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MX2008010804A - Derivados de rapamicina para tratar neuroblastoma. - Google Patents

Derivados de rapamicina para tratar neuroblastoma.

Info

Publication number
MX2008010804A
MX2008010804A MX2008010804A MX2008010804A MX2008010804A MX 2008010804 A MX2008010804 A MX 2008010804A MX 2008010804 A MX2008010804 A MX 2008010804A MX 2008010804 A MX2008010804 A MX 2008010804A MX 2008010804 A MX2008010804 A MX 2008010804A
Authority
MX
Mexico
Prior art keywords
rapamycin derivatives
treating neuroblastoma
neuroblastoma
treating
rapamycin
Prior art date
Application number
MX2008010804A
Other languages
English (en)
Inventor
Hans Schaller
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MX2008010804A publication Critical patent/MX2008010804A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Un derivado de rapamicina para uso en el tratamiento de neuroblastoma, opcionalmente en combinación con una segunda sustancia de fármaco.
MX2008010804A 2006-02-24 2007-02-22 Derivados de rapamicina para tratar neuroblastoma. MX2008010804A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0603782.4A GB0603782D0 (en) 2006-02-24 2006-02-24 Organic compounds
PCT/EP2007/001551 WO2007096174A1 (en) 2006-02-24 2007-02-22 Rapamycin derivatives for treating neuroblastoma

Publications (1)

Publication Number Publication Date
MX2008010804A true MX2008010804A (es) 2008-10-31

Family

ID=36178746

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2008010804A MX2008010804A (es) 2006-02-24 2007-02-22 Derivados de rapamicina para tratar neuroblastoma.

Country Status (12)

Country Link
US (1) US20090023768A1 (es)
EP (1) EP1988894A1 (es)
JP (1) JP2009527520A (es)
KR (1) KR20080100346A (es)
CN (1) CN101389337A (es)
AU (1) AU2007217705A1 (es)
BR (1) BRPI0708160A2 (es)
CA (1) CA2642243A1 (es)
GB (1) GB0603782D0 (es)
MX (1) MX2008010804A (es)
RU (1) RU2008137723A (es)
WO (1) WO2007096174A1 (es)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2589383A1 (en) 2011-11-06 2013-05-08 Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. Berlin FKBP subtype-specific rapamycin analogue for use in treatment of diseases

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102268015B (zh) * 2011-08-30 2013-08-28 成都摩尔生物医药有限公司 一种依维莫司的合成方法
UY37900A (es) * 2017-09-26 2019-04-30 Novartis Ag Nuevos derivados de rapamicina
AU2019409366B2 (en) 2018-12-18 2022-10-27 Novartis Ag Rapamycin derivatives
PT3947392T (pt) * 2019-03-26 2024-05-14 Novartis Ag Derivados de rapamicina contendo 1,1-dióxido de isotiazolidina e 1,4-butano sultona e seus usos
CN113181117B (zh) * 2021-03-22 2022-08-26 沈阳药科大学 一种紫草素和蒽环类化疗药共载脂质体及其制备方法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0210101A (pt) * 2001-06-01 2004-06-08 Wyeth Corp Combinações antineoplásticas
AU2003241359A1 (en) * 2002-05-06 2003-11-11 Functional Genetics, Inc. Mammalian genes involed in rapamycin resistance and tumorgenesis: annexin xiii genes
WO2004004644A2 (en) * 2002-07-05 2004-01-15 Beth Israel Deaconess Medical Center Combination of mtor inhibitor and a tyrosine kinase inhibitor for the treatment of neoplasms
GB0217777D0 (en) * 2002-07-31 2002-09-11 Novartis Ag Organic compounds
US20060099676A1 (en) * 2002-08-15 2006-05-11 Limin Li Mammalian genes involved in rapamycin resistance and tumorgenesis: rapr6 genes
GB0327840D0 (en) * 2003-12-01 2003-12-31 Novartis Ag Organic compounds

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2589383A1 (en) 2011-11-06 2013-05-08 Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. Berlin FKBP subtype-specific rapamycin analogue for use in treatment of diseases
WO2013064703A2 (en) 2011-11-06 2013-05-10 MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. Fkbp subtype-specific rapamycin analogue for use in treatment of diseases

Also Published As

Publication number Publication date
AU2007217705A1 (en) 2007-08-30
BRPI0708160A2 (pt) 2011-05-17
GB0603782D0 (en) 2006-04-05
JP2009527520A (ja) 2009-07-30
KR20080100346A (ko) 2008-11-17
RU2008137723A (ru) 2010-03-27
EP1988894A1 (en) 2008-11-12
CN101389337A (zh) 2009-03-18
CA2642243A1 (en) 2007-08-30
WO2007096174A1 (en) 2007-08-30
US20090023768A1 (en) 2009-01-22

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal