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CHEN et al., 2013 - Google Patents

as pure agonists (eg, morphine, hydromorphone, meperidine, fen-tanyl, methadone, levorphanol, oxycodone) or agonist-antagonists (eg, pentazocine, dezocine …

CHEN et al., 2013

Document ID
88686666072245696
Author
CHEN L
COHEN S
MAO J
Publication year
Publication venue
Managing Pain: Essentials of Diagnosis and Treatment

External Links

Snippet

Opioids act on three major classes of endogenous receptors to achieve their analgesic effects: μ, κ, and 8 (mu, kappa, and delta receptors). These receptors are widely distributed throughout the body, including in the central and peripheral nervous systems, as well as …
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Classifications

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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    • A61K31/445—Non condensed piperidines, e.g. piperocaine
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
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    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
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