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IL147803A0 - 28-epirapalogs - Google Patents

28-epirapalogs

Info

Publication number
IL147803A0
IL147803A0 IL14780300A IL14780300A IL147803A0 IL 147803 A0 IL147803 A0 IL 147803A0 IL 14780300 A IL14780300 A IL 14780300A IL 14780300 A IL14780300 A IL 14780300A IL 147803 A0 IL147803 A0 IL 147803A0
Authority
IL
Israel
Prior art keywords
epirapalogs
epirapamycin
analogs
disclosed
methods
Prior art date
Application number
IL14780300A
Other languages
English (en)
Original Assignee
Ariad Gene Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ariad Gene Therapeutics Inc filed Critical Ariad Gene Therapeutics Inc
Publication of IL147803A0 publication Critical patent/IL147803A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K48/00—Medicinal preparations containing genetic material which is inserted into cells of the living body to treat genetic diseases; Gene therapy
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12N—MICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N9/00—Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
    • C12N9/10—Transferases (2.)
    • C12N9/12—Transferases (2.) transferring phosphorus containing groups, e.g. kinases (2.7)
    • C12N9/1205—Phosphotransferases with an alcohol group as acceptor (2.7.1), e.g. protein kinases
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K2319/00—Fusion polypeptide

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Zoology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Wood Science & Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Microbiology (AREA)
  • General Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Transplantation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Peptides Or Proteins (AREA)
  • Saccharide Compounds (AREA)
IL14780300A 1999-08-24 2000-08-24 28-epirapalogs IL147803A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US15044799P 1999-08-24 1999-08-24
PCT/US2000/023334 WO2001014387A1 (en) 1999-08-24 2000-08-24 28-epirapalogs

Publications (1)

Publication Number Publication Date
IL147803A0 true IL147803A0 (en) 2002-08-14

Family

ID=22534571

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14780300A IL147803A0 (en) 1999-08-24 2000-08-24 28-epirapalogs
IL147803A IL147803A (en) 1999-08-24 2002-01-23 28-epi-rapamycin derivatives, their preparation, pharmaceutical compositions containing them and preparation of compositions for in vitro and pharmaceutical applications

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL147803A IL147803A (en) 1999-08-24 2002-01-23 28-epi-rapamycin derivatives, their preparation, pharmaceutical compositions containing them and preparation of compositions for in vitro and pharmaceutical applications

Country Status (10)

Country Link
US (1) US7196192B2 (zh)
EP (1) EP1212331B1 (zh)
CN (1) CN1293081C (zh)
AT (1) ATE264863T1 (zh)
AU (1) AU783158B2 (zh)
CA (1) CA2383451A1 (zh)
DE (1) DE60010098T2 (zh)
ES (1) ES2219388T3 (zh)
IL (2) IL147803A0 (zh)
WO (1) WO2001014387A1 (zh)

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* Cited by examiner, † Cited by third party
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