CU20100125A7 - BIS- (SULFONYLAMINE) DERIVATIVES FOR USE IN THERAPY - Google Patents
BIS- (SULFONYLAMINE) DERIVATIVES FOR USE IN THERAPYInfo
- Publication number
- CU20100125A7 CU20100125A7 CU20100125A CU20100125A CU20100125A7 CU 20100125 A7 CU20100125 A7 CU 20100125A7 CU 20100125 A CU20100125 A CU 20100125A CU 20100125 A CU20100125 A CU 20100125A CU 20100125 A7 CU20100125 A7 CU 20100125A7
- Authority
- CU
- Cuba
- Prior art keywords
- therapy
- sulfonylamine
- bis
- derivatives
- formula
- Prior art date
Links
- 238000002560 therapeutic procedure Methods 0.000 title abstract 2
- QECVIPBZOPUTRD-UHFFFAOYSA-N N=S(=O)=O Chemical class N=S(=O)=O QECVIPBZOPUTRD-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 102100033076 Prostaglandin E synthase Human genes 0.000 abstract 1
- 101710096361 Prostaglandin E synthase Proteins 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000003287 optical effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La invención proporciona compuestos de fórmula (I): ESPACIO PARA LA FÓRMULA donde R1, R3, L1, L2, G1, G2, A y m son como se definió en la descripción e isómeros ópticos, racematos y tautómeros de los mismos, y sales farmacéuticamente aceptables de los mismos; junto con procesos para su preparación, composiciones farmacéuticas que los contienen y su uso en terapia. Los compuestos son inhibidores de la prostaglandina E sintasa-1 microsomal.The invention provides compounds of formula (I): SPACE FOR THE FORMULA where R1, R3, L1, L2, G1, G2, A and m are as defined in the description and optical isomers, racemates and tautomers thereof, and pharmaceutically salts acceptable thereof; together with processes for its preparation, pharmaceutical compositions containing them and their use in therapy. The compounds are microsomal prostaglandin E synthase-1 inhibitors.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20100125A CU20100125A7 (en) | 2010-06-18 | 2010-06-18 | BIS- (SULFONYLAMINE) DERIVATIVES FOR USE IN THERAPY |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20100125A CU20100125A7 (en) | 2010-06-18 | 2010-06-18 | BIS- (SULFONYLAMINE) DERIVATIVES FOR USE IN THERAPY |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CU20100125A7 true CU20100125A7 (en) | 2011-10-14 |
Family
ID=45000103
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CU20100125A CU20100125A7 (en) | 2010-06-18 | 2010-06-18 | BIS- (SULFONYLAMINE) DERIVATIVES FOR USE IN THERAPY |
Country Status (1)
| Country | Link |
|---|---|
| CU (1) | CU20100125A7 (en) |
-
2010
- 2010-06-18 CU CU20100125A patent/CU20100125A7/en unknown
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