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BR9607374A - Processo para sintetizar um composto j. - Google Patents

Processo para sintetizar um composto j.

Info

Publication number
BR9607374A
BR9607374A BR9607374A BR9607374A BR9607374A BR 9607374 A BR9607374 A BR 9607374A BR 9607374 A BR9607374 A BR 9607374A BR 9607374 A BR9607374 A BR 9607374A BR 9607374 A BR9607374 A BR 9607374A
Authority
BR
Brazil
Prior art keywords
synthesizing
compound
Prior art date
Application number
BR9607374A
Other languages
English (en)
Inventor
David Askin
Steven J Cianciosi
Robert S Hoerrner
Original Assignee
Usmerck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Usmerck & Co Inc filed Critical Usmerck & Co Inc
Publication of BR9607374A publication Critical patent/BR9607374A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
BR9607374A 1995-03-15 1996-03-11 Processo para sintetizar um composto j. BR9607374A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/404,776 US5508404A (en) 1995-03-15 1995-03-15 Reductive amination process
PCT/US1996/002646 WO1996028440A1 (en) 1995-03-15 1996-03-11 REDUCTIVE ALKYLATION PROCESS FOR THE PREPARATION N-(2-(R)-HYDROXY-1-(S)-INDANYL)-2(R)-PHENYLMETHYL-4(S)-HYDROXY-5-(1-(4-(3-PYRIDYLMETHYL)-2(S)-N'-(t-BUTYLCARBOXAMIDO)-PIPERAZINYL))-PENTANEAMIDE (=COMPOUND J OR L-735,524)

Publications (1)

Publication Number Publication Date
BR9607374A true BR9607374A (pt) 1997-12-30

Family

ID=23600989

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9607374A BR9607374A (pt) 1995-03-15 1996-03-11 Processo para sintetizar um composto j.

Country Status (13)

Country Link
US (1) US5508404A (pt)
EP (1) EP0815102A1 (pt)
CN (1) CN1183780A (pt)
AR (1) AR001153A1 (pt)
AU (1) AU5175196A (pt)
BR (1) BR9607374A (pt)
CZ (1) CZ291035B6 (pt)
EA (1) EA000635B1 (pt)
HR (1) HRP960113A2 (pt)
SK (1) SK122797A3 (pt)
TW (1) TW349947B (pt)
WO (1) WO1996028440A1 (pt)
YU (1) YU15596A (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6576664B1 (en) * 1997-08-18 2003-06-10 Bristol-Myers Squibb Pharma Company Inhibitors of aggrecanase and matrix metalloproteinases for the treatment of arthritis
US7199240B2 (en) * 2002-12-11 2007-04-03 Merck & Co., Inc. Reductive alkylation of saturated cyclic amines

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB705979A (en) * 1951-03-22 1954-03-24 Henri Morren 1.4-aralkyl piperazines and process for the preparation thereof
JPS57106681A (en) * 1980-12-24 1982-07-02 Dainippon Pharmaceut Co Ltd 1,8-naphthyridine derivative and its salt
ES2112880T3 (es) * 1991-11-08 1998-04-16 Merck & Co Inc Inhibidores de la proteasa de vih utiles para el tratamiento del sida.

Also Published As

Publication number Publication date
US5508404A (en) 1996-04-16
YU15596A (sh) 1999-07-28
EA199700234A1 (ru) 1998-04-30
CZ291035B6 (cs) 2002-12-11
WO1996028440A1 (en) 1996-09-19
HRP960113A2 (en) 1997-10-31
CN1183780A (zh) 1998-06-03
TW349947B (en) 1999-01-11
AR001153A1 (es) 1997-09-24
SK122797A3 (en) 1998-03-04
EA000635B1 (ru) 1999-12-29
EP0815102A1 (en) 1998-01-07
AU5175196A (en) 1996-10-02
CZ286497A3 (cs) 1998-02-18

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Legal Events

Date Code Title Description
EG Technical examination (opinion): publication of technical examination (opinion)
FC Decision: refusal