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NO874834L - Fremgangsmaate for fremstilling av terapeutisk aktive tienopyridinoner. - Google Patents

Fremgangsmaate for fremstilling av terapeutisk aktive tienopyridinoner.

Info

Publication number
NO874834L
NO874834L NO874834A NO874834A NO874834L NO 874834 L NO874834 L NO 874834L NO 874834 A NO874834 A NO 874834A NO 874834 A NO874834 A NO 874834A NO 874834 L NO874834 L NO 874834L
Authority
NO
Norway
Prior art keywords
formula
compounds
mixture
methyl
prepared
Prior art date
Application number
NO874834A
Other languages
English (en)
Norwegian (no)
Other versions
NO874834D0 (no
Inventor
Roy Victor Davies
Original Assignee
Boots Co Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boots Co Plc filed Critical Boots Co Plc
Publication of NO874834D0 publication Critical patent/NO874834D0/no
Publication of NO874834L publication Critical patent/NO874834L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Liquid Crystal Substances (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Pyridine Compounds (AREA)
NO874834A 1986-11-20 1987-11-19 Fremgangsmaate for fremstilling av terapeutisk aktive tienopyridinoner. NO874834L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868627698A GB8627698D0 (en) 1986-11-20 1986-11-20 Therapeutic agents

Publications (2)

Publication Number Publication Date
NO874834D0 NO874834D0 (no) 1987-11-19
NO874834L true NO874834L (no) 1988-05-24

Family

ID=10607612

Family Applications (1)

Application Number Title Priority Date Filing Date
NO874834A NO874834L (no) 1986-11-20 1987-11-19 Fremgangsmaate for fremstilling av terapeutisk aktive tienopyridinoner.

Country Status (24)

Country Link
US (1) US4877793A (es)
EP (1) EP0269295B1 (es)
JP (1) JPS63141984A (es)
KR (1) KR880006247A (es)
CN (1) CN1019491B (es)
AT (1) ATE64736T1 (es)
AU (1) AU599721B2 (es)
DD (1) DD282690A5 (es)
DE (1) DE3771039D1 (es)
DK (1) DK599887A (es)
ES (1) ES2038188T3 (es)
FI (1) FI875020A7 (es)
GB (1) GB8627698D0 (es)
GR (1) GR3002500T3 (es)
HU (1) HU198060B (es)
IL (1) IL84505A (es)
JO (1) JO1520B1 (es)
MX (1) MX9428A (es)
NO (1) NO874834L (es)
NZ (1) NZ222554A (es)
PH (1) PH23293A (es)
PL (1) PL149617B1 (es)
PT (1) PT86115B (es)
ZA (1) ZA878306B (es)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8726950D0 (en) * 1987-11-18 1987-12-23 Boots Co Plc Chemical process
NZ230711A (en) * 1988-09-23 1990-10-26 Ortho Pharma Corp Substituted thienopyrans as antihypertensive agents
US5026700A (en) * 1989-05-16 1991-06-25 Merrell Dow Pharmaceuticals Certain quinolines and thienopyridines as excitatory amino acid antagonists
ZA903588B (en) * 1989-05-16 1991-02-27 Merrell Dow Pharma Excitatory amino acid antagonists
US5219864A (en) * 1991-03-12 1993-06-15 Kyowa Hakko Kogyo Co., Ltd. Thienopyridine derivatives
JP2699794B2 (ja) * 1992-03-12 1998-01-19 三菱化学株式会社 チエノ〔３，２−ｂ〕ピリジン誘導体
DE4227747A1 (de) * 1992-08-21 1994-02-24 Basf Ag Heteroaromatisch kondensierte Hydroxypyridoncarbonsäureamide, deren Herstellung und Verwendung
RU2150470C1 (ru) * 1994-04-19 2000-06-10 Такеда Кемикал Индастриз Лтд. Бициклические производные тиофена, способ их получения и композиция на их основе
AU5509099A (en) * 1998-08-03 2000-02-28 Basf Corporation Pyridinones for the treatment of sexual dysfunction
US6458804B1 (en) 2001-01-26 2002-10-01 R.T. Alamo Venturesi, Llc Methods for the treatment of central nervous system disorders in certain patient groups
US6451813B1 (en) 2001-01-26 2002-09-17 R. T. Alamo Ventures I, Llc Treatment of gastroparesis in certain patient groups
US6562838B2 (en) * 2001-01-26 2003-05-13 R. T. Alamo Ventures I, L.L.C. Treatment of cardiovascular disease with quinolinone enantiomers
US8329924B2 (en) 2001-06-11 2012-12-11 Vertex Pharmaceuticals (Canada) Incorporated Compounds and methods for the treatment or prevention of Flavivirus infections
EA007484B1 (ru) 2001-06-11 2006-10-27 Вирокем Фарма Инк. Соединения и способы лечения или предупреждения инфекций flavivirus
WO2003020728A1 (en) 2001-08-30 2003-03-13 Pharmacia & Upjohn Company 4-THIOXO-4,7-DIHYDRO-THIENO[2,3-b]PYRIDINE-5-CARBOTHIOAMIDES AS ANTIVIRAL AGENTS
AR038294A1 (es) 2002-01-14 2005-01-12 Upjohn Co Oxotieno(3,2-b)piridincarboxamidas como agentes antivirales
AR038118A1 (es) 2002-01-14 2004-12-29 Upjohn Co Compuestos derivados de la bencinamida del acido 7-oxo-4,7-dihidrotien[2,3-b[piridin-6-carboxilico 3-sustituido que son utiles como antivirales
AR038117A1 (es) 2002-01-14 2004-12-29 Upjohn Co Agentes antivirales derivados de la 4- oxo-4,7 -dihidrofuro [2,3-b]piridin-5-carboxamida
US7402608B2 (en) 2002-12-10 2008-07-22 Virochem Pharma Inc. Compounds and methods for the treatment or prevention of Flavivirus infections
BRPI0610283A2 (pt) 2005-05-13 2010-10-19 Virochem Pharma Inc composto, uso do mesmo na preparação de um medicamento para o tratamento ou prevenção de uma infecção por vìrus de hepatite c, composição farmacêutica e combinação farmacêutica
JP2008093872A (ja) * 2006-10-09 2008-04-24 Kouritsu Kogyo:Kk 表示装置
CN101568538B (zh) 2006-11-15 2012-09-05 Viro化学制药公司 用于治疗或预防黄病毒属感染的噻吩类似物
EP2280952B1 (en) * 2008-05-05 2012-06-27 Merck Patent GmbH Thienopyridone derivatives as amp-activated protein kinase (ampk) activators
CN103517936A (zh) * 2011-04-27 2014-01-15 巴斯夫欧洲公司 基于二噻吩并吡啶酮共聚物的半导体材料
KR102604900B1 (ko) * 2017-05-11 2023-11-21 브리스톨-마이어스 스큅 컴퍼니 Irak4 억제제로서 유용한 티에노피리딘 및 벤조티오펜

