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Blazer et al., 2010 - Google Patents

Reversible, allosteric small-molecule inhibitors of regulator of G protein signaling proteins

Blazer et al., 2010

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Document ID
2482772195226194347
Author
Blazer L
Roman D
Chung A
Larsen M
Greedy B
Husbands S
Neubig R
Publication year
Publication venue
Molecular pharmacology

External Links

Snippet

Regulators of G protein signaling (RGS) proteins are potent negative modulators of G protein signaling and have been proposed as potential targets for small-molecule inhibitor development. We report a high-throughput time-resolved fluorescence resonance energy …
Continue reading at pmc.ncbi.nlm.nih.gov (PDF) (other versions)

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