UA48989C2 - Похідні 1-арилсульфоніл, арил(тіо)карбонілпіридазину, спосіб їх одержання, фармацевтична композиція та спосіб лікування - Google Patents
Похідні 1-арилсульфоніл, арил(тіо)карбонілпіридазину, спосіб їх одержання, фармацевтична композиція та спосіб лікуванняInfo
- Publication number
- UA48989C2 UA48989C2 UA98052267A UA98052267A UA48989C2 UA 48989 C2 UA48989 C2 UA 48989C2 UA 98052267 A UA98052267 A UA 98052267A UA 98052267 A UA98052267 A UA 98052267A UA 48989 C2 UA48989 C2 UA 48989C2
- Authority
- UA
- Ukraine
- Prior art keywords
- derivatives
- carbonylpyridazine
- arylsulfonyl
- thio
- aryl
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- 125000003118 aryl group Chemical group 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- RJKFOVLPORLFTN-LEKSSAKUSA-N Progesterone Chemical class C1CC2=CC(=O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H](C(=O)C)[C@@]1(C)CC2 RJKFOVLPORLFTN-LEKSSAKUSA-N 0.000 abstract 2
- 239000000583 progesterone congener Substances 0.000 abstract 2
- 201000009273 Endometriosis Diseases 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 230000000708 anti-progestin effect Effects 0.000 abstract 1
- 239000003418 antiprogestin Substances 0.000 abstract 1
- 125000005129 aryl carbonyl group Chemical group 0.000 abstract 1
- 210000000988 bone and bone Anatomy 0.000 abstract 1
- 210000000481 breast Anatomy 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 150000002391 heterocyclic compounds Chemical class 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 238000000338 in vitro Methods 0.000 abstract 1
- 230000009245 menopause Effects 0.000 abstract 1
- 210000004291 uterus Anatomy 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/26—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/06—Antiabortive agents; Labour repressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/26—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
- C07D237/36—Benzo-cinnolines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Physical Education & Sports Medicine (AREA)
- Reproductive Health (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Gynecology & Obstetrics (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Pregnancy & Childbirth (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US790095P | 1995-11-06 | 1995-11-06 | |
| PCT/US1996/016227 WO1997017332A1 (en) | 1995-11-06 | 1996-10-10 | 1-arylsulphonyl, aryl(thio)carbonyl pyridazino derivatives and methods of preparation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA48989C2 true UA48989C2 (uk) | 2002-09-16 |
Family
ID=21728709
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UA98052267A UA48989C2 (uk) | 1995-11-06 | 1996-10-10 | Похідні 1-арилсульфоніл, арил(тіо)карбонілпіридазину, спосіб їх одержання, фармацевтична композиція та спосіб лікування |
Country Status (17)
| Country | Link |
|---|---|
| JP (1) | JP2000501073A (zh) |
| KR (1) | KR100360614B1 (zh) |
| CN (1) | CN1110485C (zh) |
| AU (1) | AU704507B2 (zh) |
| BR (1) | BR9611407A (zh) |
| CZ (1) | CZ286789B6 (zh) |
| HU (1) | HU225162B1 (zh) |
| IL (1) | IL124320A (zh) |
| MX (1) | MX9803605A (zh) |
| NO (1) | NO310460B1 (zh) |
| NZ (1) | NZ319979A (zh) |
| PL (1) | PL185618B1 (zh) |
| RU (1) | RU2175969C2 (zh) |
| TW (1) | TW460467B (zh) |
| UA (1) | UA48989C2 (zh) |
| WO (1) | WO1997017332A1 (zh) |
| ZA (1) | ZA969298B (zh) |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4816467A (en) * | 1987-01-09 | 1989-03-28 | Farmitalia Carlo Erba S.R.L | Heteroaryl 3-oxo-propanenitrile derivatives, pharmaceutical compositions and use |
| WO1989004306A1 (fr) * | 1987-11-02 | 1989-05-18 | Yoshitomi Pharmaceutical Industries, Ltd. | Composes de pyridazine fusionnes et leurs utilisations medicales |
| WO1993004069A1 (fr) * | 1991-08-27 | 1993-03-04 | Yoshitomi Pharmaceutical Industries, Ltd. | Compose de pyridazine lie par fusion et utilisation pharmaceutique d'un tel compose |
-
1996
- 1996-10-10 NZ NZ319979A patent/NZ319979A/xx unknown
- 1996-10-10 JP JP9518177A patent/JP2000501073A/ja not_active Ceased
- 1996-10-10 PL PL96326669A patent/PL185618B1/pl not_active IP Right Cessation
- 1996-10-10 IL IL12432096A patent/IL124320A/en not_active IP Right Cessation
- 1996-10-10 WO PCT/US1996/016227 patent/WO1997017332A1/en not_active Ceased
- 1996-10-10 UA UA98052267A patent/UA48989C2/uk unknown
- 1996-10-10 RU RU98110813/04A patent/RU2175969C2/ru not_active IP Right Cessation
- 1996-10-10 AU AU72637/96A patent/AU704507B2/en not_active Ceased
- 1996-10-10 CZ CZ19981380A patent/CZ286789B6/cs not_active IP Right Cessation
- 1996-10-10 CN CN96199481A patent/CN1110485C/zh not_active Expired - Fee Related
- 1996-10-10 BR BR9611407-0A patent/BR9611407A/pt not_active Application Discontinuation
- 1996-10-10 KR KR10-1998-0703345A patent/KR100360614B1/ko not_active Expired - Fee Related
- 1996-10-10 HU HU0201305A patent/HU225162B1/hu not_active IP Right Cessation
- 1996-11-05 ZA ZA9609298A patent/ZA969298B/xx unknown
- 1996-11-25 TW TW085114479A patent/TW460467B/zh not_active IP Right Cessation
-
1998
- 1998-05-05 NO NO19982030A patent/NO310460B1/no unknown
- 1998-05-06 MX MX9803605A patent/MX9803605A/es not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| PL326669A1 (en) | 1998-10-12 |
| HUP0201305A3 (en) | 2003-02-28 |
| NO310460B1 (no) | 2001-07-09 |
| CZ286789B6 (en) | 2000-07-12 |
| BR9611407A (pt) | 1999-12-28 |
| CN1207091A (zh) | 1999-02-03 |
| IL124320A0 (en) | 1998-12-06 |
| TW460467B (en) | 2001-10-21 |
| ZA969298B (en) | 1998-05-05 |
| AU7263796A (en) | 1997-05-29 |
| CN1110485C (zh) | 2003-06-04 |
| HUP0201305A2 (hu) | 2002-12-28 |
| KR19990067340A (ko) | 1999-08-16 |
| CZ138098A3 (cs) | 1998-09-16 |
| IL124320A (en) | 2001-10-31 |
| RU2175969C2 (ru) | 2001-11-20 |
| NO982030D0 (no) | 1998-05-05 |
| KR100360614B1 (ko) | 2003-06-02 |
| PL185618B1 (pl) | 2003-06-30 |
| NO982030L (no) | 1998-06-23 |
| AU704507B2 (en) | 1999-04-22 |
| HU225162B1 (en) | 2006-07-28 |
| MX9803605A (es) | 1998-09-30 |
| JP2000501073A (ja) | 2000-02-02 |
| WO1997017332A1 (en) | 1997-05-15 |
| NZ319979A (en) | 1999-11-29 |
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