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FI811857L - Nya 2beta 16beta-dipiperidino -5 alfa-androstan bis-och monokvaternaera ammoniumderivat foerfarande foer deras framstaellning och farmaceutiska produkter - Google Patents

Nya 2beta 16beta-dipiperidino -5 alfa-androstan bis-och monokvaternaera ammoniumderivat foerfarande foer deras framstaellning och farmaceutiska produkter

Info

Publication number
FI811857L
FI811857L FI811857A FI811857A FI811857L FI 811857 L FI811857 L FI 811857L FI 811857 A FI811857 A FI 811857A FI 811857 A FI811857 A FI 811857A FI 811857 L FI811857 L FI 811857L
Authority
FI
Finland
Prior art keywords
och
monoquaternaera
16beta
dipiperidino
2beta
Prior art date
Application number
FI811857A
Other languages
English (en)
Other versions
FI66394C (fi
FI66394B (fi
Inventor
Jan Kelder
Original Assignee
Akzo Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nv filed Critical Akzo Nv
Publication of FI811857L publication Critical patent/FI811857L/fi
Application granted granted Critical
Publication of FI66394B publication Critical patent/FI66394B/fi
Publication of FI66394C publication Critical patent/FI66394C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
FI811857A 1979-12-12 1981-06-15 Foerfarande foer framstaellning av nya biskvaternaera ammoniumderivat av 2beta 16beta-dipiperidino-5alfa-androstaner FI66394C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB7942883 1979-12-12
GB7942883 1979-12-12
EP8000143 1980-12-09
PCT/EP1980/000143 WO1981001710A1 (fr) 1979-12-12 1980-12-09 Mono et bis piperidinium androstanes

Publications (3)

Publication Number Publication Date
FI811857L true FI811857L (fi) 1981-06-15
FI66394B FI66394B (fi) 1984-06-29
FI66394C FI66394C (fi) 1984-10-10

Family

ID=10509800

Family Applications (1)

Application Number Title Priority Date Filing Date
FI811857A FI66394C (fi) 1979-12-12 1981-06-15 Foerfarande foer framstaellning av nya biskvaternaera ammoniumderivat av 2beta 16beta-dipiperidino-5alfa-androstaner

Country Status (12)

Country Link
US (1) US4348390A (fi)
EP (1) EP0032261B1 (fi)
JP (1) JPH026360B2 (fi)
AU (1) AU534992B2 (fi)
CA (1) CA1153366A (fi)
DE (1) DE3065088D1 (fi)
DK (1) DK158741C (fi)
ES (1) ES8204443A1 (fi)
FI (1) FI66394C (fi)
HU (1) HU185865B (fi)
IE (1) IE50675B1 (fi)
WO (1) WO1981001710A1 (fi)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE53463B1 (en) * 1981-06-15 1988-11-23 Akzo Nv Mono-and bisquaternary ammonium derivatives of 2 beta,16 beta-d-amino-5 alpha-androstane derivatives and pharmaceutical preparations containing same
US4726275A (en) * 1983-05-10 1988-02-23 Synthaxe Limited Electronic musical instrument
US5418226A (en) * 1992-04-22 1995-05-23 Akzo N.V. Monoquaternary 2,16-bispiperidinylandrostane derivatives
US5926516A (en) * 1995-05-24 1999-07-20 Siemens Aktiengesellschaft Absorption structure for absorbing neutrons and method for producing an absorption structure
IT1277700B1 (it) * 1995-12-22 1997-11-11 Poli Ind Chimica Spa Processo di preparazione di 2-beta, 16-beta-diamino 3-alfa, 17-beta- diacilossi 5-alfaandrostani, bloccanti neuromuscolari a struttura
US5990124A (en) 1997-10-24 1999-11-23 Gyermek; Laszlo Neuromuscular relaxants
CN116925171B (zh) * 2023-07-10 2025-06-27 时森海(杭州)医药科技有限公司 含环丙甲基甾体类季铵盐化合物、中间体及其制备方法和应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1138605A (en) * 1965-02-19 1969-01-01 Organon Labor Ltd Improvements in or relating to new 2-ß,16-ß-diamino-androstanes
GB1454749A (en) * 1972-11-29 1976-11-03 Akzo Nv 2beta, 16beta-diamino-androstanes and their preparation
HU172522B (hu) * 1975-08-01 1978-09-28 Richter Gedeon Vegyeszet Sposob poluchenija novykh proizvodnykh 2beta, 16beta-diamino-androstana i ikh chetvertichnykh solej
EP0008824B1 (en) * 1978-09-05 1982-04-28 Akzo N.V. Acid addition salts of 16-beta-monoquaternary ammonium derivatives of 2-beta, 16-beta-bis-piperidino-androstanes and pharmaceutical preparations containing same

Also Published As

Publication number Publication date
JPS56501761A (fi) 1981-12-03
AU6640581A (en) 1981-07-06
DE3065088D1 (en) 1983-11-03
IE50675B1 (en) 1986-06-11
WO1981001710A1 (fr) 1981-06-25
IE802566L (en) 1981-06-12
US4348390A (en) 1982-09-07
FI66394C (fi) 1984-10-10
JPH026360B2 (fi) 1990-02-08
DK158741C (da) 1990-11-26
DK158741B (da) 1990-07-09
EP0032261B1 (en) 1983-09-28
HU185865B (en) 1985-04-28
DK260881A (da) 1981-06-25
AU534992B2 (en) 1984-02-23
ES497724A0 (es) 1982-05-01
ES8204443A1 (es) 1982-05-01
FI66394B (fi) 1984-06-29
CA1153366A (en) 1983-09-06
EP0032261A1 (en) 1981-07-22

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: AKZO N.V.