (fr) 2009-07-21 2011-01-27 Theravance, Inc. Composés de la 3-phénoxyméthylpyrrolidine
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