BRPI0819957A2 - "composição farmacêutica estável e sustentada de hidrocloreto de bupropiona e processo para a preparação da mesma" - Google Patents
"composição farmacêutica estável e sustentada de hidrocloreto de bupropiona e processo para a preparação da mesma"Info
- Publication number
- BRPI0819957A2 BRPI0819957A2 BRPI0819957A BRPI0819957A BRPI0819957A2 BR PI0819957 A2 BRPI0819957 A2 BR PI0819957A2 BR PI0819957 A BRPI0819957 A BR PI0819957A BR PI0819957 A BRPI0819957 A BR PI0819957A BR PI0819957 A2 BRPI0819957 A2 BR PI0819957A2
- Authority
- BR
- Brazil
- Prior art keywords
- preparing
- stable
- pharmaceutical composition
- bupropion hydrochloride
- sustained pharmaceutical
- Prior art date
Links
- IKBZAUYPBWFMDI-UHFFFAOYSA-N 5-bromo-4-methoxy-7-methyl-2,3-dihydro-1h-indene Chemical group C1=C(Br)C(OC)=C2CCCC2=C1C IKBZAUYPBWFMDI-UHFFFAOYSA-N 0.000 title 1
- 229960004367 bupropion hydrochloride Drugs 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 230000002459 sustained effect Effects 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Emergency Medicine (AREA)
- Pain & Pain Management (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN117DE2008 | 2008-01-14 | ||
| PCT/IN2008/000777 WO2009090670A2 (en) | 2008-01-14 | 2008-11-19 | Stabilized sustained release composition of bupropion hydrochloride and process for preparing the same |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0819957A2 true BRPI0819957A2 (pt) | 2015-09-15 |
Family
ID=54291754
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0819957A BRPI0819957A2 (pt) | 2008-01-14 | 2008-11-19 | "composição farmacêutica estável e sustentada de hidrocloreto de bupropiona e processo para a preparação da mesma" |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20100291225A1 (pt) |
| EP (1) | EP2229053A4 (pt) |
| KR (1) | KR20100107044A (pt) |
| AU (1) | AU2008347949A1 (pt) |
| BR (1) | BRPI0819957A2 (pt) |
| CA (1) | CA2713365A1 (pt) |
| MX (1) | MX2010007672A (pt) |
| RU (1) | RU2010133982A (pt) |
| WO (1) | WO2009090670A2 (pt) |
| ZA (1) | ZA201004830B (pt) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US12194006B2 (en) | 2013-11-05 | 2025-01-14 | Antecip Bioventures Ii Llc | Bupropion as a modulator of drug activity |
| US12109178B2 (en) | 2013-11-05 | 2024-10-08 | Antecip Bioventures Ii Llc | Bupropion as a modulator of drug activity |
| US11433067B2 (en) | 2013-11-05 | 2022-09-06 | Antecip Bioventures Ii Llc | Bupropion as a modulator of drug activity |
| US11534414B2 (en) | 2013-11-05 | 2022-12-27 | Antecip Bioventures Ii Llc | Bupropion as a modulator of drug activity |
| US11969421B2 (en) | 2013-11-05 | 2024-04-30 | Antecip Bioventures Ii Llc | Bupropion as a modulator of drug activity |
| US9687475B1 (en) | 2016-03-24 | 2017-06-27 | Ezra Pharma Llc | Extended release pharmaceutical formulations with controlled impurity levels |
| US9675585B1 (en) * | 2016-03-24 | 2017-06-13 | Ezra Pharma | Extended release pharmaceutical formulations |
| US12433884B2 (en) | 2020-06-05 | 2025-10-07 | Antecip Bioventures Ii Llc | Compounds and combinations thereof for treating neurological and psychiatric conditions |
| US12472156B2 (en) | 2020-06-05 | 2025-11-18 | Antecip Bioventures Ii Llc | Compounds and combinations thereof for treating neurological and psychiatric conditions |
| KR102536511B1 (ko) * | 2020-06-25 | 2023-05-26 | (주) 넥스팜코리아 | 날트렉손 서방형 매트릭스 제제와 부프로피온 서방형 매트릭스 제제의 단층정 복합제제와 그 제조 방법 |
| WO2022119981A1 (en) | 2020-12-01 | 2022-06-09 | Antecip Bioventures Ii Llc | Bupropion and dextromethrophan for reduction of suicide risk in depression patients |
| US11717518B1 (en) | 2022-06-30 | 2023-08-08 | Antecip Bioventures Ii Llc | Bupropion dosage forms with reduced food and alcohol dosing effects |
