IL111008A0 - Rapamycin formulations for intraveneous injection and their preparation - Google Patents
Rapamycin formulations for intraveneous injection and their preparationInfo
- Publication number
- IL111008A0 IL111008A0 IL11100894A IL11100894A IL111008A0 IL 111008 A0 IL111008 A0 IL 111008A0 IL 11100894 A IL11100894 A IL 11100894A IL 11100894 A IL11100894 A IL 11100894A IL 111008 A0 IL111008 A0 IL 111008A0
- Authority
- IL
- Israel
- Prior art keywords
- preparation
- intraveneous injection
- rapamycin formulations
- rapamycin
- formulations
- Prior art date
Links
- 238000009472 formulation Methods 0.000 title 1
- 238000002347 injection Methods 0.000 title 1
- 239000007924 injection Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
- ZAHRKKWIAAJSAO-UHFFFAOYSA-N rapamycin Natural products COCC(O)C(=C/C(C)C(=O)CC(OC(=O)C1CCCCN1C(=O)C(=O)C2(O)OC(CC(OC)C(=CC=CC=CC(C)CC(C)C(=O)C)C)CCC2C)C(C)CC3CCC(O)C(C3)OC)C ZAHRKKWIAAJSAO-UHFFFAOYSA-N 0.000 title 1
- QFJCIRLUMZQUOT-HPLJOQBZSA-N sirolimus Chemical compound C1C[C@@H](O)[C@H](OC)C[C@@H]1C[C@@H](C)[C@H]1OC(=O)[C@@H]2CCCCN2C(=O)C(=O)[C@](O)(O2)[C@H](C)CC[C@H]2C[C@H](OC)/C(C)=C/C=C/C=C/[C@@H](C)C[C@@H](C)C(=O)[C@H](OC)[C@H](O)/C(C)=C/[C@@H](C)C(=O)C1 QFJCIRLUMZQUOT-HPLJOQBZSA-N 0.000 title 1
- 229960002930 sirolimus Drugs 0.000 title 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US12952693A | 1993-09-30 | 1993-09-30 | |
| US08/302,190 US5616588A (en) | 1993-09-30 | 1994-09-12 | Rapamycin formulation for IV injection |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL111008A0 true IL111008A0 (en) | 1994-11-28 |
| IL111008A IL111008A (en) | 1999-10-28 |
Family
ID=26827650
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL11100894A IL111008A (en) | 1993-09-30 | 1994-09-19 | Rapamycin formulations for intravenous injection and their preparation |
Country Status (6)
| Country | Link |
|---|---|
| JP (1) | JP3584064B2 (en) |
| CN (1) | CN1109748A (en) |
| BR (1) | BR9403945A (en) |
| CA (1) | CA2133180A1 (en) |
| IL (1) | IL111008A (en) |
| TW (1) | TW438586B (en) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2001253824A (en) * | 2000-03-14 | 2001-09-18 | Mitsukazu Matsumoto | Formulated agent for local injection |
| KR101131794B1 (en) * | 2002-07-30 | 2012-03-30 | 와이어쓰 엘엘씨 | A CCI-779 cosolvent concentrate, a parenteral CCI-779 formulation, and a process for preparing a parenteral CCI-779 formulation |
| US20080096972A1 (en) * | 2004-07-30 | 2008-04-24 | Thitiwan Buranachokpaisan | Compound formulations of 2-amino-1, 3-propanediol compounds |
| CN1919194A (en) * | 2006-08-17 | 2007-02-28 | 刘瑜玲 | Liquid composition of sirolimus |
| CN109431997B (en) * | 2018-12-20 | 2021-06-04 | 武汉科福新药有限责任公司 | Local rapamycin injection and preparation method thereof |
-
1994
- 1994-09-19 IL IL11100894A patent/IL111008A/en active IP Right Grant
- 1994-09-26 TW TW83108922A patent/TW438586B/en not_active IP Right Cessation
- 1994-09-28 CA CA 2133180 patent/CA2133180A1/en not_active Abandoned
- 1994-09-29 BR BR9403945A patent/BR9403945A/en not_active Application Discontinuation
- 1994-09-29 JP JP23487494A patent/JP3584064B2/en not_active Expired - Fee Related
- 1994-09-29 CN CN 94116781 patent/CN1109748A/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| TW438586B (en) | 2001-06-07 |
| CA2133180A1 (en) | 1995-03-31 |
| CN1109748A (en) | 1995-10-11 |
| BR9403945A (en) | 1995-06-13 |
| JP3584064B2 (en) | 2004-11-04 |
| JPH07196507A (en) | 1995-08-01 |
| IL111008A (en) | 1999-10-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed | ||
| HCA | Change of name of proprietor(s) after amalgamation | ||
| KB | Patent renewed |