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3903095A (en) * 1972-02-18 1975-09-02 Merck & Co Inc Certain substituted-thieno{8 3,2-c{9 -pyridines
US3997545A (en) * 1973-07-23 1976-12-14 Takeda Chemical Industries, Ltd. Thienopyridine-carboxylic acid derivatives
NZ193167A (en) * 1979-03-27 1984-08-24 Boots Co Plc Quinoline derivatives and pharmaceutical compositions
JPS5742690A (en) * 1980-08-28 1982-03-10 Kanebo Ltd Thieno 3,2-b pyridinecarboxylic acid derivative
IE51542B1 (en) * 1980-09-26 1987-01-07 Boots Co Ltd Therapeutic agents
EP0126970A3 (en) * 1983-04-27 1985-11-06 Beecham Group Plc Anxiolytic and anti-depressant thienopyridine derivatives
PT79031B (en) * 1983-08-20 1986-08-22 Boots Co Plc Therapeutic agents
US4552884A (en) * 1984-01-13 1985-11-12 The Boots Company Plc Method of treating heart disease
GB2161524B (en) * 1984-07-13 1988-01-06 Pandrol Ltd Improvements in or relating to rail pads and rail assemblies including such pads
DE3576686D1 (de) * 1984-08-15 1990-04-26 Boots Co Ltd Chinolinone, verfahren zu ihrer herstellung und die sie enthaltenden pharmazeutischen praeparate.
GB8515209D0 (en) * 1985-06-15 1985-07-17 Boots Co Plc Therapeutic agents
GB8515207D0 (en) * 1985-06-15 1985-07-17 Boots Co Plc Therapeutic agents

Also Published As

Publication number Publication date
PT86115B (pt) 1990-08-31
JPS63141984A (ja) 1988-06-14
AU599721B2 (en) 1990-07-26
NO874834D0 (no) 1987-11-19
HU198060B (en) 1989-07-28
ATE64736T1 (de) 1991-07-15
EP0269295B1 (en) 1991-06-26
AU8144087A (en) 1988-05-26
NZ222554A (en) 1989-08-29
ES2038188T3 (es) 1993-07-16
PL149617B1 (en) 1990-03-31
CN1019491B (zh) 1992-12-16
DK599887D0 (da) 1987-11-16
PT86115A (en) 1987-12-01
US4877793A (en) 1989-10-31
IL84505A (en) 1990-12-23
GB8627698D0 (en) 1986-12-17
JO1520B1 (en) 1989-01-25
DK599887A (da) 1988-05-21
FI875020L (fi) 1988-05-21
FI875020A0 (fi) 1987-11-13
MX9428A (es) 1993-10-01
EP0269295A1 (en) 1988-06-01
FI875020A7 (fi) 1988-05-21
CN87107975A (zh) 1988-06-01
GR3002500T3 (en) 1992-12-30
PL268925A1 (en) 1988-09-01
DD282690A5 (de) 1990-09-19
ZA878306B (en) 1988-05-02
DE3771039D1 (de) 1991-08-01
KR880006247A (ko) 1988-07-22
HUT47289A (en) 1989-02-28
PH23293A (en) 1989-06-30

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