| US12156914B2 (en) | 2022-06-30 | 2024-12-03 | Axsome Therapeutics, Inc. | Pharmaceutical compositions comprising bupropion and cysteine |
| US20240000729A1 (en) * | 2022-06-30 | 2024-01-04 | Axsome Therapeutics, Inc. | Microparticles containing bupropion |
| US12036191B1 (en) | 2022-06-30 | 2024-07-16 | Antecip Bioventures Ii Llc | Treatment of poor metabolizers of dextromethorphan with a combination of bupropion and dextromethorphan |
| US11730706B1 (en) | 2022-07-07 | 2023-08-22 | Antecip Bioventures Ii Llc | Treatment of depression in certain patient populations |
| US11844797B1 (en) | 2023-04-20 | 2023-12-19 | Antecip Bioventures Ii Llc | Combination of dextromethorphan and bupropion for treating depression |
| US12194036B2 (en) | 2022-07-07 | 2025-01-14 | Antecip Bioventures Ii Llc | Combination of dextromethorphan and bupropion for treating depression |
| CN117224495A (zh) * | 2023-11-03 | 2023-12-15 | 迪沙药业集团有限公司 | 一种盐酸安非他酮缓释制剂及其制备方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6337328B1 (en) * | 1999-03-01 | 2002-01-08 | Sepracor, Inc. | Bupropion metabolites and methods of use |
| US6306436B1 (en) * | 2000-04-28 | 2001-10-23 | Teva Pharmaceuticals Usa, Inc. | Stabilized, acid-free formulation for sustained release of bupropion hydrochloride |
| NZ544281A (en) * | 2003-08-08 | 2008-07-31 | Biovail Lab Int Srl | Modified-release tablet of bupropion hydrochloride |
| WO2005065308A2 (en) * | 2003-12-29 | 2005-07-21 | Jason Mcdevitt | Compositions and methods to treat recurrent medical conditions |
| US20060204571A1 (en) * | 2005-03-12 | 2006-09-14 | Sun Pharmaceutical Industries Limited | Stable compositions of bupropion or its pharmaceutically acceptable salts |
| US7884136B2 (en) * | 2005-06-27 | 2011-02-08 | Biovail Laboratories International S.R.L. | Modified-release formulations of a bupropion salt |
| WO2008023390A2 (en) * | 2006-08-21 | 2008-02-28 | Jubilant Organosys Limited | Modified release pharmaceutical composition of bupropion hydrochloride |
| WO2010004386A2 (en) * | 2008-06-16 | 2010-01-14 | Glenmark Generics Limited | Amorphous bupropion hydrobromide and preparation thereof |
-
2008
- 2008-11-09 US US12/812,693 patent/US20100291225A1/en not_active Abandoned
- 2008-11-19 BR BRPI0819957A patent/BRPI0819957A2/pt not_active IP Right Cessation
- 2008-11-19 KR KR1020107018010A patent/KR20100107044A/ko not_active Withdrawn
- 2008-11-19 EP EP08870575A patent/EP2229053A4/en not_active Withdrawn
- 2008-11-19 MX MX2010007672A patent/MX2010007672A/es not_active Application Discontinuation
- 2008-11-19 AU AU2008347949A patent/AU2008347949A1/en not_active Abandoned
- 2008-11-19 CA CA2713365A patent/CA2713365A1/en not_active Abandoned
- 2008-11-19 RU RU2010133982/13A patent/RU2010133982A/ru not_active Application Discontinuation
- 2008-11-19 WO PCT/IN2008/000777 patent/WO2009090670A2/en not_active Ceased
-
2010
- 2010-07-08 ZA ZA2010/04830A patent/ZA201004830B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009090670A3 (en) | 2009-12-30 |
| MX2010007672A (es) | 2010-10-07 |
| RU2010133982A (ru) | 2012-02-27 |
| WO2009090670A8 (en) | 2009-09-11 |
| ZA201004830B (en) | 2011-03-30 |
| US20100291225A1 (en) | 2010-11-18 |
| EP2229053A2 (en) | 2010-09-22 |
| CA2713365A1 (en) | 2009-07-23 |
| WO2009090670A2 (en) | 2009-07-23 |
| AU2008347949A1 (en) | 2009-07-23 |
| EP2229053A4 (en) | 2011-01-12 |
| KR20100107044A (ko) | 2010-10-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application fees: application dismissed [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 4A, 5A, 6A E 7A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2344 DE 08-12-2015 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |