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HK1172325B - 新型fxr(nr1h4)结合和活性调节化合物 - Google Patents

新型fxr(nr1h4)结合和活性调节化合物 Download PDF

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Publication number
HK1172325B
HK1172325B HK12113083.7A HK12113083A HK1172325B HK 1172325 B HK1172325 B HK 1172325B HK 12113083 A HK12113083 A HK 12113083A HK 1172325 B HK1172325 B HK 1172325B
Authority
HK
Hong Kong
Prior art keywords
cyclopropyl
compound
mmol
phenyl
solution
Prior art date
Application number
HK12113083.7A
Other languages
German (de)
English (en)
French (fr)
Other versions
HK1172325A1 (zh
Inventor
Claus Kremoser
Ulrich Abel
Christoph Steeneck
Olaf Kinzel
Original Assignee
Gilead Sciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP09010676A external-priority patent/EP2289883A1/en
Application filed by Gilead Sciences, Inc. filed Critical Gilead Sciences, Inc.
Publication of HK1172325A1 publication Critical patent/HK1172325A1/zh
Publication of HK1172325B publication Critical patent/HK1172325B/zh

Links

HK12113083.7A 2009-08-19 2010-08-19 新型fxr(nr1h4)结合和活性调节化合物 HK1172325B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US23511709P 2009-08-19 2009-08-19
EP09010676A EP2289883A1 (en) 2009-08-19 2009-08-19 Novel FXR (NR1H4) binding and activity modulating compounds
EP09010676.6 2009-08-19
US61/235,117 2009-08-19
PCT/EP2010/005093 WO2011020615A1 (en) 2009-08-19 2010-08-19 Novel fxr (nr1h4 ) binding and activity modulating compounds

Publications (2)

Publication Number Publication Date
HK1172325A1 HK1172325A1 (zh) 2013-04-19
HK1172325B true HK1172325B (zh) 2015-09-18

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