PE20030136A1 - BIOADHESIVE TABLETS FOR PROGRESSIVE HYDRATION - Google Patents
BIOADHESIVE TABLETS FOR PROGRESSIVE HYDRATIONInfo
- Publication number
- PE20030136A1 PE20030136A1 PE2001000582A PE2001000582A PE20030136A1 PE 20030136 A1 PE20030136 A1 PE 20030136A1 PE 2001000582 A PE2001000582 A PE 2001000582A PE 2001000582 A PE2001000582 A PE 2001000582A PE 20030136 A1 PE20030136 A1 PE 20030136A1
- Authority
- PE
- Peru
- Prior art keywords
- water
- progressive hydration
- polymer
- composition
- sponged
- Prior art date
Links
- 239000000227 bioadhesive Substances 0.000 title abstract 2
- 230000036571 hydration Effects 0.000 title abstract 2
- 238000006703 hydration reaction Methods 0.000 title abstract 2
- 230000000750 progressive effect Effects 0.000 title abstract 2
- MUMGGOZAMZWBJJ-DYKIIFRCSA-N Testostosterone Chemical compound O=C1CC[C@]2(C)[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CCC2=C1 MUMGGOZAMZWBJJ-DYKIIFRCSA-N 0.000 abstract 4
- 239000000203 mixture Substances 0.000 abstract 2
- 229920000642 polymer Polymers 0.000 abstract 2
- 229960003604 testosterone Drugs 0.000 abstract 2
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 2
- 229920003169 water-soluble polymer Polymers 0.000 abstract 2
- XWTYSIMOBUGWOL-UHFFFAOYSA-N (+-)-Terbutaline Chemical compound CC(C)(C)NCC(O)C1=CC(O)=CC(O)=C1 XWTYSIMOBUGWOL-UHFFFAOYSA-N 0.000 abstract 1
- 229940031663 carbomer-974p Drugs 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 229960000195 terbutaline Drugs 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
SE REFIERE A UNA COMPOSICION FARMACEUTICA BIOADHESIVA PARA HIDRATACION PROGRESIVA QUE COMPRENDE: a) UNA CANTIDAD EFECTIVA DE TESTOSTERONA; b) UN POLIMERO POLICARBOXILICO INSOLUBLE, DEGRADABLE QUE SE PUEDE ESPONJAR CON AGUA COMO POLICARBOFIL; c) UN POLIMERO HIDROSOLUBLE (CARBOMERO 974P) . LA TESTOSTERONA ESTA PRESENTE EN 30 mg POR DOSIS UNITARIA DE LA COMPOSICION. SE REFIERE TAMBIEN A UNA COMPOSICION QUE COMPRENDE TERBUTALINA, UN POLIMERO POLICARBOXILICO INSOLUBLE DEGRADABLE QUE SE PUEDE ESPONJAR CON AGUA Y UN POLIMERO HIDROSOLUBLEIT REFERS TO A BIOADHESIVE PHARMACEUTICAL COMPOSITION FOR PROGRESSIVE HYDRATION INCLUDING: a) AN EFFECTIVE AMOUNT OF TESTOSTERONE; b) AN INSOLUBLE, DEGRADABLE POLYCARBOXYL POLYMER THAT CAN BE SPONGED WITH WATER AS POLYCARBOFIL; c) A WATER-SOLUBLE POLYMER (CARBOMER 974P). TESTOSTERONE IS PRESENT IN 30 mg PER UNIT DOSE OF THE COMPOSITION. IT ALSO REFERS TO A COMPOSITION INCLUDING TERBUTALIN, A DEGRADABLE INSOLUBLE POLYCARBOXYL POLYMER THAT CAN BE SPONGED WITH WATER AND A WATER-SOLUBLE POLYMER
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US59607300A | 2000-06-16 | 2000-06-16 | |
| US09/877,218 US6624200B2 (en) | 1998-08-25 | 2001-06-11 | Bioadhesive progressive hydration tablets |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20030136A1 true PE20030136A1 (en) | 2003-03-18 |
Family
ID=24385886
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2001000582A PE20030136A1 (en) | 2000-06-16 | 2001-06-15 | BIOADHESIVE TABLETS FOR PROGRESSIVE HYDRATION |
Country Status (4)
| Country | Link |
|---|---|
| CO (1) | CO5270003A1 (en) |
| PE (1) | PE20030136A1 (en) |
| TW (2) | TWI311916B (en) |
| ZA (1) | ZA200104935B (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI554708B (en) | 2015-11-11 | 2016-10-21 | 宣明智 | Affixation Element for Micro Devices and Micro Devices |
-
2001
- 2001-03-15 TW TW090106120A patent/TWI311916B/en not_active IP Right Cessation
- 2001-06-14 TW TW090114486A patent/TWI319987B/en not_active IP Right Cessation
- 2001-06-15 CO CO01048291A patent/CO5270003A1/en not_active Application Discontinuation
- 2001-06-15 ZA ZA200104935A patent/ZA200104935B/en unknown
- 2001-06-15 PE PE2001000582A patent/PE20030136A1/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| TWI311916B (en) | 2009-07-11 |
| TWI319987B (en) | 2010-02-01 |
| ZA200104935B (en) | 2002-12-11 |
| CO5270003A1 (en) | 2003-04-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC | Refusal |