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PE20030136A1 - BIOADHESIVE TABLETS FOR PROGRESSIVE HYDRATION - Google Patents

BIOADHESIVE TABLETS FOR PROGRESSIVE HYDRATION

Info

Publication number
PE20030136A1
PE20030136A1 PE2001000582A PE2001000582A PE20030136A1 PE 20030136 A1 PE20030136 A1 PE 20030136A1 PE 2001000582 A PE2001000582 A PE 2001000582A PE 2001000582 A PE2001000582 A PE 2001000582A PE 20030136 A1 PE20030136 A1 PE 20030136A1
Authority
PE
Peru
Prior art keywords
water
progressive hydration
polymer
composition
sponged
Prior art date
Application number
PE2001000582A
Other languages
Spanish (es)
Inventor
William J Bologna
Howard L Levine
Ziegler Dominique De
Original Assignee
Columbia Lab Bermuda Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/877,218 external-priority patent/US6624200B2/en
Application filed by Columbia Lab Bermuda Ltd filed Critical Columbia Lab Bermuda Ltd
Publication of PE20030136A1 publication Critical patent/PE20030136A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

SE REFIERE A UNA COMPOSICION FARMACEUTICA BIOADHESIVA PARA HIDRATACION PROGRESIVA QUE COMPRENDE: a) UNA CANTIDAD EFECTIVA DE TESTOSTERONA; b) UN POLIMERO POLICARBOXILICO INSOLUBLE, DEGRADABLE QUE SE PUEDE ESPONJAR CON AGUA COMO POLICARBOFIL; c) UN POLIMERO HIDROSOLUBLE (CARBOMERO 974P) . LA TESTOSTERONA ESTA PRESENTE EN 30 mg POR DOSIS UNITARIA DE LA COMPOSICION. SE REFIERE TAMBIEN A UNA COMPOSICION QUE COMPRENDE TERBUTALINA, UN POLIMERO POLICARBOXILICO INSOLUBLE DEGRADABLE QUE SE PUEDE ESPONJAR CON AGUA Y UN POLIMERO HIDROSOLUBLEIT REFERS TO A BIOADHESIVE PHARMACEUTICAL COMPOSITION FOR PROGRESSIVE HYDRATION INCLUDING: a) AN EFFECTIVE AMOUNT OF TESTOSTERONE; b) AN INSOLUBLE, DEGRADABLE POLYCARBOXYL POLYMER THAT CAN BE SPONGED WITH WATER AS POLYCARBOFIL; c) A WATER-SOLUBLE POLYMER (CARBOMER 974P). TESTOSTERONE IS PRESENT IN 30 mg PER UNIT DOSE OF THE COMPOSITION. IT ALSO REFERS TO A COMPOSITION INCLUDING TERBUTALIN, A DEGRADABLE INSOLUBLE POLYCARBOXYL POLYMER THAT CAN BE SPONGED WITH WATER AND A WATER-SOLUBLE POLYMER

PE2001000582A 2000-06-16 2001-06-15 BIOADHESIVE TABLETS FOR PROGRESSIVE HYDRATION PE20030136A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US59607300A 2000-06-16 2000-06-16
US09/877,218 US6624200B2 (en) 1998-08-25 2001-06-11 Bioadhesive progressive hydration tablets

Publications (1)

Publication Number Publication Date
PE20030136A1 true PE20030136A1 (en) 2003-03-18

Family

ID=24385886

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2001000582A PE20030136A1 (en) 2000-06-16 2001-06-15 BIOADHESIVE TABLETS FOR PROGRESSIVE HYDRATION

Country Status (4)

Country Link
CO (1) CO5270003A1 (en)
PE (1) PE20030136A1 (en)
TW (2) TWI311916B (en)
ZA (1) ZA200104935B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI554708B (en) 2015-11-11 2016-10-21 宣明智 Affixation Element for Micro Devices and Micro Devices

Also Published As

Publication number Publication date
TWI311916B (en) 2009-07-11
TWI319987B (en) 2010-02-01
ZA200104935B (en) 2002-12-11
CO5270003A1 (en) 2003-04-30

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